Novel library synthesis of 3,4-disubstituted pyridin-2(1 H )-ones via cleavage of pyridine-2-oxy-7-azabenzotriazole ethers under ionic hydrogenation conditions at room temperature von Pierre, Romain, Brethon, Anne, Jacques, Sylvain A, Blond, Aurélie, Chambon, Sandrine, Talano, Sandrine, Raffin, Catherine, Musicki, Branislav, Bouix-Peter, Claire, Tomas, Loic, Ouvry, Gilles, Morgentin, Rémy, Hennequin, Laurent F, Harris, Craig S

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Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists von Ouvry, Gilles, Bouix-Peter, Claire, Ciesielski, Fabrice, Chantalat, Laurent, Christin, Olivier, Comino, Catherine, Duvert, Denis, Feret, Christophe, Harris, Craig S., Lamy, Laurent, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Pascau, Jonathan, Parnet, Véronique, Perrin, Agnès, Pierre, Romain, Polge, Gaëlle, Raffin, Catherine, Rival, Yves, Taquet, Nathalie, Thoreau, Etienne, Hennequin, Laurent F.

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Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma von Fournier, Jean-François, Bhurruth-Alcor, Yushma, Musicki, Branislav, Aubert, Jérome, Aurelly, Michèle, Bouix-Peter, Claire, Bouquet, Karinne, Chantalat, Laurent, Delorme, Marion, Drean, Bénédicte, Duvert, Gwenaelle, Fleury-Bregeot, Nicolas, Gauthier, Blanche, Grisendi, Karine, Harris, Craig S., Hennequin, Laurent F., Isabet, Tatiana, Joly, Florence, Lafitte, Guillaume, Millois, Corinne, Morgentin, Rémy, Pascau, Jonathan, Piwnica, David, Rival, Yves, Soulet, Catherine, Thoreau, Étienne, Tomas, Loïc

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Route scouting and optimization of a potent sulfoximine-based inverse agonist of RORγt von Lafitte, Guillaume, Parnet, Veronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Musicki, Branislav, Tomas, Loic, Bouix-Peter, Claire, Ouvry, Gilles, Daver, Sebastien, Arlabosse, Jean-Marie, Boiteau, Jean-Guy, Gerfaud, Thibaud, Harris, Craig S.

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Sulfoximines as potent RORγ inverse agonists von Ouvry, Gilles, Bihl, Franck, Bouix-Peter, Claire, Christin, Olivier, Defoin-Platel, Claire, Deret, Sophie, Feret, Christophe, Froude, David, Hacini-Rachinel, Feriel, Harris, Craig S., Hervouet, Catherine, Lafitte, Guillaume, Luzy, Anne-Pascale, Musicki, Branislav, Orfila, Danielle, Parnet, Veronique, Pascau, Coralie, Pascau, Jonathan, Pierre, Romain, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent F.

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A convenient one-pot synthesis of boroxoles from diboronic acid von Lafitte, Guillaume, Kunihiro, Kana, Bonneaud, Céline, Dréan, Bénédicte, Gaigne, Frédéric, Parnet, Véronique, Pierre, Romain, Raffin, Catherine, Vatinel, Rodolphe, Fournier, Jean-François, Musicki, Branislav, Ouvry, Gilles, Bouix-Peter, Claire, Tomas, Loic, Harris, Craig S.

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Synthesis and in vitro evaluation of novel highly potent coumarin inhibitors of gyrase B von Laurin, Patrick, Ferroud, Didier, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav

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Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis von Ouvry, Gilles, Atrux‐Tallau, Nicolas, Bihl, Franck, Bondu, Aline, Bouix‐Peter, Claire, Carlavan, Isabelle, Christin, Olivier, Cuadrado, Marie‐Josée, Defoin‐Platel, Claire, Deret, Sophie, Duvert, Denis, Feret, Christophe, Forissier, Mathieu, Fournier, Jean‐François, Froude, David, Hacini‐Rachinel, Fériel, Harris, Craig Steven, Hervouet, Catherine, Huguet, Hélène, Lafitte, Guillaume, Luzy, Anne‐Pascale, Musicki, Branislav, Orfila, Danielle, Ozello, Benjamin, Pascau, Coralie, Pascau, Jonathan, Parnet, Véronique, Peluchon, Guillaume, Pierre, Romain, Piwnica, David, Raffin, Catherine, Rossio, Patricia, Spiesse, Delphine, Taquet, Nathalie, Thoreau, Etienne, Vatinel, Rodolphe, Vial, Emmanuel, Hennequin, Laurent François

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Reaction of pyrrolo[1,2-c]imidazole mesomeric betaines with diphenylcyclopropenone derivatives von Musicki, Branislav

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Structure of the light emitter in krill (Euphausia pacifica) bioluminescence von Nakamura, Hideshi, Musicki, Branislav, Kishi, Yoshito, Shimomura, Osamu

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Early Development Scale-Up of a Novel CXCR Antagonist: Focus on Racemic and Stereoselective Routes of a Key Intermediate von Tabet, Samuel, Rodeville, Nicolas, Mathieu, Arnaud, Raffin, Catherine, Millois-Barbuis, Corinne, Musicki, Branislav, Muller, Franck, Gerfaud, Thibaud, Boiteau, Jean-Guy, Cardinaud, Isabelle

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Synthesis of nucleoside sulfonates and sulfones von Musicki, Branislav, Widlanski, Theodore S.

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Process Development and Good Manufacturing Practice Production of a Tyrosinase Inhibitor via Titanium-Mediated Coupling between Unprotected Resorcinols and Ketones von Gerfaud, Thibaud, Martin, Cédric, Bouquet, Karinne, Talano, Sandrine, Millois-Barbuis, Corinne, Musicki, Branislav, Boiteau, Jean-Guy, Cardinaud, Isabelle

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Noviose mimics of the coumarin inhibitors of gyrase B von Musicki, Branislav, Periers, Anne-Marie, Piombo, Laurent, Laurin, Patrick, Klich, Michel, Dupuis-Hamelin, Claudine, Lassaigne, Patrice, Bonnefoy, Alain

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Synthesis of the 4’-desmethoxy analogue of RU79115 von Musicki, Branislav, Periers, Anne-Marie, Tessot, Nicole, Klich, Michel

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Structure-activity relationship in two series of aminoalkyl substituted coumarin inhibitors of gyrase B von Laurin, Patrick, Ferroud, Didier, Schio, Laurent, Klich, Michael, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav

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Synthesis of carbohydrate sulfonates and sulfonate esters von Musicki, Branislav, Widlanski, Theodore S

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Synthesis and biological evaluation of coumarincarboxylic acids as inhibitors of gyrase B. L-rhamnose as an effective substitute for L-noviose von Ferroud, Didier, Collard, Jeannine, Klich, Michel, Dupuis-Hamelin, Claudine, Mauvais, Pascale, Lassaigne, Patrice, Bonnefoy, Alain, Musicki, Branislav

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Synthesis and 1,3-dipolar cycloaddition reactions of novel heteropentalene mesomeric betaines, pyrrolo[1,2-c]imidazole mesomeric betaines von Musicki, Branislav

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Syntheses of conformationally restricted analogues of an angiotensin II receptor antagonist. General synthetic approach to functionalized imidazo[1,5- a]pyridine derivatives von Musicki, Branislav, Vevert, Jean-Paul

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