Anti‐inflammatory activity of phosphodiesterase (PDE)‐IV inhibitors in acute and chronic models of inflammation von SEKUT, L., YARNALL, D., STIMPSON, S. A., NOEL, L. S., BATEMAN‐FITE, R., CLARK, R. L., BRACKEEN, M. F., MENIUS, J. A., CONNOLLY, K. M.

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Design and Synthesis of Conformationally Constrained Analogs of 4-(3-Butoxy-4-methoxybenzyl)imidazolidin-2-one (Ro 20-1724) as Potent Inhibitors of cAMP-Specific Phosphodiesterase von Brackeen, Marcus F, Stafford, Jeffrey A, Cowan, David J, Brown, Peter J, Domanico, Paul L, Feldman, Paul L, Rose, Dudley, Strickland, Alan B, Veal, James M, Verghese, Margrith

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Design, synthesis, and pharmacological evaluation of ultrashort- to long-acting opioid analgetics von FELDMAN, P. L, JAMES, M. K, BRACKEEN, M. F, BILOTTA, J. M, SCHUSTER, S. V, LAHEY, A. P, LUTZ, M. W, JOHNSON, M. R, LEIGHTON, H. J

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Phosphodiesterase Type IV Inhibition. Structure-Activity Relationships of 1,3-Disubstituted Pyrrolidines von Feldman, Paul L, Brackeen, Marcus F, Cowan, David J, Marron, Brian E, Schoenen, Frank J, Stafford, Jeffrey A, Suh, Edward M, Domanico, Paul L, Rose, Dudley

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Introduction of a conformational switching element on a pyrrolidine ring. Synthesis and evaluation of methyl (R,R)-(.+-.)-3-acetyl-4-[3- (cyclopentyloxy)-4-methoxyphenyl]-3- methyl... von Stafford, Jeffrey A, Veal, James M, Feldman, Paul L, Valvano, Nicole L, Baer, Philip G, Brackeen, Marcus F, Brawley, E. Sloan, Connolly, Kevin M, Domanico, Paul L

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A highly selective protocol for the deprotection of BOC-protected amides and carbamates von Stafford, Jeffrey A., Brackeen, Marcus F., Karanewsky, Donald S., Valvano, Nicole L.

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An efficient and mild synthesis of highly substituted imidazoles von Brackeen, Marcus F., Stafford, Jeffrey A., Feldman, Paul L., Karanewsky, Donald S.

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A novel route to the 4-anilido-4-(methoxycarbonyl)piperidine class of analgetics von Feldman, Paul L., Brackeen, Marcus F.

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N-(2-Benzoylphenyl)-L-tyrosine PPARgamma agonists. 1. Discovery of a novel series of potent antihyperglycemic and antihyperlipidemic agents von Henke, B R, Blanchard, S G, Brackeen, M F, Brown, K K, Cobb, J E, Collins, J L, Harrington, Jr, W W, Hashim, M A, Hull-Ryde, E A, Kaldor, I, Kliewer, S A, Lake, D H, Leesnitzer, L M, Lehmann, J M, Lenhard, J M, Orband-Miller, L A, Miller, J F, Mook, Jr, R A, Noble, S A, Oliver, Jr, W, Parks, D J, Plunket, K D, Szewczyk, J R, Willson, T M

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Identification of a Potent Human Trace Amine-Associated Receptor 1 Antagonist von Decker, Ann M, Brackeen, Marcus F, Mohammadkhani, Aida, Kormos, Chad M, Hesk, David, Borgland, Stephanie L, Blough, Bruce E

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N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic Agents von Henke, Brad R, Blanchard, Steven G, Brackeen, Marcus F, Brown, Kathleen K, Cobb, Jeff E, Collins, Jon L, Harrington, W. Wallace, Hashim, Mir A, Hull-Ryde, Emily A, Kaldor, Istvan, Kliewer, Steven A, Lake, Debra H, Leesnitzer, Lisa M, Lehmann, Jürgen M, Lenhard, James M, Orband-Miller, Lisa A, Miller, John F, Mook, Robert A, Noble, Stewart A, Oliver, William, Parks, Derek J, Plunket, Kelli D, Szewczyk, Jerzy R, Willson, Timothy M

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Conformational characteristics of the interaction of SR141716A with the CB1 cannabinoid receptor as determined through the use of conformationally constrained analogs von Thomas, Brian F, Zhang, Yanan, Brackeen, Marcus, Page, Kevin M, Mascarella, S Wayne, Seltzman, Herbert H

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Design, synthesis, and pharmacological evaluation of ultrashort- to long-acting opioid analgesics von Feldman, Paul L, James, Michael K, Brackeen, Marcus F, Bilotta, Joanne M, Schuster, Suzanne V, Lahey, Avis P, Lutz, Michael W, Johnson, M. Ross, Leighton, H. Jeff

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