11β-hydroxysteroid dehydrogenase type 1 inhibitors: a review of recent patents von Boyle, Craig D, Kowalski, Timothy J

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Synthesis of Mono- and Difluoronaphthoic Acids von Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis V, Boyle, Craig D, Kozlowski, Joseph A, Chackalamannil, Samuel, Josien, Hubert, Wang, Yuguang, Zhou, Guowei

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The discovery of azepane sulfonamides as potent 11β-HSD1 inhibitors von Neelamkavil, Santhosh F., Boyle, Craig D., Chackalamannil, Samuel, Greenlee, William J., Zhang, Lili, Terracina, Giuseppe

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Azabicyclic sulfonamides as potent 11β-HSD1 inhibitors von Shah, Unmesh, Boyle, Craig D., Chackalamannil, Samuel, Baker, Hana, Kowalski, Timothy, Lee, Julie, Terracina, Giuseppe, Zhang, Lili

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Absolute configuration at the tricarballylic acid moieties of fumonisin B2 von Boyle, Craig D, Kishi, Yoshito

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Design, synthesis, and evaluation of fused heterocyclic analogs of SCH 58261 as adenosine A2A receptor antagonists von Shah, Unmesh, Lankin, Claire M, Boyle, Craig D, Chackalamannil, Samuel, Greenlee, William J, Neustadt, Bernard R, Cohen-Williams, Mary E, Higgins, Guy A, Ng, Kwokei, Varty, Geoffrey B, Zhang, Hongtao, Lachowicz, Jean E

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Biaryl and heteroaryl derivatives of SCH 58261 as potent and selective adenosine A2A receptor antagonists von SHAH, Unmesh, BOYLE, Craig D, SHIYONG WANG, MONOPOLI, Angela, LACHOWICZ, Jean E, CHACKALAMANNIL, Samuel, NEUSTADT, Bernard R, LINDO, Neil, GREENLEE, William J, FOSTER, Carolyn, ARIK, Leyla, YING ZHAI, NG, Kwokei

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Design, synthesis, and evaluation of fused heterocyclic analogs of SCH 58261 as adenosine A2A receptor antagonists von SHAH, Unmesh, LANKIN, Claire M, HONGTAO ZHANG, LACHOWICZ, Jean E, BOYLE, Craig D, CHACKALAMANNIL, Samuel, GREENLEE, William J, NEUSTADT, Bernard R, COHEN-WILLIAMS, Mary E, HIGGINS, Guy A, NG, Kwokei, VARTY, Geoffrey B

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Optimization of purine based PDE1/PDE5 inhibitors to a potent and selective PDE5 inhibitor for the treatment of male ED von Boyle, Craig D., Xu, Ruo, Asberom, Theodros, Chackalamannil, Samuel, Clader, John W., Greenlee, William J., Guzik, Henry, Hu, Yuequing, Hu, Zhiyong, Lankin, Claire M., Pissarnitski, Dmitri A., Stamford, Andrew W., Wang, Yuguang, Skell, Jeffrey, Kurowski, Stanley, Vemulapalli, Subbarao, Palamanda, Jairam, Chintala, Madhu, Wu, Ping, Myers, Joyce, Wang, Peng

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SAR development of polycyclic guanine derivatives targeted to the discovery of a selective PDE5 inhibitor for treatment of erectile dysfunction von PISSARNITSKI, Dmitri A, ASBEROM, Theodros, PALAMANDA, Jairam, STAMFORD, Andrew W, VEMULAPALLI, Subbarao, YUGUANG WANG, PENG WANG, PING WU, RUO XU, BOYLE, Craig D, CHACKALAMANNIL, Samuel, CHINTALA, Madhu, CLADER, John W, GREENLEE, William J, YUEQING HU, KUROWSKI, Stanley, MYERS, Joyce

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Design and synthesis of xanthine analogues as potent and selective PDE5 inhibitors von Wang, Yuguang, Chackalamannil, Samuel, Hu, Zhiyong, Boyle, Craig D, Lankin, Claire M, Xia, Yan, Xu, Ruo, Asberom, Theodros, Pissarnitski, Dmitri, Stamford, Andrew W, Greenlee, William J, Skell, Jeffrey, Kurowski, Stanley, Vemulapalli, Subbarao, Palamanda, Jairam, Chintala, Madhu, Wu, Ping, Myers, Joyce, Wang, Peng

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Novel Structure Elucidation of AAL Toxin TA Backbone von Boyle, Craig D, Harmange, Jean-Christophe, Kishi, Yoshito

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Improving the Oral Efficacy of CNS Drug Candidates:  Discovery of Highly Orally Efficacious Piperidinyl Piperidine M2 Muscarinic Receptor Antagonists von Wang, Yuguang, Chackalamannil, Samuel, Hu, Zhiyong, Greenlee, William J, Clader, John, Boyle, Craig D, Kaminski, James J, Billard, William, Binch, Crosby, Gordon, Ruperto, Vilma, Duffy, Ruth A, Cohen-Williams, Mary, Coffin, Vicki L, Cox, Kathleen A, Grotz, Diane E, Lachowicz, Jean E

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Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification von BOYLE, Craig D, VICE, Susan F, COFFIN, Vicki L, COX, Kathleen A, GROTZ, Diane E, DUFFY, Ruth A, RUPERTO, Vilma, LACHOWICZ, Jean E, CAMPION, Jennifer, CHACKALAMANNIL, Samuel, LANKIN, Claire M, MCCOMBIE, Stuart W, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, WILLIAMS, Mary-Cohen

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Metabolic stabilization of benzylidene ketal M2 muscarinic receptor antagonists via halonaphthoic acid substitution von BOYLE, Craig D, CHACKALAMANNIL, Samuel, YUGUANG WANG, GUOWEI ZHOU, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, COHEN-WILLIAMS, Mary, COFFIN, Vicki L, COX, Kathleen A, GROTZ, Diane E, DUFFY, Ruth A, CLADER, John W, RUPERTO, Vilma, LACHOWICZ, Jean E, GREENLEE, William J, JOSIEN, Hubert B, KAMINSKI, James J, KOZLOWSKI, Joseph A, MCCOMBIE, Stuart W, NAZARENO, Dennis V, TAGAT, Jayaram R

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Benzylidene ketal derivatives as M2 muscarinic receptor antagonists von BOYLE, Craig D, CHACKALAMANNIL, Samuel, DUFFY, Ruth A, RUPERTO, Vilma, LACHOWICZ, Jean E, CHEN, Lian-Yong, DUGAR, Sundeep, PUSHPAVANAM, Pradeep, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, COHEN-WILLIAMS, Mary, COFFIN, Vicki L

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Azabicyclic sulfonamides as potent 11b-HSD1 inhibitors von Shah, Unmesh, Boyle, Craig D, Chackalamannil, Samuel, Baker, Hana, Kowalski, Timothy, Lee, Julie, Terracina, Giuseppe, Zhang, Lili

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11beta-hydroxysteroid dehydrogenase type 1 inhibitors: a review of recent patents von Boyle, Craig D, Kowalski, Timothy J

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Design, synthesis, and evaluation of fused heterocyclic analogs of SCH 58261 as adenosine A sub(2A) receptor antagonists von Shah, Unmesh, Lankin, Claire M, Boyle, Craig D, Chackalamannil, Samuel, Greenlee, William J, Neustadt, Bernard R, Cohen-Williams, Mary E, Higgins, Guy A, Ng, Kwokei, Varty, Geoffrey B, Zhang, Hongtao, Lachowicz, Jean E

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Orally active and selective benzylidene ketal M2 muscarinic receptor antagonists for the treatment of Alzheimer's disease von Boyle, Craig D., Lachowicz, Jean E.

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