State-dependent energetics of GABAA receptor modulators von Borghese, Cecilia M., Goldschen-Ohm, Marcel P.

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A potential cost of evolving epibatidine resistance in poison frogs von York, Julia M, Borghese, Cecilia M, George, Andrew A, Cannatella, David C, Zakon, Harold H

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Interacting amino acid replacements allow poison frogs to evolve epibatidine resistance von Tarvin, Rebecca D., Borghese, Cecilia M., Sachs, Wiebke, Santos, Juan C., Lu, Ying, O’Connell, Lauren A., Cannatella, David C., Harris, R. Adron, Zakon, Harold H.

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(+)-Catharanthine potentiates the GABAA receptor by binding to a transmembrane site at the β(+)/α(-) interface near the TM2-TM3 loop von Arias, Hugo R., Borghese, Cecilia M., Germann, Allison L., Pierce, Spencer R., Bonardi, Alessandro, Nocentini, Alessio, Gratteri, Paola, Thodati, Thanvi M., Lim, Natalie J., Harris, R. Adron, Akk, Gustav

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Modulation of α1β3γ2 GABAA receptors expressed in X. laevis oocytes using a propofol photoswitch tethered to the transmembrane helix von Borghese, Cecilia M., Wang, Hua-Yu L., McHardy, Stanton F., Messing, Robert O., Trudell, James R., Harris, R. Adron, Bertaccini, Edward J.

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Apremilast regulates acute effects of ethanol and other GABAergic drugs via protein kinase A-dependent signaling von Blednov, Yuri A., Borghese, Cecilia M., Dugan, Michael P., Pradhan, Swetak, Thodati, Thanvi M., Kichili, Nikhita R., Harris, R. Adron, Messing, Robert O.

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Modulation of α1β3γ2 GABA A receptors expressed in X. laevis oocytes using a propofol photoswitch tethered to the transmembrane helix von Borghese, Cecilia M, Wang, Hua-Yu L, McHardy, Stanton F, Messing, Robert O, Trudell, James R, Harris, R Adron, Bertaccini, Edward J

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Mutation of the inhibitory ethanol site in GABAA ρ1 receptors promotes tolerance to ethanol-induced motor incoordination von Blednov, Yuri A., Borghese, Cecilia M., Ruiz, Carlos I., Cullins, Madeline A., Da Costa, Adriana, Osterndorff-Kahanek, Elizabeth A., Homanics, Gregg E., Harris, R. Adron

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The molecular pharmacology of volatile anesthetics von Borghese, Cecilia M

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Novel Molecule Exhibiting Selective Affinity for GABAA Receptor Subtypes von Borghese, Cecilia M., Herman, Melissa, Snell, Lawrence D., Lawrence, Keri J., Lee, Hyun-Young, Backos, Donald S., Vanderlinden, Lauren A., Harris, R. Adron, Roberto, Marisa, Hoffman, Paula L., Tabakoff, Boris

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GABAA receptor transmembrane amino acids are critical for alcohol action: disulfide cross‐linking and alkyl methanethiosulfonate labeling reveal relative location of binding sites... von Borghese, Cecilia M., Hicks, Jessica A., Lapid, Daniel J., Trudell, James R., Harris, R. Adron

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GABA(A) receptor transmembrane amino acids are critical for alcohol action: disulfide cross-linking and alkyl methanethiosulfonate labeling reveal relative location of binding site... von Borghese, Cecilia M, Hicks, Jessica A, Lapid, Daniel J, Trudell, James R, Harris, R Adron

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GABAA receptors containing ρ1 subunits contribute to in vivo effects of ethanol in mice von Blednov, Yuri A, Benavidez, Jillian M, Black, Mendy, Leiter, Courtney R, Osterndorff-Kahanek, Elizabeth, Johnson, David, Borghese, Cecilia M, Hanrahan, Jane R, Johnston, Graham A R, Chebib, Mary, Harris, R Adron

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Mutation of the inhibitory ethanol site in GABA A ρ1 receptors promotes tolerance to ethanol-induced motor incoordination von Blednov, Yuri A, Borghese, Cecilia M, Ruiz, Carlos I, Cullins, Madeline A, Da Costa, Adriana, Osterndorff-Kahanek, Elizabeth A, Homanics, Gregg E, Harris, R Adron

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Studies of ethanol actions on recombinant δ-containing γ-aminobutyric acid type A receptors yield contradictory results von Borghese, Cecilia M, Harris, R. Adron

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A transmembrane amino acid in the GABAA receptor β2 subunit critical for the actions of alcohols and anesthetics von McCracken, Mandy L, Borghese, Cecilia M, Trudell, James R, Harris, R Adron

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Functional validation of virtual screening for novel agents with general anesthetic action at ligand-gated ion channels von Heusser, Stephanie A, Howard, Rebecca J, Borghese, Cecilia M, Cullins, Madeline A, Broemstrup, Torben, Lee, Ui S, Lindahl, Erik, Carlsson, Jens, Harris, R Adron

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Characterization of two mutations, M287L and Q266I, in the α1 glycine receptor subunit that modify sensitivity to alcohols von Borghese, Cecilia M, Blednov, Yuri A, Quan, Yu, Iyer, Sangeetha V, Xiong, Wei, Mihic, S John, Zhang, Li, Lovinger, David M, Trudell, James R, Homanics, Gregg E, Harris, R Adron

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Identification of an Inhibitory Alcohol Binding Site in GABAA ρ1 Receptors von Borghese, Cecilia M, Ruiz, Carlos I, Lee, Ui S, Cullins, Madeline A, Bertaccini, Edward J, Trudell, James R, Harris, R. Adron

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Effects of Acamprosate on Neuronal Receptors and Ion Channels Expressed in Xenopus Oocytes von Reilly, Matthew T., Lobo, Ingrid A., McCracken, Lindsay M., Borghese, Cecilia M., Gong, Diane, Horishita, Takafumi, Adron Harris, R.

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