Identification of a Selective Nonpeptide Antagonist of the Anaphylatoxin C3a Receptor That Demonstrates Antiinflammatory Activity in Animal Models von Ames, Robert S, Lee, Dennis, Foley, James J, Jurewicz, Anthony J, Tornetta, Mark A, Bautsch, Wilfried, Settmacher, Britta, Klos, Andreas, Erhard, Karl F, Cousins, Russell D, Sulpizio, Anthony C, Hieble, J. Paul, McCafferty, Gerald, Ward, Keith W, Adams, Jerry L, Bondinell, William E, Underwood, David C, Osborn, Ruth R, Badger, Alison M, Sarau, Henry M

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Direct design of a potent non-peptide fibrinogen receptor antagonist based on the structure and conformation of a highly constrained cyclic RGD peptide von Ku, Thomas W, Ali, Fadia E, Barton, Linda S, Bean, John W, Bondinell, William E, Burgess, Joelle L, Callahan, James F, Calvo, Raul R, Chen, Lichong

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Enantiospecific synthesis of SB 214857, a potent, orally active, nonpeptide fibrinogen receptor antagonist von Miller, William H., Ku, Thomas W., Ali, Fadia E., Bondinell, William E., Calvo, Raul R., Davis, Larry D., Erhard, Karl F., Hall, Leon B., Huffman, William F., Keenan, Richard M., Kwon, Chet, Newlander, Kenneth A., Ross, Stephen T., Samanen, James M., Takata, Dennis T., Yuan, Chuan-Kui

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Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification von Hieble, J P, Bondinell, W E, Ruffolo, Jr, R R

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Potent non-peptide fibrinogen receptor antagonists which present an alternative pharmacophore von Ku, Thomas W, Miller, William H, Bondinell, William E, Erhard, Karl F, Keenan, Richard M, Nichols, Andrew J, Peishoff, Catherine E, Samanen, James M, Wong, Angela S, Huffman, William F

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Orally Active and Potent Inhibitors of γ-Aminobutyric Acid Uptake von Ali, Fadia E, Bondinell, William E, Dandridge, Penelope A, Frazee, James S, Garvey, Eleanor, Girard, Gerald R, Kaiser, Carl, Ku, Thomas W, Lafferty, John J, Moonsammy, George I, Oh, Hye-Ja, Rush, Julia A, Setler, Paulette E, Stringer, Orum D, Venslavsky, Joseph W, Volpe, Beth W, Yunger, Libby M, Zirkle, Charles L

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Discovery of Orally Active Nonpeptide Vitronectin Receptor Antagonists Based on a 2-Benzazepine Gly-Asp Mimetic von Miller, William H, Alberts, Doreen P, Bhatnagar, Pradip K, Bondinell, William E, Callahan, James F, Calvo, Raul R, Cousins, Russell D, Erhard, Karl F, Heerding, Dirk A, Keenan, Richard M, Kwon, Chet, Manley, Peter J, Newlander, Kenneth A, Ross, Stephen T, Samanen, James M, Uzinskas, Irene N, Venslavsky, Joseph W, Yuan, Catherine C.-K, Haltiwanger, R. Curtis, Gowen, Maxine, Hwang, Shing-Mei, James, Ian E, Lark, Michael W, Rieman, David J, Stroup, George B, Azzarano, Leonard M, Salyers, Kevin L, Smith, Brian R, Ward, Keith W, Johanson, Kyung O, Huffman, William F

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The use of rabbit intestinal permeability as an in vitro assay in the search for orally active GPIIb/IIIa antagonists von Samanen, James M., Lee, Chao-Pin, Smith, Philip L., Bondinell, William E., Calvo, Raul R., Jakas, Dalia R., Newlander, Kenneth A., Parker, Michael, Uzinskas, Irene, Yellin, Tobias O., Nichols, Andrew J.

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Conformational Preferences in a Benzodiazepine Series of Potent Nonpeptide Fibrinogen Receptor Antagonists von Keenan, Richard M, Callahan, James F, Samanen, James M, Bondinell, William E, Calvo, Raul R, Chen, Lichong, DeBrosse, Charles, Eggleston, Drake S, Haltiwanger, R. Curtis, Hwang, Shing Mei, Jakas, Dalia R, Ku, Thomas W, Miller, William H, Newlander, Kenneth A, Nichols, Andrew, Parker, Michael F, Southhall, Linda S, Uzinskas, Irene, Vasko-Moser, Janice A, Venslavsky, Joseph W, Wong, Angela S, Huffman, William F

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6-(Phenylthio)-substituted 2,3,4,5-tetrahydro-1H-3-benzazepines, a novel class of dopamine receptor antagonists and neuroleptics von Kaiser, Carl, Ali, Fadia E, Bondinell, William E, Brenner, Martin, Holden, Kenneth G, Ku, Thomas W, Oh, Hye-Ja, Ross, Stephen T, Yim, Nelson C. F

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DIBENZOCYCLOHEPTENE DERIVATIVES AS VITRONECTIN RECEPTOR ANTAGONISTS, PROCESS FOR PRODUCING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von SAMANEN JAMES MARTIN SAMANEN JAMES MARTIN, MILLER WILLIAM H. MILLER WILLIAM H, HEERDING DIRK HEERDING DIRK, BONDINELL WILLIAM E. BONDINELL WILLIAM E

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Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model von Miller, William H., Bondinell, William E., Cousins, Russell D., Erhard, Karl F., Jakas, Dalia R., Keenan, Richard M., Ku, Thomas W., Newlander, Kenneth A., Ross, Stephen T., Haltiwanger, R.Curtis, Bradbeer, Jeremy, Drake, Fred H., Gowen, Maxine, Hoffman, Sandra J., Hwang, Shing-Mei, James, Ian E., Lark, Michael W., Lechowska, Beata, Rieman, David J., Stroup, George B., Vasko-Moser, Janice A., Zembryki, Denise L., Azzarano, Leonard M., Adams, Paula C., Salyers, Kevin L., Smith, Brian R., Ward, Keith W., Johanson, Kyung O., Huffaman, William F.

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Potent, Selective, Orally Active 3-Oxo-1,4-benzodiazepine GPIIb/IIIa Integrin Antagonists von Samanen, James M, Ali, Fadia E, Barton, Linda S, Bondinell, William E, Burgess, Joelle L, Callahan, James F, Calvo, Raul R, Chen, Wenting, Chen, Lichong, Erhard, Karl, Feuerstein, Giora, Heys, Richard, Hwang, Shing-Mei, Jakas, Dalia R, Keenan, Richard M, Ku, Thomas W, Kwon, Chet, Lee, Chao-Pin, Miller, William H, Newlander, Kenneth A, Nichols, Andrew, Parker, Michael, Peishoff, Catherine E, Rhodes, Gerald, Ross, Steven, Shu, Arthur, Simpson, Richard, Takata, Dennis, Yellin, Tobias O, Uzsinskas, Irene, Venslavsky, Joseph W, Yuan, Chuan-Kui, Huffman, William F

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Orally bioavailable nonpeptide vitronectin receptor antagonists containing 2-aminopyridine arginine mimetics von Keenan, Richard M., Miller, William H., Barton, Linda S., Bondinell, William E., Cousins, Russell D., Eppley, Daniel F., Hwang, Shing-Mei, Kwon, Chet, Lago, M.Amparo, Nguyen, Thomas T., Smith, Brian R., Uzinskas, Irene N., Yuan, Catherine C.K.

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Benzimidazole derivatives as arginine mimetics in 1,4-benzodiazepine nonpeptide vitronectin receptor (αvβ3) antagonists von Keenan, Richard M., Miller, William H., Lago, M.Amparo, Ali, Fadia E., Bondinell, William E., Callahan, James F., Calvo, Raul R., Cousins, Russell D., Hwang, Shing-Mei, Jakas, Dalia R., Ku, Thomas W., Kwon, Chet, Nguyen, Thomas T., Reader, Valerie A., Rieman, David J., Ross, Steven T., Takata, Dennis T., Uzinskas, Irene N., Yuan, Catherine C.K., Smith, Brian R.

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Tetrahydro thiadiazolo isoquinolines: synthesis and inhibition of phenylethanolamine-N-methyltransferase von Girard, Gerald R, Bondinell, William E, Hillegass, Leonard M, Holden, Kenneth G, Pendleton, Robert G, Uzinskas, Irene

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Carcinogenicity of Methylchrysenes von Hoffmann, Dietrich, Bondinell, William E., Wynder, Ernst L.

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Antagonista de receptor vitronectina von WILLIAM E. BONDINELL

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Inhibitors of phenylethanolamine N-methyltransferase and epinephrine biosynthesis. 1. Chloro-Substituted 1,2,3,4-tetrahydroisoquinolines von Bondinell, William E, Chapin, Frederic W, Girard, Gerald R, Kaiser, Carl, Krog, Arnold J, Pavloff, Alex M, Schwartz, Mark S, Silvestri, Joanne S, Vaidya, Praful D

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Stereochemical studies of the pyruvate kinase reaction with (Z)- and (E)-phosphoenol-α-ketobutyrate von Adlersberg, Mella, Dayan, Jean, Bondinell, William E, Sprinson, David B

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