Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer von Lücking, Ulrich, Kosemund, Dirk, Böhnke, Niels, Lienau, Philip, Siemeister, Gerhard, Denner, Karsten, Bohlmann, Rolf, Briem, Hans, Terebesi, Ildiko, Bömer, Ulf, Schäfer, Martina, Ince, Stuart, Mumberg, Dominik, Scholz, Arne, Izumi, Raquel, Hwang, Stuart, von Nussbaum, Franz

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A Novel NAMPT Inhibitor-Based Antibody–Drug Conjugate Payload Class for Cancer Therapy von Böhnke, Niels, Berger, Markus, Griebenow, Nils, Rottmann, Antje, Erkelenz, Michael, Hammer, Stefanie, Berndt, Sandra, Günther, Judith, Wengner, Antje M., Stelte-Ludwig, Beatrix, Mahlert, Christoph, Greven, Simone, Dietz, Lisa, Jörißen, Hannah, Barak, Naomi, Bömer, Ulf, Hillig, Roman C., Eberspaecher, Uwe, Weiske, Jörg, Giese, Anja, Mumberg, Dominik, Nising, Carl Friedrich, Weinmann, Hilmar, Sommer, Anette

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Radiofluorinated Derivatives of 2‑(Phosphonomethyl)pentanedioic Acid as Inhibitors of Prostate Specific Membrane Antigen (PSMA) for the Imaging of Prostate Cancer von Graham, Keith, Lesche, Ralf, Gromov, Alexey V, Böhnke, Niels, Schäfer, Martina, Hassfeld, Jorma, Dinkelborg, Ludger, Kettschau, Georg

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Discovery of Rigidified ?,?-Unsaturated Imines as New Resistance-breaking Insecticides for Malaria Vector Control von Arlt, Alexander, Böhnke, Niels, Horstmann, Sebastian, Vermeer, Arnoldus W. P., Werner, Stefan, Velten, Robert

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Discovery of potent SOS1 inhibitors that block RAS activation via disruption of the RAS–SOS1 interaction von Hillig, Roman C., Sautier, Brice, Schroeder, Jens, Moosmayer, Dieter, Hilpmann, André, Stegmanna, Christian M., Werbeck, Nicolas D., Briem, Hans, Boemer, Ulf, Weiske, Joerg, Badock, Volker, Mastouri, Julia, Petersen, Kirstin, Siemeister, Gerhard, Kahmann, Jan D., Wegener, Dennis, Böhnke, Niels, Eis, Knut, Graham, Keith, Wortmann, Lars, von Nussbaum, Franz, Bader, Benjamin

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Preclinical evaluation of BAY 1075553, a novel super(18)F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer von Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V, Bohnke, Niels, Borkowski, Sandra, Monning, Ursula, Hegele-Hartung, Christa, Dohr, Olaf, Dinkelborg, Ludger M, Graham, Keith

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Mono- and multimeric PSMA-targeting small molecule-thorium-227 conjugates for optimized efficacy and biodistribution in preclinical models von Böhnke, Niels, Indrevoll, Bård, Hammer, Stefanie, Papple, Alex, Kristian, Alexander, Briem, Hans, Celik, Arif, Mumberg, Dominik, Cuthbertson, Alan, Zitzmann-Kolbe, Sabine

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Preparation of (2R)-2-acetoxy-D-forosamine for the total synthesis of spinosyns von Tietze, Lutz F., Böhnke, Niels, Brasche, Gordon

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Abstract 2907: Identification and optimization of a novel NAMPT inhibitor-based ADC payload class for cancer therapy von Böhnke, Niels, Berger, Markus, Griebenow, Nils, Giese, Anja, Günther, Judith, Sommer, Anette, Hammer, Stefanie, Berndt, Sandra, Wengner, Antje M., Beier, Rudolf, Stelte-Ludwig, Beatrix, Mahlert, Christoph, Greven, Simone, Dietz, Lisa, Joerissen, Hannah, Rottmann, Antje, Erkelenz, Michael, Barak, Naomi, Bömer, Ulf, Mumber, Dominik, Kreft, Bertolt, Linden, Lars, Nising, Carl Friedrich, Weinmann, Hilmar

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Preclinical evaluation of BAY 1075553, a novel 18F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer von Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V., Böhnke, Niels, Borkowski, Sandra, Mönning, Ursula, Hegele-Hartung, Christa, Döhr, Olaf, Dinkelborg, Ludger M., Graham, Keith

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Preclinical evaluation of BAY 1075553, a novel (18)F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer von Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V, Böhnke, Niels, Borkowski, Sandra, Mönning, Ursula, Hegele-Hartung, Christa, Döhr, Olaf, Dinkelborg, Ludger M, Graham, Keith

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Three-Component Domino Knoevenagel/Hetero-Diels-Alder Reaction for the Synthesis of the Amino Sugars 2-Acetoxyforosamine and 2-Acetoxyossamine - Experimental and Theoretical Result... von Tietze, Lutz F., Dietz, Simone, Böhnke, Niels, Düfert, M. Alexander, Objartel, Ina, Stalke, Dietmar

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Discovery of Rigidified α,β-Unsaturated Imines as New Resistance-breaking Insecticides for Malaria Vector Control von Arlt, Alexander, Böhnke, Niels, Horstmann, Sebastian, Vermeer, Arnoldus W P, Werner, Stefan, Velten, Robert

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Targeted radiopharmaceuticals for the diagnosis and treatment of cancer von BOHNKE, NIELS, CUTHBERTSON, ALAN

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Synthesis of Novel Spinosyn A Analogues by Pd-Mediated Transformations von Tietze, Lutz F., Brasche, Gordon, Grube, Alexander, Böhnke, Niels, Stadler, Christian

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Synthesis of Enantiomerically Pure Cyclopentene Building Blocks von Tietze, Lutz F., Stadler, Christian, Böhnke, Niels, Brasche, Gordon, Grube, Alexander

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Preclinical evaluation of BAY 1075553, a novel ^sup 18^F-labelled inhibitor of prostate-specific membrane antigen for PET imaging of prostate cancer von Lesche, Ralf, Kettschau, Georg, Gromov, Alexey V, Böhnke, Niels, Borkowski, Sandra, Mönning, Ursula, Hegele-hartung, Christa, Döhr, Olaf, Dinkelborg, Ludger M, Graham, Keith

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2-((2-(PHENYLOXYMETHYL)PYRIDIN-5-YL)OXY)-ETHANAMIN-DERIVATIVES AND RELATED COMPOUNDS AS PESTICIDES E.G. FOR CROP PROTECTION von GORGENS Ulrich, ILG Kerstin, TURBERG Andreas, VERMEER Arnoldus, HORN Karin, HORSTMANN Sebastian, PORTZ Daniela, VELTEN Robert, ARLT Alexander, BOHNKE Niels

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Multiple Palladium-Catalyzed Reactions for the Synthesis of Analogues of the Highly Potent Insecticide Spinosyn A von Tietze, Lutz F., Brasche, Gordon, Stadler, Christian, Grube, Alexander, Böhnke, Niels

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2-Methyl-Quinazolines von SCHRODER, Jens, WORTMANN, Lars, SAUTIER, Brice, BOHNKE, Niels, BADER, Benjamin, PETERSEN, Kirstin, MOOSMAYER, Dieter, WANG, Qiuwen, VON NUSSBAUM, Franz, WENGNER, Antje Margret, LIENAU, Philip, SCHICK, Hans, BRIEM, Hans, HILLIG, Roman, EIS, Knut

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