Organic synthesis provides opportunities to transform drug discovery von Blakemore, David C., Castro, Luis, Churcher, Ian, Rees, David C., Thomas, Andrew W., Wilson, David M., Wood, Anthony

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Modern advances in heterocyclic chemistry in drug discovery von Taylor, Alexandria P, Robinson, Ralph P, Fobian, Yvette M, Blakemore, David C, Jones, Lyn H, Fadeyi, Olugbeminiyi

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Site-selective Suzuki-Miyaura coupling of heteroaryl halides - understanding the trends for pharmaceutically important classes von Almond-Thynne, Joshua, Blakemore, David C, Pryde, David C, Spivey, Alan C

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Heterocyclic Allylsulfones as Latent Heteroaryl Nucleophiles in Palladium-Catalyzed Cross-Coupling Reactions von Markovic, Tim, Murray, Philip R. D, Rocke, Benjamin N, Shavnya, Andre, Blakemore, David C, Willis, Michael C

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One-Pot Synthesis of Sulfonamides from Unactivated Acids and Amines via Aromatic Decarboxylative Halosulfonylation von Pedersen, P. Scott, Blakemore, David C., Chinigo, Gary M., Knauber, Thomas, MacMillan, David W. C.

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Decarboxylative Borylation and Cross-Coupling of (Hetero)aryl Acids Enabled by Copper Charge Transfer Catalysis von Dow, Nathan W, Pedersen, P. Scott, Chen, Tiffany Q, Blakemore, David C, Dechert-Schmitt, Anne-Marie, Knauber, Thomas, MacMillan, David W. C

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A Unified Approach to Decarboxylative Halogenation of (Hetero)aryl Carboxylic Acids von Chen, Tiffany Q., Pedersen, P. Scott, Dow, Nathan W., Fayad, Remi, Hauke, Cory E., Rosko, Michael C., Danilov, Evgeny O., Blakemore, David C., Dechert-Schmitt, Anne-Marie, Knauber, Thomas, Castellano, Felix N., MacMillan, David W. C.

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Iterative reactions of transient boronic acids enable sequential C–C bond formation von Battilocchio, Claudio, Feist, Florian, Hafner, Andreas, Simon, Meike, Tran, Duc N., Allwood, Daniel M., Blakemore, David C., Ley, Steven V.

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Three-Component Assembly of Multiply Substituted Homoallylic Alcohols and Amines Using a Flow Chemistry Photoreactor von Chen, Yiding, Blakemore, David C, Pasau, Patrick, Ley, Steven V

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One-pot three-component sulfone synthesis exploiting palladium-catalysed aryl halide aminosulfonylation von Richards-Taylor, Charlotte S, Blakemore, David C, Willis, Michael C

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Fluorodecarboxylation for the Synthesis of Trifluoromethyl Aryl Ethers von Zhang, Qing-Wei, Brusoe, Andrew T., Mascitti, Vincent, Hesp, Kevin D., Blakemore, David C., Kohrt, Jeffrey T., Hartwig, John F.

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Catalyst Selection Facilitates the Use of Heterocyclic Sulfinates as General Nucleophilic Coupling Partners in Palladium-Catalyzed Coupling Reactions von Markovic, Tim, Rocke, Benjamin N., Blakemore, David C., Mascitti, Vincent, Willis, Michael C.

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Pyridine sulfinates as general nucleophilic coupling partners in palladium-catalyzed cross-coupling reactions with aryl halides von Markovic, Tim, Rocke, Benjamin N, Blakemore, David C, Mascitti, Vincent, Willis, Michael C

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Photoredox Generation of Sulfonyl Radicals and Coupling with Electron Deficient Olefins von Chen, Yiding, McNamara, Nicole, May, Oliver, Pillaiyar, Thanigaimalai, Blakemore, David C, Ley, Steven V

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Redefining the Synthetic Logic of Medicinal Chemistry. Photoredox-Catalyzed Reactions as a General Tool for Aliphatic Core Functionalization von Fernández, David F., González-Esguevillas, María, Keess, Sebastian, Schäfer, Felix, Mohr, Jens, Shavnya, Andre, Knauber, Thomas, Blakemore, David C., MacMillan, David W. C.

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Selection of a novel anti-nicotine vaccine: influence of antigen design on antibody function in mice von Pryde, David C, Jones, Lyn H, Gervais, David P, Stead, David R, Blakemore, David C, Selby, Matthew D, Brown, Alan D, Coe, Jotham W, Badland, Matthew, Beal, David M, Glen, Rebecca, Wharton, Yvonne, Miller, Gavin J, White, Phil, Zhang, Ningli, Benoit, Michelle, Robertson, Karen, Merson, James R, Davis, Heather L, McCluskie, Michael J

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A Photoredox Coupling Reaction of Benzylboronic Esters and Carbonyl Compounds in Batch and Flow von Chen, Yiding, May, Oliver, Blakemore, David C, Ley, Steven V

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Decarbonylative Pd-Catalyzed Suzuki Cross-Coupling for the Synthesis of Structurally Diverse Heterobiaryls von Cervantes-Reyes, Alejandro, Smith, Aaron C, Chinigo, Gary M, Blakemore, David C, Szostak, Michal

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Reductant‐Free Cross‐Electrophile Synthesis of Di(hetero)arylmethanes by Palladium‐Catalyzed Desulfinative C−C Coupling von McKnight, Janette, Shavnya, Andre, Sach, Neal W., Blakemore, David C., Moses, Ian B., Willis, Michael C.

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Synthesis of 3‑Substituted 2‑Arylpyridines via Cu/Pd-Catalyzed Decarboxylative Cross-Coupling of Picolinic Acids with (Hetero)Aryl Halides von Hackenberger, Dagmar, Weber, Philip, Blakemore, David C, Goossen, Lukas J

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