Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology von Blagg, Julian, Workman, Paul

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Anticancer Inhibitors of Hsp90 Function: Beyond the Usual Suspects von Garg, Gaurav, Khandelwal, Anuj, Blagg, Brian S J

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Recent advances toward the development of Hsp90 C-terminal inhibitors von Amatya, Eva, Blagg, Brian S.J.

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Magnetic relaxation pathways in lanthanide single-molecule magnets von Blagg, Robin J., Ungur, Liviu, Tuna, Floriana, Speak, James, Comar, Priyanka, Collison, David, Wernsdorfer, Wolfgang, McInnes, Eric J. L., Chibotaru, Liviu F., Winpenny, Richard E. P.

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Development of Phenyl Cyclohexylcarboxamides as a Novel Class of Hsp90 C‐terminal Inhibitors von Garg, Gaurav, Forsberg, Leah K, Zhao, Huiping, Blagg, Brian S. J

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The role and therapeutic potential of Hsp90, Hsp70, and smaller heat shock proteins in peripheral and central neuropathies von Chaudhury, Subhabrata, Keegan, Bradley M., Blagg, Brian S. J.

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The Development of Hsp90β-Selective Inhibitors to Overcome Detriments Associated with pan-Hsp90 Inhibition von Mishra, Sanket J, Liu, Weiya, Beebe, Kristin, Banerjee, Monimoy, Kent, Caitlin N, Munthali, Vitumbiko, Koren, John, Taylor, John A, Neckers, Leonard M, Holzbeierlein, Jeffrey, Blagg, Brian S. J

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Investigation of the site 2 pocket of Grp94 with KUNG65 benzamide derivatives von Pugh, Kyler, Xu, Hao, Blagg, Brian S.J.

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The disruption of protein−protein interactions with co-chaperones and client substrates as a strategy towards Hsp90 inhibition von Serwetnyk, Michael A., Blagg, Brian S.J.

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A first-in-class Polymerase Theta Inhibitor selectively targets Homologous-Recombination-Deficient Tumors von Zhou, Jia, Gelot, Camille, Pantelidou, Constantia, Li, Adam, Yücel, Hatice, Davis, Rachel E, Färkkilä, Anniina, Kochupurakkal, Bose, Syed, Aleem, Shapiro, Geoffrey I, Tainer, John A, Blagg, Brian S J, Ceccaldi, Raphael, D'Andrea, Alan D

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Structure-guided design of an Hsp90β N-terminal isoform-selective inhibitor von Khandelwal, Anuj, Kent, Caitlin N., Balch, Maurie, Peng, Shuxia, Mishra, Sanket J., Deng, Junpeng, Day, Victor W., Liu, Weiya, Subramanian, Chitra, Cohen, Mark, Holzbeierlein, Jeffery M., Matts, Robert, Blagg, Brian S. J.

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Novel C-Terminal Heat Shock Protein 90 Inhibitors (KU711 and Ku757) Are Effective in Targeting Head and Neck Squamous Cell Carcinoma Cancer Stem cells von Subramanian, C., Kovatch, K.J., Sim, M.W., Wang, G., Prince, M.E., Carey, T.E., Davis, R., Blagg, B.S.J., Cohen, M.S.

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Engineering an Antibiotic to Fight Cancer: Optimization of the Novobiocin Scaffold to Produce Anti-proliferative Agents von Zhao, Huiping, Donnelly, Alison C, Kusuma, Bhaskar R, Brandt, Gary E. L, Brown, Douglas, Rajewski, Roger A, Vielhauer, George, Holzbeierlein, Jeffrey, Cohen, Mark S, Blagg, Brian S. J

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Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding von Que, Nanette L. S, Crowley, Vincent M, Duerfeldt, Adam S, Zhao, Jinbo, Kent, Caitlin N, Blagg, Brian S. J, Gewirth, Daniel T

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Natural products and other inhibitors of F1FO ATP synthase von Patel, Bhargav A., D’Amico, Terin L., Blagg, Brian S.J.

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Extracellular heat shock protein 90 alpha (eHsp90α)'s role in cancer progression and the development of therapeutic strategies von Reynolds, Tyelor S., Blagg, Brian S.J.

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The heat shock response and small molecule regulators von Kurop, Margaret K., Huyen, Cormac M., Kelly, John H., Blagg, Brian S.J.

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Natural Product Inspired N-Terminal Hsp90 Inhibitors: From Bench to Bedside? von Khandelwal, Anuj, Crowley, Vincent M., Blagg, Brian S. J.

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Hsp90 activator Aha1 drives production of pathological tau aggregates von Shelton, Lindsey B., Baker, Jeremy D., Zheng, Dali, Sullivan, Leia E., Solanki, Parth K., Webster, Jack M., Sun, Zheying, Sabbagh, Jonathan J., Nordhues, Bryce A., Koren, John, Ghosh, Suman, Blagg, Brian S. J., Blair, Laura J., Dickey, Chad A.

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Synthesis and Biological Evaluation of Novobiocin Core Analogues as Hsp90 Inhibitors von Byrd, Katherine M., Subramanian, Chitra, Sanchez, Jacqueline, Motiwala, Hashim F., Liu, Weiya, Cohen, Mark S., Holzbeierlein, Jeffrey, Blagg, Brian S. J.

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