A model for interfacial activation in lipases from the structure of a fungal lipase-inhibitor complex von Brzozowski, A. M, Derewenda, U, Derewenda, Z. S, Dodson, G. G, Lawson, D. M, Turkenburg, J. P, Bjorkling, F, Huge-Jensen, B, Patkar, S. A, Thim, L

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Anticancer agent CHS-828 inhibits cellular synthesis of NAD von Olesen, Uffe Høgh, Christensen, Mette Knak, Björkling, Fredrik, Jäättelä, Marja, Jensen, Peter Buhl, Sehested, Maxwell, Nielsen, Søren Jensby

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Evaluation of the topoisomerase II-inactive bisdioxopiperazine ICRF-161 as a protectant against doxorubicin-induced cardiomyopathy von Martin, Elke, Thougaard, Annemette Vinding, Grauslund, Morten, Jensen, Peter B, Bjorkling, Fredrik, Hasinoff, Brian B, Tjørnelund, Jette, Sehested, Maxwell, Jensen, Lars H

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Rapid Synthesis of Aryl Azides from Aryl Halides under Mild Conditions von Andersen, Jacob, Madsen, Ulf, Björkling, Fredrik, Liang, Xifu

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Synthesis and Conformational Analysis of Fusidic Acid Side Chain Derivatives in Relation to Antibacterial Activity von Duvold, Tore, Sørensen, Morten Dahl, Björkling, Fredrik, Henriksen, Anne S, Rastrup-Andersen, Niels

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Lipase catalyzed synthesis of peroxycarboxylic acids and lipase mediated oxidations von Björkling, Fredrik, Frykman, Hans, Godtfredsen, Sven Erik, Kirk, Ole

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Early stimulation of acidification rate by novel cytotoxic pyridyl cyanoguanidines in human tumor cells: comparison with m-Iodobenzylguanidine von Ekelund, Sara, Liminga, Gunnar, Björkling, Fredrik, Ottosen, Erik, Schou, Charlotte, Binderup, Lise, Larsson, Rolf

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Novel cyanoguanidines with potent oral antitumour activity von Schou, Charlotte, Ottosen, Erik R., Petersen, Hans Jørgen, Björkling, Fredrik, Latini, Scilla, Hjarnaa, Pernille V., Bramm, Erik, Binderup, Lise

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NEW ESTERS OF SUCCINIC ACID AND MIXED MOLECULES FORMED BY SUCH ESTERS AND A MEGLITINIDE ANALOG: STUDY OF THEIR INSULINOTROPIC POTENTIAL von LAGHMICH, A., LADRIERE, L., DANNACHER, H., BJORKLING, F., MALAISSE, W.J.

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Recombinant Human PPAR-β/δ Ligand-binding Domain is Locked in an Activated Conformation by Endogenous Fatty Acids von Fyffe, Stewart A., Alphey, Magnus S., Buetow, Lori, Smith, Terry K., Ferguson, Michael A.J., Sørensen, Morten D., Björkling, Fredrik, Hunter, William N.

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Synthesis and Structure−Activity Relationship of Aminobenzophenones. A Novel Class of p38 MAP Kinase Inhibitors with High Antiinflammatory Activity von Ottosen, Erik Rytter, Sørensen, Morten Dahl, Björkling, Fredrik, Skak-Nielsen, Tine, Fjording, Marianne Scheel, Aaes, Helle, Binderup, Lise

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Switched enantiopreference of Humicola lipase for 2-phenoxyalkanoic acid ester homologs can be rationalized by different substrate binding modes von Berglund, Per, Vallikivi, Imre, Fransson, Linda, Dannacher, Heinz, Holmquist, Mats, Martinelle, Mats, Björkling, Fredrik, Parve, Omar, Hult, Karl

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EB1627: a soluble prodrug of the potent anticancer cyanoguanidine CHS828 von Binderup, Ernst, Björkling, Fredrik, Hjarnaa, Pernille Vig, Latini, Scilla, Baltzer, Bodil, Carlsen, Morten, Binderup, Lise

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Studies on the Interaction between the Vitamin D Receptor and the Radiolabelled 20-epi Vitamin D Analogue GS 1500 von Mathiasen, I.S., Grue-Sørensen, G., Hansen, C.Mørk, Binderup, L., Björkling, F.

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Metabolism of glycerol-1,2,3-trimethylsuccinate in rat hepatocytes von Ladrière, L, Grue-Sørensen, G, Björkling, F, Malaisse, W J

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Cyclic phosphinamides and phosphonamides, novel series of potent matrix metalloproteinase inhibitors with antitumour activity von Sørensen, Morten Dahl, Blæhr, Lars K.A., Christensen, Mette K., Høyer, Thomas, Latini, Scilla, Hjarnaa, Pernille-Julia V., Björkling, Fredrik

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In Vivo Stimulation of Insulin Secretion by Novel Esters of Succinic Acid von Zhang, T.-M., Björkling, F., Malaisse, W. J.

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Improved viability and metabolic behavior of hepatocytes after liver storage in the presence of a succinic acid ester von LADRIERE, L, MERCAN, D, BJÖRKLING, F, MALAISSE, W. J

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Structural variants of the vitamin D analogue EB1089 reduce its ligand sensitivity and promoter selectivity von Quack, Marcus, Clarin, Andreas, Binderup, Ernst, Björkling, Fredrik, Hansen, Christina Mørk, Carlberg, Carsten

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Metabolism of [1,3-13C]glycerol-1,2,3-tris(methylsuccinate) and glycerol-1,2,3-tris(methyl[2,3-13C]succinate) in rat hepatocytes von MALAISSE, W. J, LADRIERE, L, VERBRUGGEN, I, GRUE-SØRENSON, G, BJÖRKLING, F, WILLEM, R

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