Evaluation of 1H‑Triazole-1‑[N,N′‑Bis(tert-butoxycarbonyl)]carboxamidine in Solution-Phase and On-Resin Guanidinylation von Wester, Anita, Björkling, Fredrik, Franzyk, Henrik

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Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment von Wróbel, Tomasz M., Jørgensen, Flemming Steen, Pandey, Amit V., Grudzińska, Angelika, Sharma, Katyayani, Yakubu, Jibira, Björkling, Fredrik

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Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids von Jørgensen, Johan Storm, Mood, Elnaz Harifi, Knap, Anne Sofie Holst, Nielsen, Simone Eidnes, Nielsen, Peter E., Żabicka, Dorota, Matias, Carina, Domraceva, Ilona, Björkling, Fredrik, Franzyk, Henrik

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Peptide/Peptoid Hybrid Oligomers: The Influence of Hydrophobicity and Relative Side-Chain Length on Antibacterial Activity and Cell Selectivity von Frederiksen, Nicki, Hansen, Paul R, Björkling, Fredrik, Franzyk, Henrik

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Optimized Synthesis of Fmoc/Boc‐Protected PNA Monomers and their Assembly into PNA Oligomers von Shaikh, Ashif Y., Björkling, Fredrik, Nielsen, Peter E., Franzyk, Henrik

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Selected strategies to fight pathogenic bacteria von Plotniece, Aiva, Sobolev, Arkadij, Supuran, Claudiu T., Carta, Fabrizio, Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, Jari, Augustyns, Koen, Cos, Paul, De Vooght, Linda, Govaerts, Matthias, Aizawa, Juliana, Tammela, Päivi, Žalubovskis, Raivis

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Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues von Shaikh, Ashif Y., Björkling, Fredrik, Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Domraceva, Ilona, Kreicberga, Agrita, Franzyk, Henrik

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Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties von Frederiksen, Nicki, Louka, Stavroula, Mudaliar, Chirag, Domraceva, Ilona, Kreicberga, Agrita, Pugovics, Osvalds, Żabicka, Dorota, Tomczak, Magdalena, Wygoda, Weronika, Björkling, Fredrik, Franzyk, Henrik

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Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET von Munk Jensen, Mette, Erichsen, Kamille Dumong, Björkling, Fredrik, Madsen, Jacob, Jensen, Peter Buhl, Sehested, Maxwell, Højgaard, Liselotte, Kjær, Andreas

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Microwave-assisted solid-phase synthesis of antisense acpP peptide nucleic acid-peptide conjugates active against colistin- and tigecycline-resistant E. coli and K. pneumoniae von Hansen, Anna Mette, Bonke, Gitte, Hogendorf, Wouter Frederik Johan, Björkling, Fredrik, Nielsen, John, Kongstad, Kenneth T., Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Nielsen, Peter E., Franzyk, Henrik

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Synthesis and Antitumor Effect in Vitro and in Vivo of Substituted 1,3-Dihydroindole-2-ones von Christensen, Mette K, Erichsen, Kamille D, Trojel-Hansen, Christina, Tjørnelund, Jette, Nielsen, Søren J, Frydenvang, Karla, Johansen, Tommy N, Nielsen, Birgitte, Sehested, Maxwell, Jensen, Peter B, Ikaunieks, Martins, Zaichenko, Andrei, Loza, Einars, Kalvinsh, Ivars, Björkling, Fredrik

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Nicotinamide Phosphoribosyltransferase Inhibitors, Design, Preparation, and Structure–Activity Relationship von Christensen, Mette K, Erichsen, Kamille D, Olesen, Uffe H, Tjørnelund, Jette, Fristrup, Peter, Thougaard, Annemette, Nielsen, Søren Jensby, Sehested, Maxwell, Jensen, Peter B, Loza, Einars, Kalvinsh, Ivars, Garten, Antje, Kiess, Wieland, Björkling, Fredrik

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Rapid Synthesis of Aryl Azides from Aryl Halides under Mild Conditions von Andersen, Jacob, Madsen, Ulf, Björkling, Fredrik, Liang, Xifu

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Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents von Craig, Alexander J., Ermolovich, Yuri, Cameron, Alan, Rodler, Agnes, Wang, Helen, Hawkes, Jeffrey A., Hubert, Madlen, Björkling, Fredrik, Molchanova, Natalia, Brimble, Margaret A., Moodie, Lindon W. K., Svenson, Johan

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Triphenylcarbenium Tetrafluoroborate as an Efficient Catalyst in the Regioselective Reductive Ring Opening of Benzylidene Acetals of Carbohydrates von Thota, Niranjan, Björkling, Fredrik, Kankala, Shravankumar

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Synthesis and Structure-Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents von Wróbel, Tomasz M, Rogova, Oksana, Sharma, Katyayani, Rojas Velazquez, Maria Natalia, Pandey, Amit V, Jørgensen, Flemming Steen, Arendrup, Frederic S, Andersen, Kasper L, Björkling, Fredrik

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Discovery of Novel Non-Steroidal Cytochrome P450 17A1 Inhibitors as Potential Prostate Cancer Agents von Wróbel, Tomasz M, Rogova, Oksana, Andersen, Kasper L, Yadav, Rahul, Brixius-Anderko, Simone, Scott, Emily E, Olsen, Lars, Jørgensen, Flemming Steen, Björkling, Fredrik

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[18F]FLT and [18F]FDG PET for non-invasive treatment monitoring of the nicotinamide phosphoribosyltransferase inhibitor APO866 in human xenografts von Jensen, Mette Munk, Erichsen, Kamille Dumong, Johnbeck, Camilla Bardram, Björkling, Fredrik, Madsen, Jacob, Bzorek, Michael, Jensen, Peter Buhl, Højgaard, Liselotte, Sehested, Maxwell, Kjær, Andreas

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Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139 von Shehata, Mohamed A., Nøhr, Anne C., Lissa, Delphine, Bisig, Christoph, Isberg, Vignir, Andersen, Kirsten B., Harpsøe, Kasper, Björkling, Fredrik, Bräuner-Osborne, Hans, Gloriam, David E.

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