Rational Design of a Triple Helix-Specific Intercalating Ligand von Escude, Christophe, Nguyen, Chi Hung, Kukreti, Shrikant, Janin, Yves, Sun, Jian-Sheng, Bisagni, Emile, Garestier, Therese, Helene, Claude

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Synthesis and evaluation of new 6-amino- substituted benzo[c]phenanthridine derivatives von Janin, Yves L, Croisy, Alain, Riou, Jean Francois, Bisagni, Emile

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In vitro cytotoxicity of s16020-2, a new olivacine derivative von LEONCE, S, PEREZ, V, CASABIANCA-PIGNEDE, M.-R, ANSTETT, M, BISAGNI, E, PIERRE, A, ATASSI, G

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Synthesis and Evaluation of 9-Hydroxy-5-methyl- (and 5,6-dimethyl)-6H-pyrido[4,3-b]carbazole-1-N-[(dialkylamino)alkyl]carboxamides, a New Promising Series of Antitumor Olivacine De... von Jaszfold-Howorko, Richard, Landras, Corinne, Pierre, Alain, Atassi, Ghanem, Guilbaud, Nicolas, Kraus-Berthier, Laurence, Leonce, Stephane, Rolland, Yves, Prost, Jean-Francois, Bisagni, Emile

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Diphenyl quinolines and isoquinolines: synthesis and primary biological evaluation von Croisy-Delcey, M, Croisy, A, Carrez, D, Huel, C, Chiaroni, A, Ducrot, P, Bisagni, E, Jin, L, Leclercq, G

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4-Benzyl and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones:  In Vitro Evaluation of New C-3-Amino-Substituted and C-5,6-Alkyl-Substituted Analogues against Clinically Important HIV M... von Benjahad, Abdellah, Croisy, Martine, Monneret, Claude, Bisagni, Emile, Mabire, Dominique, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Guillemont, Jérôme, Meyer, Christophe, Andries, Koen, Pauwels, Rudi, de Béthune, Marie-Pierre, Himmel, Daniel M, Das, Kalyan, Arnold, Eddy, Nguyen, Chi Hung, Grierson, David S

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Triple-Helix Directed Cleavage of Double-Stranded DNA by Benzoquinoquinoxaline-1,10-phenanthroline Conjugates von Zaid, Ahmed, Sun, Jian-Sheng, Nguyen, Chi-Hung, Bisagni, Emile, Garestier, Thérèse, Grierson, David S, Zain, Rula

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Synthesis of 9-O-Substituted Derivatives of 9-Hydroxy-5,6-dimethyl-6H- pyrido[4,3-b]carbazole-1-carboxylic Acid (2-(Dimethylamino)ethyl)amide and Their 10- and 11-Methyl Analogues... von Guillonneau, Claude, Pierré, Alain, Charton, Yves, Guilbaud, Nicolas, Kraus-Berthier, Laurence, Léonce, Stéphane, Michel, André, Bisagni, Emile, Atassi, Ghanem

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Synthesis and Biological Evaluation of 6-(9-Hydroxy-5-methyl (and 5, 6-Dimethyl)-6H-pyrido[4, 3-b]carbazol-1-yl)picolinic Amides as New Olivacine Derivatives von LANDRAS, Corinne, JASZTOLD-HOWORKO, Richard, PIERRE, Alain, LEONCE, Stephane, GUILBAUD, Nicolas, KRAUS-BERTHIER, Laurence, GUILLONNEAU, Claude, ROLLAND, Yves, ATASSI, Ghanem, BISAGNI, Emile

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Synthesis and in vitro evaluation of novel 2,6,9-trisubstituted purines acting as cyclin-dependent kinase inhibitors von LEGRAVEREND, M, LUDWIG, O, BISAGNI, E, LECLERC, S, MEIJER, L, GIOCANTI, N, SADRI, R, FAVAUDON, V

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Synthesis of 13H-Benzo[6,7]- and 13H-Benzo[4,5]indolo[3,2-c]- quinolines: A New Series of Potent Specific Ligands for Triplex DNA von Nguyen, Chi Hung, Marchand, Christophe, Delage, Stéphane, Sun, Jian-Sheng, Garestier, Thérèse, Hélène, Claude, Bisagni, Emile

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Synthesis of C2 alkynylated purines, a new family of potent inhibitors of cyclin-dependent kinases von Legraverend, Michel, Ludwig, Odile, Bisagni, Emile, Leclerc, Sophie, Meijer, Laurent

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4-Benzyl- and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones, a New Family of Potent Anti-HIV Agents:  Optimization and in Vitro Evaluation against Clinically Important HIV Mutant Str... von Benjahad, Abdellah, Courté, Karine, Guillemont, Jérôme, Mabire, Dominique, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Andries, Koen, Pauwels, Rudi, de Béthune, Marie-Pierre, Monneret, Claude, Bisagni, Emile, Nguyen, Chi Hung, Grierson, David S

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Diphenyl quinolines and isoquinolines : Synthesis and primary biological evaluation von CROISY-DELCEY, Martine, CROISY, Alain, CARREZ, Danièle, HUEL, Christiane, CHIARONI, Angèle, DUCROT, Pierre, BISAGNI, Emile, LU JIN, LECLERCQ, Guy

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Synthesis and Evaluation of “AZT-HEPT”, “AZT-Pyridinone”, and “ddC-HEPT” Conjugates as Inhibitors of HIV Reverse Transcriptase von Pontikis, Renée, Dollé, Valérie, Guillaumel, Jean, Dechaux, Elsa, Note, Reine, Nguyen, Chi Hung, Legraverend, Michel, Bisagni, Emile, Aubertin, Anne-Marie, Grierson, David S, Monneret, Claude

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A New Series of Pyridinone Derivatives as Potent Non-Nucleoside Human Immunodeficiency Virus Type 1 Specific Reverse Transcriptase Inhibitors von Dolle, Valerie, Fan, E, Nguyen, Chi Hung, Aubertin, Anne-Marie, Kirn, Andre, Andreola, Marie Line, Jamieson, Gordon, Tarrago-Litvak, Laura, Bisagni, Emile

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Stable Triple-Helical DNA Complexes Formed by Benzopyridoindole− and Benzopyridoquinoxaline− Oligonucleotide Conjugates von Silver, Gail C, Sun, Jian-Sheng, Nguyen, Chi Hung, Boutorine, Alexandre S, Bisagni, Emile, Hélène, Claude

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Synthesis and Biological Properties of New Benz[h]isoquinoline Derivatives von JANIN, Yves L., CARREZ, Daniele, RIOU, Jean-Francois, BISAGNI, Emile

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Synthesis of psoralens and analogues von Bisagni, Emile

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Synthesis and Binding Properties of Oligo-2‘-deoxyribonucleotides Conjugated with Triple-Helix-Specific Intercalators:  Benzo[e] and Benzo[g] Pyridoindoles von Vinogradov, Serguei, Roig, Victoria, Sergueeva, Zinaida, Nguyen, Chi Hung, Arimondo, Paola, Thuong, Nguyen T, Bisagni, Emile, Sun, Jian-Sheng, Hélène, Claude, Asseline, Ulysse

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