Optimization of pyrazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1) von Huynh, Tram, Chen, Zhong, Pang, Suhong, Geng, Jieping, Bandiera, Tiziano, Bindi, Simona, Vianello, Paola, Roletto, Fulvia, Thieffine, Sandrine, Galvani, Arturo, Vaccaro, Wayne, Poss, Michael A., Trainor, George L., Lorenzi, Matthew V., Gottardis, Marco, Jayaraman, Lata, Purandare, Ashok V.

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Discovery and optimization of 4-pyrazolyl-2-aminopyrimidine derivatives as potent spleen tyrosine kinase (SYK) inhibitors von Cervi, Giovanni, D'Alessio, Roberto, Bindi, Simona, Buffa, Laura, Burocchi, Alessia, Canevari, Giulia, Modugno, Michele, Motto, Ilaria, Saturno, Grazia, Orsini, Paolo

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1,4,5,6-Tetrahydropyrrolo[3,4-c]pyrazoles:  Identification of a Potent Aurora Kinase Inhibitor with a Favorable Antitumor Kinase Inhibition Profile von Fancelli, Daniele, Moll, Jürgen, Varasi, Mario, Bravo, Rodrigo, Artico, Roberta, Berta, Daniela, Bindi, Simona, Cameron, Alexander, Candiani, Ilaria, Cappella, Paolo, Carpinelli, Patrizia, Croci, Walter, Forte, Barbara, Giorgini, Maria Laura, Klapwijk, Jan, Marsiglio, Aurelio, Pesenti, Enrico, Rocchetti, Maurizio, Roletto, Fulvia, Severino, Dino, Soncini, Chiara, Storici, Paola, Tonani, Roberto, Zugnoni, Paola, Vianello, Paola

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Abstract 5163: Characterization of NMS-E194, a selective and potent PERK inhibitor with efficacy in the KMS-11 multiple myeloma von Perrera, Claudia, Pulici, Maurizio, Carenzi, Davide, Motto, Ilaria, Fasolini, Marina, Casale, Elena, Depaolini, Stefania Re, Rizzi, Simona, Asa, Daniela, Roletto, Fulvia, Bindi, Simona, Casero, Daniele, Banfi, Patrizia, Ardini, Elena, Amboldi, Nadia, Ballinari, Dario, Gasparri, Fabio, Cribioli, Sabrina, Mancini, Laura, Ciomei, Marina, Donati, Daniele, Felder, Eduard, Galvani, Arturo, Isacchi, Antonella, Valsasina, Barbara

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Discovery of NMS-E973 as novel, selective and potent inhibitor of heat shock protein 90 (Hsp90) von Brasca, Maria Gabriella, Mantegani, Sergio, Amboldi, Nadia, Bindi, Simona, Caronni, Dannica, Casale, Elena, Ceccarelli, Walter, Colombo, Nicoletta, De Ponti, Anna, Donati, Daniele, Ermoli, Antonella, Fachin, Gabriele, Felder, Eduard R., Ferguson, Ronald D., Fiorelli, Claudio, Guanci, Marco, Isacchi, Antonella, Pesenti, Enrico, Polucci, Paolo, Riceputi, Laura, Sola, Francesco, Visco, Carlo, Zuccotto, Fabio, Fogliatto, Gianpaolo

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Novel pyrrole carboxamide inhibitors of JAK2 as potential treatment of myeloproliferative disorders von Brasca, Maria Gabriella, Gnocchi, Paola, Nesi, Marcella, Amboldi, Nadia, Avanzi, Nilla, Bertrand, Jay, Bindi, Simona, Canevari, Giulia, Casero, Daniele, Ciomei, Marina, Colombo, Nicoletta, Cribioli, Sabrina, Fachin, Gabriele, Felder, Eduard R., Galvani, Arturo, Isacchi, Antonella, Motto, Ilaria, Panzeri, Achille, Donati, Daniele

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Potent and Selective Aurora Inhibitors Identified by the Expansion of a Novel Scaffold for Protein Kinase Inhibition von Fancelli, Daniele, Berta, Daniela, Bindi, Simona, Cameron, Alexander, Cappella, Paolo, Carpinelli, Patrizia, Catana, Cornel, Forte, Barbara, Giordano, Patrizia, Giorgini, Maria Laura, Mantegani, Sergio, Marsiglio, Aurelio, Meroni, Maurizio, Moll, Juergen, Pittalà, Valeria, Roletto, Fulvia, Severino, Dino, Soncini, Chiara, Storici, Paola, Tonani, Roberto, Varasi, Mario, Vulpetti, Anna, Vianello, Paola

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Pyrrole-3-carboxamides as potent and selective JAK2 inhibitors von Brasca, Maria Gabriella, Nesi, Marcella, Avanzi, Nilla, Ballinari, Dario, Bandiera, Tiziano, Bertrand, Jay, Bindi, Simona, Canevari, Giulia, Carenzi, Davide, Casero, Daniele, Ceriani, Lucio, Ciomei, Marina, Cirla, Alessandra, Colombo, Maristella, Cribioli, Sabrina, Cristiani, Cinzia, Della Vedova, Franco, Fachin, Gabriele, Fasolini, Marina, Felder, Eduard R., Galvani, Arturo, Isacchi, Antonella, Mirizzi, Danilo, Motto, Ilaria, Panzeri, Achille, Pesenti, Enrico, Vianello, Paola, Gnocchi, Paola, Donati, Daniele

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Abstract A179: NMS-P113, a novel orally available JAK2 selective inhibitor von Gnocchi, Paola, Brasca, Maria Gabriella, Amboldi, Nadia, Avanzi, Nilla, Bindi, Simona, Canevari, Giulia, Casero, Daniele, Ceruti, Roberta, Ciomei, Marina, Cribioli, Sabrina, Cristiani, Cinzia, Nesi, Marcella, Pastori, Wilma, Patton, Veronica, Pellizzoni, Cinzia, Texido, Gemma, Ardini, Elena, Felder, Eduard R., Isacchi, Antonella, Donati, Daniele, Galvani, Arturo

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Different Pathways in the Base-Promoted Isomerization of Benzyl Oxiranyl Ethers von Mordini, Alessandro, Bindi, Simona, Pecchi, Sabina, Degl'Innocenti, Alessandro, Reginato, Gianna, Serci, Alessandro

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Thieno[3,2- c]pyrazoles: A novel class of Aurora inhibitors with favorable antitumor activity von Bindi, Simona, Fancelli, Daniele, Alli, Cristina, Berta, Daniela, Bertrand, Jay A., Cameron, Alexander D., Cappella, Paolo, Carpinelli, Patrizia, Cervi, Giovanni, Croci, Valter, D’Anello, Matteo, Forte, Barbara, Laura Giorgini, M., Marsiglio, Aurelio, Moll, Juergen, Pesenti, Enrico, Pittalà, Valeria, Pulici, Maurizio, Riccardi-Sirtori, Federico, Roletto, Fulvia, Soncini, Chiara, Storici, Paola, Varasi, Mario, Volpi, Daniele, Zugnoni, Paola, Vianello, Paola

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Corrigendum to “Discovery of NMS-E973 as novel, selective and potent inhibitor of heat shock protein 90 (Hsp90)” [Bioorg. Med. Chem. 21 (2013) 7047–7063] von Brasca, Maria Gabriella, Mantegani, Sergio, Amboldi, Nadia, Bindi, Simona, Caronni, Dannica, Casale, Elena, Ceccarelli, Walter, Colombo, Nicoletta, De Ponti, Anna, Donati, Daniele, Ermoli, Antonella, Fachin, Gabriele, Felder, Eduard R., Ferguson, Ronald D., Fiorelli, Claudio, Guanci, Marco, Isacchi, Antonella, Pesenti, Enrico, Polucci, Paolo, Riceputi, Laura, Sola, Francesco, Visco, Carlo, Zuccotto, Fabio, Fogliatto, Gianpaolo

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N-(SUBSTITUTED-PHENYL)-SULFONAMIDE DERIVATIVES AS KINASE INHIBITORS von BINDI, SIMONA, MOTTO, ILARIA, CARENZI, DAVIDE, PULICI, MAURIZIO

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N-(SUBSTITUTED-PHENYL)-SULFONAMIDE DERIVATIVES AS KINASE INHIBITORS von BINDI, Simona, CARENZI, Davide, PULICI, Maurizio, MOTTO, Ilaria

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N-(SUBSTITUTED-PHENYL)-SULFONAMIDE DERIVATIVES AS KINASE INHIBITORS von PULICI Maurizio, MOTTO Ilaria, BINDI Simona, CARENZI Davide

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N-(SUBSTITUTED-PHENYL)-SULFONAMIDE DERIVATIVES AS KINASE INHIBITORS von BINDI, Simona, CARENZI, Davide, PULICI, Maurizio, MOTTO, Ilaria

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N-(SUBSTITUEREREDE-PHENYL)-SULFONAMIDDERIVATER SOM KINASEHÆMMERE von BINDI, Simona, CARENZI, Davide, PULICI, Maurizio, MOTTO, Ilaria

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N-(substituted-phenyl)-sulfonamide derivatives as kinase inhibitors von Motto, Ilaria, Bindi, Simona, Carenzi, Davide, Pulici, Maurizio

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N-(SUBSTITUTED-PHENYL)-SULFONAMIDE DERIVATIVES AS KINASE INHIBITORS von BINDI, Simona, CARENZI, Davide, PULICI, Maurizio, MOTTO, Ilaria

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N-(SUBSTITUTED-PHENYL)-SULFONAMIDE DERIVATIVES AS KINASE INHIBITORS von Motto, Ilaria, Bindi, Simona, Carenzi, Davide, Pulici, Maurizio

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