Improved Diazo-Transfer Reaction for DNA-Encoded Chemistry and Its Potential Application for Macrocyclic DEL-Libraries von Ede, Selahattin, Schenk, Mandy, Bierer, Donald, Weinmann, Hilmar, Graham, Keith

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Construction of diverse peptide structural architectures via chemoselective peptide ligation von Cheung, Carina Hey Pui, Xu, Jianchao, Lee, Chi Lung, Zhang, Yanfeng, Wei, Ruohan, Bierer, Donald, Huang, Xuhui, Li, Xuechen

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Efficient synthesis of hydrocarbon-bridged diaminodiacids through nickel-catalyzed reductive cross-coupling von Wang, Tao, Kong, Yi-Fu, Xu, Yang, Fan, Jian, Xu, Hua-Jian, Bierer, Donald, Wang, Jun, Shi, Jing, Li, Yi-Ming

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Chemical synthesis and racemic crystallization of rat C5a-desArg von Zuo, Chao, Zhang, Baochang, Wu, Meng, Bierer, Donald, Shi, Jing, Fang, Ge-Min

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Biomimetic enantioselective synthesis of β,β-difluoro-α-amino acid derivatives von Peng, Qiupeng, Yan, Bingjia, Li, Fangyi, Lang, Ming, Zhang, Bei, Guo, Donghui, Bierer, Donald, Wang, Jian

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Nickel Phosphite/Phosphine-Catalyzed C–S Cross-Coupling of Aryl Chlorides and Thiols von Jones, Kieran D, Power, Dennis J, Bierer, Donald, Gericke, Kersten M, Stewart, Scott G

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Potent Inhibition of HIF1α and p300 Interaction by a Constrained Peptide Derived from CITED2 von Qin, Xuan, Chen, Hailing, Tu, Licheng, Ma, Yue, Liu, Na, Zhang, Haowei, Li, Di, Riedl, Bernd, Bierer, Donald, Yin, Feng, Li, Zigang

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A Diaminodiacid (DADA) Strategy for the Development of Disulfide Surrogate Peptides von Qi, Yun‐Kun, Qu, Qian, Bierer, Donald, Liu, Lei

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Application of tert-Butyl Disulfide-Protected Amino Acids for the Fmoc Solid-Phase Synthesis of Lactam Cyclic Peptides under Mild Metal-Free Conditions von Chen, Junyou, Cui, Tingting, Sun, Shuaishuai, Guo, Yanyan, Chen, Jingnan, Wang, Jun, Bierer, Donald, Li, Yi-Ming

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Total Chemical Synthesis of Correctly Folded Disulfide-Rich Proteins Using a Removable O‑Linked β‑N‑Acetylglucosamine Strategy von Shi, Wei-Wei, Shi, Chaowei, Wang, Tong-Yue, Li, Yu-Lei, Zhou, Yong-Kang, Zhang, Xu-Han, Bierer, Donald, Zheng, Ji-Shen, Liu, Lei

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Synthesis of Disulfide Surrogate Peptides Incorporating Large‐Span Surrogate Bridges Through a Native‐Chemical‐Ligation‐Assisted Diaminodiacid Strategy von Qu, Qian, Gao, Shuai, Wu, Fangming, Zhang, Meng‐Ge, Li, Ying, Zhang, Long‐Hua, Bierer, Donald, Tian, Chang‐Lin, Zheng, Ji‐Shen, Liu, Lei

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Cyclobutane-bearing restricted anchoring residues enabled geometry-specific hydrocarbon peptide stapling von Chen, Baobao, Liu, Chao, Cong, Wei, Gao, Fei, Zou, Yan, Su, Li, Liu, Lei, Hillisch, Alexander, Lehmann, Lutz, Bierer, Donald, Li, Xiang, Hu, Hong-Gang

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Chemical synthesis and biological activity of peptides incorporating an ether bridge as a surrogate for a disulfide bond von Zhao, Rui, Shi, Pan, Chen, Junyou, Sun, Shuaishuai, Chen, Jingnan, Cui, Jibin, Wu, Fangming, Fang, Gemin, Tian, Changlin, Shi, Jing, Bierer, Donald, Liu, Lei, Li, Yi-Ming

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Antihyperglycemic Activities of Cryptolepine Analogues:  An Ethnobotanical Lead Structure Isolated from Cryptolepis sanguinolenta von Bierer, Donald E, Dubenko, Larisa G, Zhang, Pingsheng, Lu, Qing, Imbach, Patricia A, Garofalo, Albert W, Phuan, Puay-Wah, Fort, Diana M, Litvak, Joane, Gerber, R. Eric, Sloan, Barbara, Luo, Jian, Cooper, Raymond, Reaven, Gerald M

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Chimeric protein probes for C5a receptors through fusion of the anaphylatoxin C5a core region with a small-molecule antagonist von Zuo, Chao, Shi, Wei-Wei, Chen, Xiao-Xu, Glatz, Marie, Riedl, Bernd, Flamme, Ingo, Pook, Elisabeth, Wang, Jiawei, Fang, Ge-Min, Bierer, Donald, Liu, Lei

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Single‐Shot Solid‐Phase Synthesis of Full‐Length H2 Relaxin Disulfide Surrogates von Zhao, Rui, Shi, Pan, Cui, Ji‐bin, Shi, Chaowei, Wei, Xiao‐Xiong, Luo, Jie, Xia, Zhemin, Shi, Wei‐Wei, Zhou, Yingxin, Tang, Jiahui, Tian, Changlin, Meininghaus, Mark, Bierer, Donald, Shi, Jing, Li, Yi‐Ming, Liu, Lei

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Palladium-Catalyzed Direct α-Arylation of p-Methoxybenzyl-Protected S,S-Dimethylsulfoximine von Sirvent, Juan A., Bierer, Donald, Webster, Robert, Lücking, Ulrich

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Synthesis of disulfide surrogate peptides incorporating an ethylene glycol bridge von Wei, Xiao-Xiong, Cui, Ji-Bin, Zhao, Rui, Luo, Jie, Li, Yi-Ming, Bierer, Donald, Shi, Jing

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Chemical synthesis of disulfide surrogate peptides by using beta-carbon dimethyl modified diaminodiacids von Cui, Ji-Bin, Wei, Xiao-Xiong, Zhao, Rui, Zhu, Huixia, Shi, Jing, Bierer, Donald, Li, Yi-Ming

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Efficient synthesis of a side-chain extended diaminodiacid for solid-phase synthesis of peptide disulfide bond mimics von Sun, Shuai-Shuai, Chen, Junyou, Zhao, Rui, Bierer, Donald, Wang, Jun, Fang, Ge-Min, Li, Yi-Ming

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