Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 von Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd

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Total Synthesis and Antitumor Activity of ZK-EPO: The First Fully Synthetic Epothilone in Clinical Development von Klar, Ulrich, Buchmann, Bernd, Schwede, Wolfgang, Skuballa, Werner, Hoffmann, Jens, Lichtner, Rosemarie B.

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Discovery of BAY-405: An Azaindole-Based MAP4K1 Inhibitor for the Enhancement of T‑Cell Immunity against Cancer von Mowat, Jeffrey, Carretero, Rafael, Leder, Gabriele, Aiguabella Font, Nuria, Neuhaus, Roland, Berndt, Sandra, Günther, Judith, Friberg, Anders, Schäfer, Martina, Briem, Hans, Raschke, Marian, Miyatake Ondozabal, Hideki, Buchmann, Bernd, Boemer, Ulf, Kreft, Bertolt, Hartung, Ingo V., Offringa, Rienk

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Identification of novel GLUT inhibitors von Siebeneicher, Holger, Bauser, Marcus, Buchmann, Bernd, Heisler, Iring, Müller, Thomas, Neuhaus, Roland, Rehwinkel, Hartmut, Telser, Joachim, Zorn, Ludwig

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Abstract 4333: Identification and optimization of the first highly selective GLUT-1 inhibitors von Bauser, Marcus, Buchmann, Bernd, Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Mueller, Thomas, Kopitz, Charlotte Christine

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Improved Cellular Pharmacokinetics and Pharmacodynamics Underlie the Wide Anticancer Activity of Sagopilone von HOFFMANN, Jens, VILALE, Ilio, PANARETAKIS, Theocharis, SIEMEISTER, Gerhard, LAGE, Hermann, NANTY, Lisa, HAMMER, Stefanie, MITTELSTAEDT, Kevin, WINSEL, Sebastian, ESCHENBRENNER, Julia, CASTEDO, Maria, DEMARCHE, Carine, BUCHMANN, Bernd, KLAR, Ulrich, KROEMER, Guido, GALLUZZI, Lorenzo, SCHWEDE, Wolfgang, SENOVILLA, Laura, SKUBALLA, Werner, VIVET, Sonia, LICHTNER, Rosemarie B, VICENCIO, José M

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Abstract 1164: Metabolic responses in cancer cells with differential susceptibility to GLUT1 inhibition von Gruenewald, Sylvia, Rennefahrt, Ulrike, Maldonado, Sandra G., Walter, Alexander, Petrul, Heike, Héroult, Mélanie, Heisler, Iring, Quanz, Maria, Steigemann, Patrick, Buchmann, Bernd, Haegebarth, Andrea

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Cover Picture: Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 (ChemMedChem 20/2016) von Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd

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Abstract 4746: Pharmacological characterization of BAY-876, a novel highly selective inhibitor of glucose transporter (GLUT)-1 in vitro and in vivo von Kopitz, Charlotte, Toschi, Luisella, Algire, Carolyn, Héroult, Mélanie, Frisk, Anna-Lena, Meyer, Kirstin, Schmitz, Arndt, Lagkadinou, Eleni, Petrul, Heike, Heisler, Iring, Neuhaus, Roland, Buchmann, Bernd, Himmel, Herbert, Bauser, Marcus, Haegebarth, Andrea, Ziegelbauer, Karl

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Abstract 1442: Effects of selective and broad glucose transporter (GLUT) inhibition on glucose distribution in tumor bearing mice von Heroult, Melanie, Steinke, Wolfram, Frisk, Anna-Lena, Borkowski, Sandra, Meyer, Kirstin, Petrul, Heike, Heisler, Iring, Quanz, Maria, Neuhaus, Roland, Buchmann, Bernd, Mueller, Thomas, Bauser, Marcus, Haegebarth, Andrea, Brands, Michael, Ziegelbauer, Karl

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Abstract 1026: Novel Tie2 inhibitor with in vivo efficacy in disseminated hematological tumor models in mice von Gruenewald, Sylvia, Schueler, Julia, Haerter, Michael, Suessmeier, Frank, Klingner, Kerstin, Boemer, Ulf, Kaulfuss, Stefan, Walter, Alexander, Lobell, Mario, Hartung, Ingo V., Buchmann, Bernd, Heldmann, Dieter, Hess-Stumpp, Holger, Ziegelbauer, Karl

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The Role of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 in the p38/TNF-α Pathway of Systemic and Cutaneous Inflammation von Schottelius, Arndt J., Zügel, Ulrich, Döcke, Wolf-Dietrich, Zollner, Thomas M., Röse, Lars, Mengel, Anne, Buchmann, Bernd, Becker, Andreas, Grütz, Gerald, Naundorf, Sandra, Friedrich, Anke, Gaestel, Matthias, Asadullah, Khusru

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The Role of Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 in the p38/TNF-[alpha] Pathway of Systemic and Cutaneous Inflammation von Schottelius, Arndt J, Zügel, Ulrich, Döcke, Wolf-dietrich, Zollner, Thomas M, Röse, Lars, Mengel, Anne, Buchmann, Bernd, Becker, Andreas, Grütz, Gerald, Naundorf, Sandra, Friedrich, Anke, Gaestel, Matthias, Asadullah, Khusru

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Cover Picture: Total Synthesis and Antitumor Activity of ZK-EPO: The First Fully Synthetic Epothilone in Clinical Development (Angew. Chem. Int. Ed. 47/2006) von Klar, Ulrich, Buchmann, Bernd, Schwede, Wolfgang, Skuballa, Werner, Hoffmann, Jens, Lichtner, Rosemarie B.

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Efficient Chiral Pool Synthesis of the C1-C6 Fragment of Epothilones von Klar, Ulrich, Röhr, Bodo, Kuczynski, Frank, Schwede, Wolfgang, Berger, Markus, Skuballa, Werner, Buchmann, Bernd

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Synthesis of 3H-labeled Efomycine M von Bader, Ben, von Bonin, Arne, Buchmann, Bernd, Gay, Juergen, Gruendemann, Stephan, Guenther, Judith, Schaefer, Martina, Spellig, Tilman, Zollner, Thomas M., Zorn, Ludwig

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Efomycine M: an inhibitor of selectins? von von Bonin, Arne, Buchmann, Bernd, Bader, Ben, Rausch, Alexandra, Venstrom, Kristine, Schäfer, Martina, Gründemann, Stephan, Günther, Judith, Zorn, Ludwig, Nubbemeyer, Reinhard, Asadullah, Khusru, Zollner, Thomas M

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Prostaglandins von Buchmann, Bernd, Rehwinkel, Hartmut

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Epothilones von Buchmann, Bernd, Klar, Ulrich

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PYRAZOLOPYRAZINES ACTING ON CANCERS VIA INHIBITION OF CDK12 von STEIGEMANN, Patrick, THEDE, Kai, BUCHGRABER, Philipp, BUCHMANN, Bernd, WENGNER, Antje Margret, LIENAU, Philip, SIEMEISTER, Gerhard, BARAK, Naomi, BÖMER, Ulf, BERGER, Markus

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