Discovery of Roblitinib (FGF401) as a Reversible-Covalent Inhibitor of the Kinase Activity of Fibroblast Growth Factor Receptor 4 von Fairhurst, Robin A, Knoepfel, Thomas, Buschmann, Nicole, Leblanc, Catherine, Mah, Robert, Todorov, Milen, Nimsgern, Pierre, Ripoche, Sebastien, Niklaus, Michel, Warin, Nicolas, Luu, Van Huy, Madoerin, Mario, Wirth, Jasmin, Graus-Porta, Diana, Weiss, Andreas, Kiffe, Michael, Wartmann, Markus, Kinyamu-Akunda, Jacqueline, Sterker, Dario, Stamm, Christelle, Adler, Flavia, Buhles, Alexandra, Schadt, Heiko, Couttet, Philippe, Blank, Jutta, Galuba, Inga, Trappe, Jörg, Voshol, Johannes, Ostermann, Nils, Zou, Chao, Berghausen, Jörg, Del Rio Espinola, Alberto, Jahnke, Wolfgang, Furet, Pascal

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Discovery and In Vivo Exploration of 1,3,4-Oxadiazole and α‑Fluoroacrylate Containing IL-17 Inhibitors von Velcicky, Juraj, Bauer, Matthias R., Schlapbach, Achim, Lapointe, Guillaume, Meyer, Arndt, Vögtle, Markus, Blum, Ernst, Ngo, Estelle, Rolando, Catherine, Nimsgern, Pierre, Teixeira-Fouchard, Sylvie, Lehmann, Hansjoerg, Furet, Pascal, Berst, Frédéric, Schümann, Jens, Stringer, Rowan, Larger, Patrice, Schmid, Cindy, Prendergast, Catriona T., Riek, Simone, Schmutz, Patrick, Lehmann, Sylvie, Berghausen, Jörg, Scheufler, Clemens, Rondeau, Jean-Michel, Burkhart, Christoph, Knoepfel, Thomas, Gommermann, Nina

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Pharmacokinetic Studies around the Mono- and Difunctionalization of a Bioavailable Cyclic Decapeptide Scaffold von Fouché, Marianne, Schäfer, Michael, Blatter, Markus, Berghausen, Jörg, Desrayaud, Sandrine, Roth, Hans-Jörg

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Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure von Fouché, Marianne, Schäfer, Michael, Berghausen, Jörg, Desrayaud, Sandrine, Blatter, Markus, Piéchon, Philippe, Dix, Ina, Martin Garcia, Aimar, Roth, Hans-Jörg

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Influence of Water-Soluble Polymers on the Shear-Induced Structure Formation in Lyotropic Lamellar Phases von Berghausen, Jörg, Zipfel, Johannes, Lindner, Peter, Richtering, Walter

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Ionic Liquid Versus Prodrug Strategy to Address Formulation Challenges von Balk, Anja, Widmer, Toni, Wiest, Johannes, Bruhn, Heike, Rybak, Jens-Christoph, Matthes, Philipp, Müller-Buschbaum, Klaus, Sakalis, Anastasios, Lühmann, Tessa, Berghausen, Jörg, Holzgrabe, Ulrike, Galli, Bruno, Meinel, Lorenz

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Shear induced structures in lamellar phases of amphiphilic block copolymers von ZIPFEL, J, BERGHAUSEN, J, SCHMIDT, G, LINDNER, P, ALEXANDRIDIS, P, TSIANOU, M, RICHTERING, W

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Accelerated Formulation Development for Nanomilled Active Pharmaceutical Ingredients Using a Screening Approach von Juhnke, M., Berghausen, J., Timpe, C.

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Orally bioavailable Syk inhibitors with activity in a rat PK/PD model von Thoma, Gebhard, Veenstra, Siem, Strang, Ross, Blanz, Joachim, Vangrevelinghe, Eric, Berghausen, Jörg, Lee, Christian C., Zerwes, Hans-Günter

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The influence of aqueous content in small scale salt screening—Improving hit rate for weakly basic, low solubility drugs von Tarsa, Peter B., Towler, Christopher S., Woollam, Grahame, Berghausen, Jörg

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Simulated rat intestinal fluid improves oral exposure prediction for poorly soluble compounds over a wide dose range von Berghausen, Joerg, Seiler, Frank Hans, Gobeau, Nathalie, Faller, Bernard

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Back Cover: Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure (ChemMedChem 10/2016) von Fouché, Marianne, Schäfer, Michael, Berghausen, Jörg, Desrayaud, Sandrine, Blatter, Markus, Piéchon, Philippe, Dix, Ina, Martin Garcia, Aimar, Roth, Hans-Jörg

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Accelerated Formulation Development for Nanomilled Active Pharmaceutical Ingredients Using a Screening Approach : Grinding and Milling von JUHNKE, Michael, BERGHAUSEN, Jörg, TIMPE, Carsten

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Influence of Shear on Lyotropic Lamellar Phases with Different Membrane Defects von Zipfel, Johannes, Berghausen, Jörg, Lindner, Peter, Richtering, Walter

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Influence of Shear on Solvated Amphiphilic Block Copolymers with Lamellar Morphology von Zipfel, Johannes, Berghausen, Jörg, Schmidt, Gudrun, Lindner, Peter, Alexandridis, Paschalis, Richtering, Walter

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Rheology and Shear Orientation of a Nematic Liquid Crystalline Side-Group Polymer with Laterally Attached Mesogenic Units von Berghausen, Jörg, Fuchs, Joachim, Richtering, Walter

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Lamellar phases under shear : variation of the layer orientation across the couette gap von BERGHAUSEN, J, ZIPFEL, J, DIAT, O, NARAYANAN, T, RICHTERING, W

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Diagnosing solubility limitations – the example of hydrate formation von Berghausen, Joerg, Faller, Bernard

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Synthesis of a crystalline form of n-(4-fluorobenzyl)-n-(1-methylpiperidin-4-yl)-n'-(4-(2-methylpropyloxy)phenylmethyl)carbamide tartrate salt von THYGESEN, MIKKEL, ANDERSSON, CARL-MAGNUS, SCHLIENGER, NATHALIE, BERGHAUSEN, JÖRG, TOLF, BO-RAGNAR, BLATTER, FRITZ

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Synthesis of a crystalline form of n-(4-fluorobenzyl)-n-(1-methylpiperidin-4-yl)-n'-(4-(2-methylpropyloxy)phenylmethyl)carbamide tartrate salt von THYGESEN, MIKKEL, ANDERSSON, CARL-MAGNUS, SCHLIENGER, NATHALIE, BERGHAUSEN, JÖRG, TOLF, BO-RAGNAR, BLATTER, FRITZ

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