Discovery of 4′-azido-2′-deoxy-2′-C-methyl cytidine and prodrugs thereof: A potent inhibitor of Hepatitis C virus replication von Nilsson, Magnus, Kalayanov, Genadiy, Winqvist, Anna, Pinho, Pedro, Sund, Christian, Zhou, Xiao-Xiong, Wähling, Horst, Belfrage, Anna-Karin, Pelcman, Michael, Agback, Tatiana, Benckestock, Kurt, Wikström, Kristina, Boothee, Mirva, Lindqvist, Anneli, Rydegård, Christina, Jonckers, Tim H.M., Vandyck, Koen, Raboisson, Pierre, Lin, Tse-I, Lachau-Durand, Sophie, de Kock, Herman, Smith, David B., Martin, Joseph A., Klumpp, Klaus, Simmen, Kenneth, Vrang, Lotta, Terelius, Ylva, Samuelsson, Bertil, Rosenquist, Åsa, Johansson, Nils Gunnar

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Synthesis and SAR of potent inhibitors of the Hepatitis C virus NS3/4A protease: Exploration of P2 quinazoline substituents von Nilsson, Magnus, Belfrage, Anna Karin, Lindström, Stefan, Wähling, Horst, Lindquist, Charlotta, Ayesa, Susana, Kahnberg, Pia, Pelcman, Mikael, Benkestock, Kurt, Agback, Tatiana, Vrang, Lotta, Terelius, Ylva, Wikström, Kristina, Hamelink, Elizabeth, Rydergård, Christina, Edlund, Michael, Eneroth, Anders, Raboisson, Pierre, Lin, Tse-I, de Kock, Herman, Wigerinck, Piet, Simmen, Kenneth, Samuelsson, Bertil, Rosenquist, Åsa

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ENABLE: an engine for European antibacterial drug discovery and development von Olliver, Marie, Griestop, Laura, Hughes, Diarmaid, Belfrage, Anna Karin, Gising, Johan, Baranczewski, Pawel, Vingsbo Lundberg, Carina, Karlén, Anders

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Pan-NS3 protease inhibitors of hepatitis C virus based on an R-elongated pyrazinone scaffold von Belfrage, Anna Karin, Abdurakhmanov, Eldar, Åkerblom, Eva, Brandt, Peter, Alogheli, Hiba, Neyts, Johan, Danielson, U. Helena, Sandström, Anja

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Pan-NS3 protease inhibitors of hepatitis C virus based on an R3-elongated pyrazinone scaffold von Belfrage, Anna Karin, Abdurakhmanov, Eldar, Åkerblom, Eva, Brandt, Peter, Alogheli, Hiba, Neyts, Johan, Danielson, U. Helena, Sandström, Anja

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Palladium-Catalyzed Carbonylation of Aryl Iodides with Sulfinamides von Belfrage, Anna Karin, Wakchaure, Prasad, Larhed, Mats, Sandström, Anja

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Efficient and Selective Palladium-Catalysed C-3 Urea Couplings to 3,5-Dichloro-2(1H)-pyrazinones von Belfrage, Anna Karin, Gising, Johan, Svensson, Fredrik, Åkerblom, Eva, Sköld, Christian, Sandström, Anja

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Discovery of pyrazinone based compounds that potently inhibit the drug-resistant enzyme variant R155K of the hepatitis C virus NS3 protease von Belfrage, Anna Karin, Abdurakhmanov, Eldar, Kerblom, Eva, Brandt, Peter, Oshalim, Anna, Gising, Johan, Skogh, Anna, Neyts, Johan, Danielson, U. Helena, Sandström, Anja

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Discovery of pyrazinone based compounds that potently inhibit the drug-resistant enzyme variant R155K of the hepatitis C virus NS3 protease von Belfrage, Anna Karin, Abdurakhmanov, Eldar, Åkerblom, Eva, Brandt, Peter, Oshalim, Anna, Gising, Johan, Skogh, Anna, Neyts, Johan, Danielson, U. Helena, Sandström, Anja

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Achiral Pyrazinone-Based Inhibitors of the Hepatitis C Virus NS3 Protease and Drug-Resistant Variants with Elongated Substituents Directed Toward the S2 Pocket von Gising, Johan, Belfrage, Anna Karin, Alogheli, Hiba, Ehrenberg, Angelica, Åkerblom, Eva, Svensson, Richard, Artursson, Per, Karlén, Anders, Danielson, U. Helena, Larhed, Mats, Sandström, Anja

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Pan-NS3 protease inhibitors of hepatitis C virus based on an R 3 -elongated pyrazinone scaffold von Belfrage, Anna Karin, Abdurakhmanov, Eldar, Åkerblom, Eva, Brandt, Peter, Alogheli, Hiba, Neyts, Johan, Danielson, U Helena, Sandström, Anja

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Design and Synthesis of Hepatitis C Virus NS3 Protease Inhibitors : Targeting Different Genotypes and Drug-Resistant Variants von Belfrage, Anna Karin

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Design and Synthesis of Hepatitis C Virus NS3 Protease Inhibitors: Targeting Different Genotypes and Drug-Resistant Variants von Belfrage, Anna Karin

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Synthesis and SAR Around the R6 Position of 2(1H)-Pyrazinone Based HCV NS3 Protease Inhibitors von Belfrage, Anna-Karin, Gising, Johan, Örtqvist, Pernilla, Alogheli, Hiba, Ehrenberg, Angelica, Larhed, Mats, Danielson, U Helena, Sandström, Anja

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Design and Synthesis of Potent Inhibitors of the Malaria Aspartyl Proteases Plasmepsin I and II. Use of Solid-Phase Synthesis to Explore Novel Statine Motifs von Johansson, Per-Ola, Chen, Yantao, Belfrage, Anna Karin, Blackman, Michael J, Kvarnström, Ingemar, Jansson, Katarina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil

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Hepatitis C Virus NS3 Protease Inhibitors based on 2(1H)-Pyrazinones von Belfrage, A. K., Gising, J., Örtqvist, P., Danielson, U. H., Larhed, M., Sandström, A.

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Design and Synthesis of Potent Inhibitors of the Malaria Aspartyl Proteases von Johansson, Per-Ola, Chen, Yantao, Belfrage, Anna Karin, Blackman, Michael J., Kvarnström, Ingemar, Jansson, Katarina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenqvist, Åsa, Samuelsson, Bertil

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ChemInform Abstract: Palladium‐Catalyzed Carbonylation of Aryl Iodides with Sulfinamides von Belfrage, Anna Karin, Wakchaure, Prasad, Larhed, Mats, Sandstroem, Anja

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INHIBITORS OF METALLO-BETA-LACTAMASES von LINDSTROM, Stefan, BRANDT, Peter, BREM, Jürgen, SCHOFIELD, Christopher J, BELFRAGE, Anna Karin, ANTONOV, Dmitry, GISING, Johan

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ChemInform Abstract: Efficient and Selective Palladium-Catalyzed C-3 Urea Couplings to 3,5-Dichloro-2(1H)-pyrazinones von Belfrage, Anna Karin, Gising, Johan, Svensson, Fredrik, Aakerblom, Eva, Skoeld, Christian, Sandstroem, Anja

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