3-Substituted Quinolines as RORγt Inverse Agonists von Tanis, Virginia M., Venkatesan, Hariharan, Cummings, Maxwell D., Albers, Michael, Kent Barbay, J., Herman, Krystal, Kummer, David A., Milligan, Cynthia, Nelen, Marina I., Nishimura, Rachel, Schlueter, Thomas, Scott, Brian, Spurlino, John, Wolin, Ronald, Woods, Craig, Xue, Xiaohua, Edwards, James P., Fourie, Anne M., Leonard, Kristi

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Synthesis and characterization of 5,6,7,8-tetrahydroquinoline C5a receptor antagonists von Barbay, J. Kent, Gong, Yong, Buntinx, Mieke, Li, Jian, Claes, Concha, Hornby, Pamela J., Van Lommen, Guy, Van Wauwe, Jean, He, Wei

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Discovery of JNJ-64264681: A Potent and Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase von Tichenor, Mark S., Wiener, John J. M., Rao, Navin L., Bacani, Genesis M., Wei, Jianmei, Pooley Deckhut, Charlotte, Barbay, J. Kent, Kreutter, Kevin D., Chang, Leon, Clancy, Kathleen W., Murrey, Heather E., Wang, Weixue, Ahn, Kay, Huber, Michael, Rex, Elizabeth, Coe, Kevin J., Wu, Jiejun, Rui, Haopeng, Sepassi, Kia, Gaudiano, Marcello, Bekkers, Mariette, Cornelissen, Ivo, Packman, Kathryn, Seierstad, Mark, Xiouras, Christos, Bembenek, Scott D., Alexander, Richard, Milligan, Cynthia, Balasubramanian, Sriram, Lebsack, Alec D., Venable, Jennifer D., Philippar, Ulrike, Edwards, James P., Hirst, Gavin

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Design and optimization of aniline-substituted tetrahydroquinoline C5a receptor antagonists von Gong, Yong, Barbay, J. Kent, Buntinx, Mieke, Li, Jian, Wauwe, Jean Van, Claes, Concha, Lommen, Guy Van, Hornby, Pamela J., He, Wei

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6-Substituted quinolines as RORγt inverse agonists von Barbay, J. Kent, Cummings, Maxwell D., Abad, Marta, Castro, Glenda, Kreutter, Kevin D., Kummer, David A., Maharoof, Umar, Milligan, Cynthia, Nishimura, Rachel, Pierce, Joan, Schalk-Hihi, Celine, Spurlino, John, Tanis, Virginia M., Urbanski, Maud, Venkatesan, Hariharan, Wang, Aihua, Woods, Craig, Wolin, Ronald, Xue, Xiaohua, Edwards, James P., Fourie, Anne M., Leonard, Kristi

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Discovery of a Potent and Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase with Oral Anti-Inflammatory Activity von Tichenor, Mark S, Wiener, John J. M, Rao, Navin L, Pooley Deckhut, Charlotte, Barbay, J. Kent, Kreutter, Kevin D, Bacani, Genesis M, Wei, Jianmei, Chang, Leon, Murrey, Heather E, Wang, Weixue, Ahn, Kay, Huber, Michael, Rex, Elizabeth, Coe, Kevin J, Wu, JieJun, Seierstad, Mark, Bembenek, Scott D, Leonard, Kristi A, Lebsack, Alec D, Venable, Jennifer D, Edwards, James P

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Substituted thieno[2,3-d]pyrimidines as adenosine A2A receptor antagonists von Shook, Brian C., Chakravarty, Devraj, Barbay, J. Kent, Wang, Aihua, Leonard, Kristi, Alford, Vernon, Powell, Mark T., Rassnick, Stefanie, Scannevin, Robert H., Carroll, Karen, Wallace, Nathaniel, Crooke, Jeffrey, Ault, Mark, Lampron, Lisa, Westover, Lori, Rhodes, Kenneth, Jackson, Paul F.

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Design and Characterization of Optimized Adenosine A2A/A1 Receptor Antagonists for the Treatment of Parkinson's Disease von Shook, Brian C, Rassnick, Stefanie, Wallace, Nathaniel, Crooke, Jeffrey, Ault, Mark, Chakravarty, Devraj, Barbay, J. Kent, Wang, Aihua, Powell, Mark T, Leonard, Kristi, Alford, Vernon, Scannevin, Robert H, Carroll, Karen, Lampron, Lisa, Westover, Lori, Lim, Heng-Keang, Russell, Ronald, Branum, Shawn, Wells, Kenneth M, Damon, Sandra, Youells, Scott, Li, Xun, Beauchamp, Derek A, Rhodes, Kenneth, Jackson, Paul F

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Optimization of arylindenopyrimidines as potent adenosine A(2A)/A(1) antagonists von Shook, Brian C, Rassnick, Stefanie, Chakravarty, Devraj, Wallace, Nathaniel, Ault, Mark, Crooke, Jeffrey, Barbay, J Kent, Wang, Aihua, Leonard, Kristi, Powell, Mark T, Alford, Vernon, Hall, Daniel, Rupert, Kenneth C, Heintzelman, Geoffrey R, Hansen, Kristen, Bullington, James L, Scannevin, Robert H, Carroll, Karen, Lampron, Lisa, Westover, Lori, Russell, Ronald, Branum, Shawn, Wells, Kenneth, Damon, Sandra, Youells, Scott, Beauchamp, Derek, Li, Xun, Rhodes, Kenneth, Jackson, Paul F

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Synthesis and SAR of pyridazinone-substituted phenylalanine amide α4 integrin antagonists von YONG GONG, BARBAY, J. Kent, KIMBALL, Edward S, SANTULLI, Rosemary J, FISHER, M. Carolyn, DYATKIN, Alexey B, MISKOWSKI, Tamara A, HORNBY, Pamela J, WEI HE

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Design and Characterization of Optimized Adenosine A 2A /A 1 Receptor Antagonists for the Treatment of Parkinson's Disease von Shook, Brian C., Rassnick, Stefanie, Wallace, Nathaniel, Crooke, Jeffrey, Ault, Mark, Chakravarty, Devraj, Barbay, J. Kent, Wang, Aihua, Powell, Mark T., Leonard, Kristi, Alford, Vernon, Scannevin, Robert H., Carroll, Karen, Lampron, Lisa, Westover, Lori, Lim, Heng-Keang, Russell, Ronald, Branum, Shawn, Wells, Kenneth M., Damon, Sandra, Youells, Scott, Li, Xun, Beauchamp, Derek A., Rhodes, Kenneth, Jackson, Paul F.

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Synthesis and Biological Evaluation of Novel Pyridazinone-Based α4 Integrin Receptor Antagonists von Gong, Yong, Barbay, J. Kent, Dyatkin, Alexey B, Miskowski, Tamara A, Kimball, Edward S, Prouty, Stephen M, Fisher, M. Carolyn, Santulli, Rosemary J, Schneider, Craig R, Wallace, Nathaniel H, Ballentine, Scott A, Hageman, William E, Masucci, John A, Maryanoff, Bruce E, Damiano, Bruce P, Andrade-Gordon, Patricia, Hlasta, Dennis J, Hornby, Pamela J, He, Wei

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Optimization of arylindenopyrimidines as potent adenosine A2A/A1 antagonists von SHOOK, Brian C, RASSNICK, Stefanie, ALFORD, Vernon, HALL, Daniel, RUPERT, Kenneth C, HEINTZELMAN, Geoffrey R, HANSEN, Kristen, BULLINGTON, James L, SCANNEVIN, Robert H, CARROLL, Karen, LAMPRON, Lisa, WESTOVER, Lori, CHAKRAVARTY, Devraj, RUSSELL, Ronald, BRANUM, Shawn, WELLS, Kenneth, DAMON, Sandra, YOUELLS, Scott, BEAUCHAMP, Derek, XUN LI, RHODES, Kenneth, JACKSON, Paul F, WALLACE, Nathaniel, AULT, Mark, CROOKE, Jeffrey, BARBAY, J. Kent, AIHUA WANG, LEONARD, Kristi, POWELL, Mark T

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Synthesis and SAR of pyridazinone-substituted phenylalanine amide α 4 integrin antagonists von Gong, Yong, Kent Barbay, J., Kimball, Edward S., Santulli, Rosemary J., Carolyn Fisher, M., Dyatkin, Alexey B., Miskowski, Tamara A., Hornby, Pamela J., He, Wei

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Optimization of arylindenopyrimidines as potent adenosine A 2A/A 1 antagonists von Shook, Brian C., Rassnick, Stefanie, Chakravarty, Devraj, Wallace, Nathaniel, Ault, Mark, Crooke, Jeffrey, Barbay, J. Kent, Wang, Aihua, Leonard, Kristi, Powell, Mark T., Alford, Vernon, Hall, Daniel, Rupert, Kenneth C., Heintzelman, Geoffrey R., Hansen, Kristen, Bullington, James L., Scannevin, Robert H., Carroll, Karen, Lampron, Lisa, Westover, Lori, Russell, Ronald, Branum, Shawn, Wells, Kenneth, Damon, Sandra, Youells, Scott, Beauchamp, Derek, Li, Xun, Rhodes, Kenneth, Jackson, Paul F.

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Aminomethyl substituted thieno[2,3-d]pyrimidines as adenosine A2A receptor antagonists von Shook, Brian C., Charavarty, Devraj, Barbay, J. Kent, Wang, Aihua, Leonard, Kristi, Alford, Vernon, Powell, Mark, Beauchamp, Derek A., Rassnick, Stefanie, Scannevin, Robert, Carroll, Karen, Wallace, Nathaniel, Crooke, Jeffrey, Ault, Mark, Lampron, Lisa, Westover, Lori, Rhodes, Kenneth, Jackson, Paul F.

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Synthesis and Biological Evaluation of Novel Pyridazinone-Based α 4 Integrin Receptor Antagonists von Gong, Yong, Barbay, J. Kent, Dyatkin, Alexey B., Miskowski, Tamara A., Kimball, Edward S., Prouty, Stephen M., Fisher, M. Carolyn, Santulli, Rosemary J., Schneider, Craig R., Wallace, Nathaniel H., Ballentine, Scott A., Hageman, William E., Masucci, John A., Maryanoff, Bruce E., Damiano, Bruce P., Andrade-Gordon, Patricia, Hlasta, Dennis J., Hornby, Pamela J., He, Wei

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Synthesis and biological evaluation of novel pyridazinone-based alpha4 integrin receptor antagonists von Gong, Yong, Barbay, J Kent, Dyatkin, Alexey B, Miskowski, Tamara A, Kimball, Edward S, Prouty, Stephen M, Fisher, M Carolyn, Santulli, Rosemary J, Schneider, Craig R, Wallace, Nathaniel H, Ballentine, Scott A, Hageman, William E, Masucci, John A, Maryanoff, Bruce E, Damiano, Bruce P, Andrade-Gordon, Patricia, Hlasta, Dennis J, Hornby, Pamela J, He, Wei

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SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE von HERRMANN Aaron T, CHAI Wenying, KRAWCZUK Paul J, KREUTTER Kevin D, ECCLES Wendy, ROVIRA Alexander R, PIPPEL Daniel J, WOLIN Ronald L, JONES William M, BARBAY J. Kent, LEBSACK Alec D, HACK Michael D

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SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE von PIPPEL, DANIEL, J, WOLIN, RONALD, L, LEBSACK, ALEC, D, HACK, MICHAEL, D, ECCLES, WENDY, ROVIRA, ALEXANDER, R, CHAI, WENYING, BARBAY, J. KENT, JONES, WILLIAM, M, KREUTTER, KEVIN, D, HERRMANN, AARON, T, KRAWCZUK, PAUL, J

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