Syntheses, biological evaluation of some novel substituted benzoic acid derivatives bearing hydrazone as linker von Mishra, Ganesh Prasad, Sharma, Rajesh, Jain, Mukul, Bandyopadhyay, Debdutta

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Pulmonary tuberculosis - An emerging risk factor for venous thromboembolism: A case series and review of literature von Gupta, Amitesh, Mrigpuri, Parul, Faye, Abhishek, Bandyopadhyay, Debdutta, Singla, Rupak

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Overexpression of histone deacetylase 1 confers resistance to sodium butyrate-mediated apoptosis in melanoma cells through a p53-mediated pathway von BANDYOPADHYAY, Debdutta, MISHRA, Anupam, MEDRANO, Estela E

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ZYBT1, a potent, irreversible Bruton’s Tyrosine Kinase (BTK) inhibitor that inhibits the C481S BTK with profound efficacy against arthritis and cancer von Ghoshdastidar, Krishnarup, Patel, Hoshang, Bhayani, Hitesh, Patel, Ankit, Thakkar, Kinjal, Patel, Dinesh, Sharma, Manoranjan, Singh, Jaideep, Mohapatra, Jogeswar, Chatterjee, Abhijit, Patel, Dipam, Bahekar, Rajesh, Sharma, Rajiv, Gupta, Lakshmikant, Patel, Nirmal, Giri, Poonam, Srinivas, Nuggehally R., Jain, Mukul, Bandyopadhyay, Debdutta, Patel, Pankaj R., Desai, Ranjit C.

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Reliability and validity of an audio signal modified shuttle walk test von Singla, Rupak, Rai, Richa, Faye, Abhishek Anil, Jain, Anil Kumar, Chowdhury, Ranadip, Bandyopadhyay, Debdutta

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Physical Interaction between Epidermal Growth Factor Receptor and DNA-dependent Protein Kinase in Mammalian Cells von Bandyopadhyay, Debdutta, Mandal, Mahitosh, Adam, Liana, Mendelsohn, John, Kumar, Rakesh

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Discovery of Orally Active, Potent, and Selective Benzotriazole-Based PTP1B Inhibitors von Patel, Dipam, Jain, Mukul, Shah, Shailesh R., Bahekar, Rajesh, Jadav, Pradip, Darji, Brijesh, Siriki, Yernaidu, Bandyopadhyay, Debdutta, Joharapurkar, Amit, Kshirsagar, Samadhan, Patel, Harilal, Shaikh, Mubeen, Sairam, Kalapatapu V. V. M., Patel, Pankaj

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Protein-Tyrosine Phosphatase 1B Complexes with the Insulin Receptor in Vivo and Is Tyrosine-phosphorylated in the Presence of Insulin von Bandyopadhyay, Debdutta, Kusari, Anasua, Kenner, Kathleen A., Liu, Feng, Chernoff, Jonathan, Gustafson, Thomas A., Kusari, Jyotirmoy

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The low molecular weight cyclin E isoforms augment angiogenesis and metastasis of human melanoma cells in vivo von BALES, Elise, MILLS, Lisa, KEYOMARSI, Khandan, MEDRANO, Estela E, MILAM, Nancy, MCGAHREN-MURRAY, Mollianne, BANDYOPADHYAY, Debdutta, DAHU CHEN, REED, Jon A, TIMCHENKO, Nikolai, VAN DEN OORD, Joost J, BAR-ELI, Menashe

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Identification of a novel orally bioavailable NLRP3 inflammasome inhibitor von Agarwal, Sameer, Pethani, Jignesh P., Shah, Hardik A., Vyas, Vismit, Sasane, Santosh, Bhavsar, Harsh, Bandyopadhyay, Debdutta, Giri, Poonam, Viswanathan, Kasinath, Jain, Mukul R., Sharma, Rajiv

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Optimisation of momelotinib with improved potency and efficacy as pan-JAK inhibitor von Desai, Jigar, Patel, Bhaumin, Gite, Archana, Panchal, Nandini, Gite, Sanjay, Argade, Anil, Kumar, Jeevan, Sachchidanand, S., Bandyopadhyay, Debdutta, Ghoshdastidar, Krishnarup, Patel, Hoshang, Chatterjee, Abhijit, Mahapatra, Jogeshwar, Sharma, Manoranjan, Giri, Poonam, Kumar, Sanjay, Jain, Mukul, Sharma, Rajiv, Desai, Ranjit

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ZYKR1, a novel, potent, and peripherally selective kappa opioid receptor agonist reduces visceral pain and pruritus in animal models von Jain, Mukul R., Patel, Rakesh B., Prajapati, Kanaiyalal D., Vyas, Purvi, Bandyopadhyay, Debdutta, Prajapati, Vijay, Bahekar, Rajesh, Patel, Prakash N., Kawade, Harish M., Kokare, Dadasaheb M., Pawar, Vishwanath, Desai, Ranjit

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Bronchogenic Cyst Presenting as Mediastinal Mass with Pleural Effusion and Unusual Bronchoscopic Findings: A Case Report and Review of Literature von Gupta, Amitesh, Mrigpuri, Parul, Singla, Rupak, Saha, Subhadeep, Anand, Shweta, Faye, Abhishek, Bandyopadhyay, Debdutta, Rathore, Roshan Singh

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Discovery of novel, potent and orally efficacious inhibitor of neutral amino acid transporter B0AT1 (SLC6A19) von Desai, Jigar, Patel, Bhaumin, Darji, Brijesh, Gite, Archana, Panchal, Nandini, Bhosale, Gokul, Shedage, Sandeep, Patel, Sandip, Kadam, Pravin, Patel, Gautam, Kumar Srivastava, Brijesh, Joharapurkar, Amit, Kshirsagar, Samadhan, Giri, Poonam, Bhayani, Hitesh, Patel, Ankit, Ghoshdastidar, Krishnarup, Bandyopadhyay, Debdutta, Kumar, Sanjay, Jain, Mukul, Sharma, Rajiv

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Discovery of a potent G-protein-coupled receptor 119 agonist for the treatment of type 2 diabetes von Pola, Suresh, Shah, Shailesh R., Pingali, Harikishore, Zaware, Pandurang, Thube, Baban, Makadia, Pankaj, Patel, Hoshang, Bandyopadhyay, Debdutta, Rath, Akshyaya, Giri, Suresh, Patel, Jitendra H., Ranvir, R.K., Sundar, S.R., Patel, Harilal, Kumar, Jeevan, Jain, Mukul R.

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Discovery of N‑Cyano-sulfoximineurea Derivatives as Potent and Orally Bioavailable NLRP3 Inflammasome Inhibitors von Agarwal, Sameer, Sasane, Santosh, Shah, Hardik A, Pethani, Jignesh P, Deshmukh, Prashant, Vyas, Vismit, Iyer, Pravin, Bhavsar, Harsh, Viswanathan, Kasinath, Bandyopadhyay, Debdutta, Giri, Poonam, Mahapatra, Jogeswar, Chatterjee, Abhijit, Jain, Mukul R, Sharma, Rajiv

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Design, synthesis and biological evaluation of novel pyrazolo-pyrimidin-amines as potent and selective BTK inhibitors von Joshi, Darshan, Bahekar, Rajesh, Soman, Shubhangi, Jadav, Pradip, Patel, Dipam, Goswami, Amitgiri, Pethani, Jignesh, Kumar, Jeevan, Patel, Jitendra, Sundar, Rajesh, Goswami, Poonamgiri, Goshdastidar, Krishnarup, Patel, Hoshang, Patel, Ankit, Bandyopadhyay, Debdutta, Chattarjee, Abhijit, Sharma, Manoranjan, Jain, Mukul, Desai, Ranjit

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Discovery of 1,3-dihydro-2H-imidazo[4,5-c]quinolin-2-ones based novel, potent and PI3Kδ selective inhibitors von Bahekar, Rajesh, Dave, Bhushan, Soman, Shubhangi, Patel, Dipam, Chopade, Rajendra, Funde, Radhika, Kumar, Jeevan, Sachchidanand, S., Giri, Poonam, Chatterjee, Abhijit, Mahapatra, Jogeswar, Vyas, Purvi, Ghoshdastidar, Krishnarup, Bandyopadhyay, Debdutta, Desai, Ranjit C.

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ZYDG2, a Potent, Selective, and Safe GPR40 Agonist for Treatment of Type 2 Diabetes von JAIN, MUKUL R., GIRI, SURESH R., TRIVEDI, CHITRANG J., BHOI, BIBHUTI B., RATH, AKSHYAYA CHANDAN, RATHOD, ROHAN MANUBHAI, SUNDAR, RAJESH, BANDYOPADHYAY, DEBDUTTA, RAMDHAVE, RASHMI, PATEL, GAUTAM D., SRIVASTAVA, BRIJESH KUMAR, DESAI, RANJIT C.

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Insulin-Induced Mitogen-Activated Protein (MAP) Kinase Phosphatase-1 (MKP-1) Attenuates Insulin-Stimulated MAP Kinase Activity: A Mechanism for the Feedback Inhibition of Insulin S... von Kusari, Anasua B, Byon, John, Bandyopadhyay, Debdutta, Kenner, Kathleen A, Kusari, Jyotirmoy

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