GSK137, a potent small-molecule BCL6 inhibitor with in vivo activity, suppresses antibody responses in mice von Pearce, Andrew C., Bamford, Mark J., Barber, Ruth, Bridges, Angela, Convery, Maire A., Demetriou, Constantinos, Evans, Sian, Gobbetti, Thomas, Hirst, David J., Holmes, Duncan S., Hutchinson, Jonathan P., Jayne, Sandrine, Lezina, Larissa, McCabe, Michael T., Messenger, Cassie, Morley, Joanne, Musso, Melissa C., Scott-Stevens, Paul, Manso, Ana Sousa, Schofield, Jennifer, Slocombe, Tom, Somers, Don, Walker, Ann L., Wyce, Anastasia, Zhang, Xi-Ping, Wagner, Simon D.

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Partial Reduction of Pyridinium Salts as a Versatile Route to Dihydropyridones von Donohoe, Timothy J., Johnson, Dale J., Mace, Laura H., Bamford, Mark J., Ichihara, Osamu

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Copper-catalyzed rearrangement of oximes into primary amides von Sharma, Sumeet K., Bishopp, Simon D., Liana Allen, C., Lawrence, Ruth, Bamford, Mark J., Lapkin, Alexei A., Plucinski, Pawel, Watson, Robert J., Williams, Jonathan M.J.

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Iridium-catalyzed formylation of amines with paraformaldehyde von Saidi, Ourida, Bamford, Mark J., Blacker, A. John, Lynch, James, Marsden, Stephen P., Plucinski, Pawel, Watson, Robert J., Williams, Jonathan M.J.

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In search of a small molecule agonist of the relaxin receptor RXFP1 for the treatment of liver fibrosis von McBride, Andrew, Hoy, Anna M., Bamford, Mark J., Mossakowska, Danuta E., Ruediger, Martin P., Griggs, Jeremy, Desai, Sapna, Simpson, Kate, Caballero-Hernandez, Ivan, Iredale, John P., Pell, Theresa, Aucott, Rebecca L., Holmes, Duncan S., Webster, Scott P., Fallowfield, Jonathan A.

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Identification of clinical candidates from the benzazepine class of histamine H3 receptor antagonists von Wilson, David M., Apps, James, Bailey, Nicholas, Bamford, Mark J., Beresford, Isabel J., Brackenborough, Kim, Briggs, Michael A., Brough, Stephen, Calver, Andrew R., Crook, Barry, Davis, Rebecca K., Davis, Robert P., Davis, Susannah, Dean, David K., Harris, Leanne, Heslop, Teresa, Holland, Vicky, Jeffrey, Phillip, Panchal, Terrance A., Parr, Christopher A., Quashie, Nigel, Schogger, Joanne, Sehmi, Sanjeet S., Stean, Tania O., Steadman, Jon G.A., Trail, Brenda, Wald, Jeffrey, Worby, Angela, Takle, Andrew K., Witherington, Jason, Medhurst, Andrew D.

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Biphenyl amide p38 kinase inhibitors 4: DFG-in and DFG-out binding modes von Angell, Richard M., Angell, Tony D., Bamborough, Paul, Bamford, Mark J., Chung, Chun-wa, Cockerill, Stuart G., Flack, Stephen S., Jones, Katherine L., Laine, Dramane I., Longstaff, Timothy, Ludbrook, Steve, Pearson, Rosannah, Smith, Kathryn J., Smee, Penny A., Somers, Don O., Walker, Ann L.

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The discovery of the benzazepine class of histamine H3 receptor antagonists von Wilson, David M., Apps, James, Bailey, Nicholas, Bamford, Mark J., Beresford, Isabel J., Briggs, Michael A., Calver, Andrew R., Crook, Barry, Davis, Robert P., Davis, Susannah, Dean, David K., Harris, Leanne, Heightman, Tom D., Panchal, Terry, Parr, Christopher A., Quashie, Nigel, Steadman, Jon G.A., Schogger, Joanne, Sehmi, Sanjeet S., Stean, Tania O., Takle, Andrew K., Trail, Brenda K., White, Trevor, Witherington, Jason, Worby, Angela, Medhurst, Andrew D.

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Orally active C-6 heteroaryl- and heterocyclyl-substituted imidazo[1,2- a]pyridine acid pump antagonists (APAs) von Bailey, Nick, Bamford, Mark J., Brissy, Delphine, Brookfield, Joanna, Demont, Emmanuel, Elliott, Richard, Garton, Neil, Farre-Gutierrez, Irene, Hayhow, Thomas, Hutley, Gail, Naylor, Antoinette, Panchal, Terry A., Seow, Hui-Xian, Spalding, David, Takle, Andrew K.

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The identification of potent, selective and CNS penetrant furan-based inhibitors of B-Raf kinase von Takle, Andrew K., Bamford, Mark J., Davies, Susannah, Davis, Robert P., Dean, David K., Gaiba, Alessandra, Irving, Elaine A., King, Frank D., Naylor, Antoinette, Parr, Christopher A., Ray, Alison M., Reith, Alastair D., Smith, Beverley B., Staton, Penelope C., Steadman, Jon G.A., Stean, Tania O., Wilson, David M.

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(1 H-Imidazo[4,5- c]pyridin-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: A novel class of potent MSK-1-inhibitors von Bamford, Mark J., Alberti, Michael J., Bailey, Nicholas, Davies, Susannah, Dean, David K., Gaiba, Alessandra, Garland, Stephen, Harling, John D., Jung, David K., Panchal, Terence A., Parr, Christopher A., Steadman, Jon G., Takle, Andrew K., Townsend, James T., Wilson, David M., Witherington, Jason

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The ammonia-free partial reduction of substituted pyridinium salts von Donohoe, Timothy J, Johnson, Dale J, Mace, Laura H, Thomas, Rhian E, Chiu, Jessica Y K, Rodrigues, Jason S, Compton, Richard G, Banks, Craig E, Tomcik, Peter, Bamford, Mark J, Ichihara, Osamu

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(1 H-Imidazo[4,5- c]pyridin-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: Further optimisation as highly potent and selective MSK-1-inhibitors von Bamford, Mark J., Bailey, Nicholas, Davies, Susannah, Dean, David K., Francis, Leann, Panchal, Terence A., Parr, Christopher A., Sehmi, Sanjeet, Steadman, Jon G., Takle, Andrew K., Townsend, James T., Wilson, David M.

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Synthesis and antiviral activity of 3'-deoxy-3'-C-hydroxymethyl nucleosides von Bamford, Mark J, Coe, Paul L, Walker, Richard T

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4-Acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a Novel Class of Non-Brain-Penetrant Histamine H3 Receptor Antagonists von Procopiou, Panayiotis A, Ancliff, Rachael A, Bamford, Mark J, Browning, Christopher, Connor, Helen, Davies, Susannah, Fogden, Yvonne C, Hodgson, Simon T, Holmes, Duncan S, Looker, Brian E, Morriss, Karen M. L, Parr, Christopher A, Pickup, Elizabeth A, Sehmi, Sanjeet S, White, Gemma V, Watts, Clarissa J, Wilson, David M, Woodrow, Michael D

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Synthesis of the potent influenza neuraminidase inhibitor 4-guanidino Neu5Ac2en. X-Ray molecular structure of 5-acetamido-4-amino-2,6-anhydro-3,4,5-trideoxy-D-erythro-L-gluco-nonon... von Chandler, Malcolm, Bamford, Mark J., Conroy, Richard, Lamont, Brian, Patel, Bina, Patel, Vipulkumar K., Steeples, Ian P., Storer, Richard, Weir, Niall G., Wright, Michael, Williamson, Christopher

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Synthesis and antiviral activity of some 3'-C-difluoromethyl- and 3'-deoxy-3'-C-fluoromethyl nucleosides von Bamford, Mark J, Coe, Paul L, Walker, Richard T

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Functionalised pyrrolidinones derived from ( S)-pyroglutamic acid von Beard, Mark J, Bailey, Jonathan H, Cherry, David T, Moloney, Mark G, Shim, Sung Bo, Statham, Kathryn A, Bamford, Mark J, Brian Lamont, R

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Corrigendum to “(1H-Imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: A novel class of potent MSK-1-inhibitors” [Bioorg. Med. Chem. Lett. 15 (2005) 3402–3406]... von Bamford, Mark J., Alberti, Michael J., Bailey, Nicholas, Davies, Susannah, Dean, David K., Gaiba, Alessandra, Garland, Stephen, Harling, John D., Jung, David K., Panchal, Terence A., Parr, Christopher A., Steadman, Jon G., Takle, Andrew K., Townsend, James T., Wilson, David M., Witherington, Jason

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A concise approach to functionalised, homochiral pyrrolidinones von Bamford, Mark J, Beard, Mark, Cherry, David T, Moloney, Mark G

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