A New Lithium Alkoxide Accelerated Diastereoselective Cyanation of Ketones von Wilkinson, H. Scott, Grover, Paul T, Vandenbossche, Charles P, Bakale, Roger P, Bhongle, Nandkumar N, Wald, Stephen A, Senanayake, Chris H

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Control of Diastereoselectivity by Solvent Effects in the Addition of Grignard Reagents to Enantiopure t-Butylsulfinimine:  Syntheses of the Stereoisomers of the Hydroxyl Derivativ... von Lu, Bruce Z, Senanayake, Chris, Li, Nansheng, Han, Zhengxu, Bakale, Roger P, Wald, Stephen A

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Albuterol. A pharmaceutical chemistry review of R-, S-, and RS-albuterol von Bakale, R P, Wald, S A, Butler, H T, Gao, Y, Hong, Y, Nie, X, Zepp, C M

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Tin-directed Baeyer-Villiger and Beckmann fragmentations von Bakale, Roger P, Scialdone, Mark A, Johnson, Carl R

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Remarkably selective palladium-catalyzed amination process: Rapid assembly of multiamino based structures von Hong, Yaping, Senanayake, Chris H., Xiang, Tingjian, Vandenbossche, Charles P., Tanoury, Gerald J., Bakale, Roger P., Wald, Stephen A.

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Rigid aminoalcohol backbone as a highly defined chiral template for the preparation of optically active tertiary α-hydroxyl acids von Senanayake, Chris H., Fang, Kevin, Grover, Paul, Bakale, Roger P., Vandenbossche, Charles P., Wald, Stephen A.

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Efficient and scalable arylation of bicyclic lactones to form quaternary centers using conventional and microwave radiation von Malcolm, Scott C., Ribe, Seth, Wang, Fengjiang, Hewitt, Michael C., Bhongle, Nandkumar, Bakale, Roger P., Shao, Liming

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Palladium catalyzed amination of 2-chloro-1,3-azole derivatives: Mild entry to potent H 1- antihistaminic norastemizole von Hong, Yaping, Tanoury, Gerald J., Wilkinson, H.Scott, Bakale, Roger P., Wald, Stephen A., Senanayake, Chris H.

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A large-scale asymmetric synthesis of ( S)-cyclohexylphenyl glycolic acid von Su, Xiping, Bhongle, Nandkumar N, Pflum, Derek, Butler, Hal, Wald, Stephen A, Bakale, Roger P, Senanayake, Chris H

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Properly tuned first fluoride-catalyzed TGME-mediated amination process for chloroimidazoles: inexpensive technology for antihistaminic norastemizole von Senanayake, Chris H., Hong, Yaping, Xiang, Tingjian, Wilkinson, H.Scott, Bakale, Roger P., Jurgens, Alex R., Pippert, Mark F., Butler, Hal T., Wald, Stephen A.

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Two approaches for the syntheis of carbon-11 labeled (R) and (S)-albuterol von Valliant, J. F., Riddoch, R. W., Dolovich, M., Chirakal, R., Hong, Y., Bakale, R. P., Wald, S. A., Schaefer, K.

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Synthesis of enantiomerically pure desmethylzopiclone and determination of its absolute configuration von Hong, Yaping, Bakale, Roger P., Fang, Qun K., Xiang, Tingjian, Han, Zhengxu, McConville, Fran X., Senanayake, Chris H., Wald, Stephen A.

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Albuterol : A pharmaceutical chemistry review of R-, S-, and RS-albuterol: R-Albuterol von BAKALE, R. P, WALD, S. A, BUTLER, H. T, YUN GAO, YAPING HONG, XIAOYI NIE, ZEPP, C. M

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ChemInform Abstract: Remarkably Selective Palladium-Catalyzed Amination Process: Rapid Assembly of Multiamino Based Structures von HONG, Y., SENANAYAKE, C. H., XIANG, T., VANDENBOSSCHE, C. P., TANOURY, G. J., BAKALE, R. P., WALD, S. A.

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Development of a Process Route to the FAK/ALK Dual Inhibitor TEV-37440 von Allwein, Shawn P, Mowrey, Dale R, Petrillo, Daniel E, Reif, James J, Purohit, Vikram C, Milkiewicz, Karen L, Bakale, Roger P, Christie, Michael A, Olsen, Mark A, Neville, Christopher J, Gilmartin, Gregory J

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Discovery and Process Synthesis of Novel 2,7-Pyrrolo[2,1-f][1,2,4]triazines von Thieu, Tho, Sclafani, Joseph A, Levy, Daniel V, McLean, Andrew, Breslin, Henry J, Ott, Gregory R, Bakale, Roger P, Dorsey, Bruce D

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Synthesis, characterization and antiproliferative activity of hexa arm star shaped thiosemicarbazones derived from cyclotriphosphazene core von Machakanur, Shrinath S., Patil, Basavaraj R., Naik, Ganesh N., Bakale, Raghavendra P., Annie Bligh, S.W., Gudasi, Kalagouda B.

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Synthesis, characterization and anticancer evaluation of novel tri-arm star shaped 1,3,5-triazine hydrazones von Machakanur, Shrinath S., Patil, Basavaraj R., Badiger, Dayananda S., Bakale, Raghavendra P., Gudasi, Kalagouda B., Annie Bligh, S.W.

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A General Preparation of Protected Phosphoamino Acids von Petrillo, Daniel E, Mowrey, Dale R, Allwein, Shawn P, Bakale, Roger P

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Development and Scale-Up of an Optimized Route to the ALK Inhibitor CEP-28122 von Allwein, Shawn P, Roemmele, Renee C, Haley, James J, Mowrey, Dale R, Petrillo, Daniel E, Reif, James J, Gingrich, Diane E, Bakale, Roger P

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