Evolution of Novartis’ Small Molecule Screening Deck Design von Schuffenhauer, Ansgar, Schneider, Nadine, Hintermann, Samuel, Auld, Douglas, Blank, Jutta, Cotesta, Simona, Engeloch, Caroline, Fechner, Nikolas, Gaul, Christoph, Giovannoni, Jerome, Jansen, Johanna, Joslin, John, Krastel, Philipp, Lounkine, Eugen, Manchester, John, Monovich, Lauren G, Pelliccioli, Anna Paola, Schwarze, Manuel, Shultz, Michael D, Stiefl, Nikolaus, Baeschlin, Daniel K

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Systematic Chemogenetic Library Assembly von Canham, Stephen M., Wang, Yuan, Cornett, Allen, Auld, Douglas S., Baeschlin, Daniel K., Patoor, Maude, Skaanderup, Philip R., Honda, Ayako, Llamas, Luis, Wendel, Greg, Mapa, Felipa A., Aspesi, Peter, Labbé-Giguère, Nancy, Gamber, Gabriel G., Palacios, Daniel S., Schuffenhauer, Ansgar, Deng, Zhan, Nigsch, Florian, Frederiksen, Mathias, Bushell, Simon M., Rothman, Deborah, Jain, Rishi K., Hemmerle, Horst, Briner, Karin, Porter, Jeffery A., Tallarico, John A., Jenkins, Jeremy L.

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Discovery of C-(1-aryl-cyclohexyl)-methylamines as selective, orally available inhibitors of dipeptidyl peptidase IV von Namoto, Kenji, Sirockin, Finton, Ostermann, Nils, Gessier, Francois, Flohr, Stefanie, Sedrani, Richard, Gerhartz, Bernd, Trappe, Jörg, Hassiepen, Ulrich, Duttaroy, Alokesh, Ferreira, Suzie, Sutton, Jon M., Clark, David E., Fenton, Garry, Beswick, Mandy, Baeschlin, Daniel K.

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Novel heterocyclic DPP-4 inhibitors for the treatment of type 2 diabetes von Sutton, Jon M., Clark, David E., Dunsdon, Stephen J., Fenton, Garry, Fillmore, Amanda, Harris, Neil V., Higgs, Chris, Hurley, Chris A., Krintel, Sussie L., MacKenzie, Robert E., Duttaroy, Alokesh, Gangl, Eric, Maniara, Wiesia, Sedrani, Richard, Namoto, Kenji, Ostermann, Nils, Gerhartz, Bernd, Sirockin, Finton, Trappe, Jörg, Hassiepen, Ulrich, Baeschlin, Daniel K.

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Concise Asymmetric Syntheses of Radicicol and Monocillin I von Garbaccio, Robert M, Stachel, Shawn J, Baeschlin, Daniel K, Danishefsky, Samuel J

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Fostering Research Synergies between Chemists in Swiss Academia and at Novartis von Meyer, Arndt, Baeschlin, Daniel, Brocklehurst, Cara E., Duckely, Myriam, Gallou, Fabrice, Lovelle, Lucie E., Parmentier, Michael, Schlama, Thierry, Snajdrova, Radka, Auberson, Yves P.

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1,2-Diacetals:  A New Opportunity for Organic Synthesis von Ley, Steven V, Baeschlin, Daniel K, Dixon, Darren J, Foster, Alison C, Ince, Stuart J, Priepke, Henning W. M, Reynolds, Dominic J

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A Novel Class of Oral Direct Renin Inhibitors: Highly Potent 3,5-Disubstituted Piperidines Bearing a Tricyclic P3 –P1 Pharmacophore von Ostermann, Nils, Ruedisser, Simon, Ehrhardt, Claus, Breitenstein, Werner, Marzinzik, Andreas, Jacoby, Edgar, Vangrevelinghe, Eric, Ottl, Johannes, Klumpp, Martin, Hartwieg, J. Constanze D, Cumin, Frederic, Hassiepen, Ulrich, Trappe, Jörg, Sedrani, Richard, Geisse, Sabine, Gerhartz, Bernd, Richert, Paul, Francotte, Eric, Wagner, Trixie, Krömer, Markus, Kosaka, Takatoshi, Webb, Randy L, Rigel, Dean F, Maibaum, Jürgen, Baeschlin, Daniel K

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5-Fluorouracil blocks quorum-sensing of biofilm-embedded methicillin-resistant Staphylococcus aureus in mice von Sedlmayer, Ferdinand, Woischnig, Anne-Kathrin, Unterreiner, Vincent, Fuchs, Florian, Baeschlin, Daniel, Khanna, Nina, Fussenegger, Martin

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A Scalable Synthesis of an Azabicyclooctanyl Derivative, a Novel DPP-4 Inhibitor von Fei, Zhongbo, Wu, Quanbing, Zhang, Fei, Cao, Yudong, Liu, Chuanqin, Shieh, Wen-Chung, Xue, Song, McKenna, Joe, Prasad, Kapa, Prashad, Mahavir, Baeschlin, Daniel, Namoto, Kenji

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Structure–activity relationship in the oxazolidinone–quinolone hybrid series: influence of the central spacer on the antibacterial activity and the mode of action von Hubschwerlen, Christian, Specklin, Jean-Luc, Baeschlin, Daniel K., Borer, Yves, Haefeli, Sascha, Sigwalt, Christine, Schroeder, Susanne, Locher, Hans H.

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Rapid assembly of oligosaccharides: 1,2-diacetal-mediated reactivity tuning in the coupling of glycosyl fluorides von Baeschlin, Daniel K, Green, Luke G, Hahn, Michael G, Hinzen, Berthold, Ince, Stuart J, Ley, Steven V

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Rapid Assembly of Oligosaccharides: Total Synthesis of a Glycosylphosphatidylinositol Anchor of Trypanosoma brucei von Baeschlin, Daniel K., Chaperon, André R., Charbonneau, Virginie, Green, Luke G., Ley, Steven V., Lücking, Ulrich, Walther, Eric

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A high-throughput drug screen reveals means to differentiate triple-negative breast cancer von Vulin, Milica, Jehanno, Charly, Sethi, Atul, Correia, Ana Luísa, Obradović, Milan M. S., Couto, Joana Pinto, Coissieux, Marie-May, Diepenbruck, Maren, Preca, Bogdan-Tiberius, Volkmann, Katrin, der Maur, Priska Auf, Schmidt, Alexander, Münst, Simone, Sauteur, Loïc, Kloc, Michal, Palafox, Marta, Britschgi, Adrian, Unterreiner, Vincent, Galuba, Olaf, Claerr, Isabelle, Lopez-Romero, Sandra, Galli, Giorgio G., Baeschlin, Daniel, Okamoto, Ryoko, Soysal, Savas D., Mechera, Robert, Weber, Walter P., Radimerski, Thomas, Bentires-Alj, Mohamed

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Identification of a Novel N-Carbamoyl Glucuronide: In Vitro, In Vivo, and Mechanistic Studies von GUNDUZ, Mithat, ARGIKAR, Upendra A, BAESCHLIN, Daniel, FERREIRA, Suzie, HOSAGRAHARA, Vinayak, HARRIMAN, Shawn

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A Novel Class of Oral Direct Renin Inhibitors: Highly Potent 3,5-Disubstituted Piperidines Bearing a Tricyclic P 3 – P 1 Pharmacophore von Ostermann, Nils, Ruedisser, Simon, Ehrhardt, Claus, Breitenstein, Werner, Marzinzik, Andreas, Jacoby, Edgar, Vangrevelinghe, Eric, Ottl, Johannes, Klumpp, Martin, Hartwieg, J. Constanze D., Cumin, Frederic, Hassiepen, Ulrich, Trappe, Jörg, Sedrani, Richard, Geisse, Sabine, Gerhartz, Bernd, Richert, Paul, Francotte, Eric, Wagner, Trixie, Krömer, Markus, Kosaka, Takatoshi, Webb, Randy L., Rigel, Dean F., Maibaum, Jürgen, Baeschlin, Daniel K.

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Chimera of Dimethylene Sulfone-, Methyl Sulfide-, and Methyl Sulfoxide-Linked Ribonucleotides and DNA von Baeschlin, Daniel K, Hyrup, Birgitte, Benner, Steven A, Richert, Clemens

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1,2-Diacetals in Synthesis: Total Synthesis of a Glycosylphosphatidylinositol Anchor of Trypanosoma brucei von Baeschlin, Daniel K., Chaperon, André R., Green, Luke G., Hahn, Michael G., Ince, Stuart J., Ley, Steven V.

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Erratum to “Novel heterocyclic DPP-4 inhibitors for the treatment of type 2 diabetes” [Bioorg. Med. Chem. Lett. 22 (2012) 1464–1468] von Sutton, Jon M., Clark, David E., Dunsdon, Stephen J., Fenton, Garry, Fillmore, Amanda, Harris, Neil V., Higgs, Chris, Hurley, Chris A., Krintel, Sussie L., MacKenzie, Robert E., Duttaroy, Alokesh, Gangl, Eric, Maniara, Wiesia, Sedrani, Richard, Namoto, Kenji, Ostermann, Nils, Gerhartz, Bernd, Sirockin, Finton, Trappe, Jörg, Hassiepen, Ulrich, Baeschlin, Daniel K.

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1,2-Diacetals in Synthesis: Total Synthesis of a Glycosylphosphatidylinositol Anchor ofTrypanosoma brucei von Baeschlin, Daniel K., Chaperon, André R., Green, Luke G., Hahn, Michael G., Ince, Stuart J., Ley, Steven V.

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