A Novel Oral Arginase 1/2 Inhibitor Enhances the Antitumor Effect of PD-1 Inhibition in Murine Experimental Gliomas by Altering the Immunosuppressive Environment von Pilanc, Paulina, Wojnicki, Kamil, Roura, Adria-Jaume, Cyranowski, Salwador, Ellert-Miklaszewska, Aleksandra, Ochocka, Natalia, Gielniewski, Bartlomiej, Grzybowski, Marcin M., Blaszczyk, Roman, Stanczak, Paulina S., Dobrzanski, Pawel, Kaminska, Bozena

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OATD-02 Validates the Benefits of Pharmacological Inhibition of Arginase 1 and 2 in Cancer von Grzybowski, Marcin Mikołaj, Stańczak, Paulina Seweryna, Pomper, Paulina, Błaszczyk, Roman, Borek, Bartłomiej, Gzik, Anna, Nowicka, Julita, Jędrzejczak, Karol, Brzezińska, Joanna, Rejczak, Tomasz, Güner-Chalimoniuk, Nazan Cemre, Kikulska, Agnieszka, Mlącki, Michał, Pęczkowicz-Szyszka, Jolanta, Olczak, Jacek, Gołębiowski, Adam, Dzwonek, Karolina, Dobrzański, Paweł, Zasłona, Zbigniew

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Comparative analysis of RNA 3D structure prediction methods: towards enhanced modeling of RNA–ligand interactions von Nithin, Chandran, Kmiecik, Sebastian, Błaszczyk, Roman, Nowicka, Julita, Tuszyńska, Irina

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Boronic acid-based arginase inhibitors in cancer immunotherapy von Borek, Bartlomiej, Gajda, Tadeusz, Golebiowski, Adam, Blaszczyk, Roman

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Small extracellular vesicles containing arginase-1 suppress T-cell responses and promote tumor growth in ovarian carcinoma von Czystowska-Kuzmicz, Malgorzata, Sosnowska, Anna, Nowis, Dominika, Ramji, Kavita, Szajnik, Marta, Chlebowska-Tuz, Justyna, Wolinska, Ewa, Gaj, Pawel, Grazul, Magdalena, Pilch, Zofia, Zerrouqi, Abdessamad, Graczyk-Jarzynka, Agnieszka, Soroczynska, Karolina, Cierniak, Szczepan, Koktysz, Robert, Elishaev, Esther, Gruca, Slawomir, Stefanowicz, Artur, Blaszczyk, Roman, Borek, Bartlomiej, Gzik, Anna, Whiteside, Theresa, Golab, Jakub

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HPLC with Post-Column Derivatization with Alizarin for Determination of OATD-02, an Anticancer Arginase Inhibitor in Clinical Development von Sobolewska, Elzbieta, Tyszkiewicz, Magdalena, Blaszczyk, Roman, Biesaga, Magdalena

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Inhibition of arginase modulates T-cell response in the tumor microenvironment of lung carcinoma von Sosnowska, Anna, Chlebowska-Tuz, Justyna, Matryba, Pawel, Pilch, Zofia, Greig, Alan, Wolny, Artur, Grzywa, Tomasz M., Rydzynska, Zuzanna, Sokolowska, Olga, Rygiel, Tomasz P., Grzybowski, Marcin, Stanczak, Paulina, Blaszczyk, Roman, Nowis, Dominika, Golab, Jakub

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Direct synthesis of protected diethyl 1,2-diaminoalkylphosphonates von Błaszczyk, Roman, Gajda, Tadeusz

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Differentiation of Diastereoisomers of Protected 1,2-Diaminoalkylphosphonic Acids by EI Mass Spectrometry and Density Functional Theory von Drabik, Ewelina, Krasiński, Grzegorz, Cypryk, Marek, Błaszczyk, Roman, Gajda, Tadeusz, Sochacki, Marek

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Potent but transient immunosuppression of T-cells is a general feature of CD71+ erythroid cells von Grzywa, Tomasz M., Sosnowska, Anna, Rydzynska, Zuzanna, Lazniewski, Michal, Plewczynski, Dariusz, Klicka, Klaudia, Malecka-Gieldowska, Milena, Rodziewicz-Lurzynska, Anna, Ciepiela, Olga, Justyniarska, Magdalena, Pomper, Paulina, Grzybowski, Marcin M., Blaszczyk, Roman, Wegrzynowicz, Michal, Tomaszewska, Agnieszka, Basak, Grzegorz, Golab, Jakub, Nowis, Dominika

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Stereochemical effects in fragmentation of diastereoisomers of protected diethyl 1,2-diamino-alkylphosphonates von Drabik, Ewelina, Błaszczyk, Roman, Gajda, Tadeusz, Sochacki, Marek

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N-Carbamate α-aminoalkyl- p-tolylsulfones - Convenient substrates in the nitro-Mannich synthesis of secondary N-carbamate protected syn-2-amino-1-nitroalkanephosphonates von Błaszczyk, Roman, Gajda, Anna, Zawadzki, Stefan, Czubacka, Ewelina, Gajda, Tadeusz

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Reaction of diethyl thiocyanatomethylphosphonate with aldehydes as a route to diethyl Z-1-alkenylphosphonates von Błaszczyk, Roman, Gajda, Tadeusz

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Stereochemical effects in fragmentation of diastereoisomers of protected diethyl 1,2-diamino-alkylphosphonates: Fragmentation of protected diethyl 1,2-diaminoalkylphosphonates von Drabik, Ewelina, Błaszczyk, Roman, Gajda, Tadeusz, Sochacki, Marek

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Novel orally bioavailable piperidine derivatives as extracellular arginase inhibitors developed by a ring expansion von Gzik, Anna, Borek, Bartlomiej, Chrzanowski, Jacek, Jedrzejczak, Karol, Dziegielewski, Marek, Brzezinska, Joanna, Nowicka, Julita, Grzybowski, Marcin M, Rejczak, Tomasz, Niedzialek, Dorota, Wieczorek, Grzegorz, Olczak, Jacek, Golebiowski, Adam, Zaslona, Zbigniew, Blaszczyk, Roman

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Discovery and Pharmacokinetics of Sulfamides and Guanidines as Potent Human Arginase 1 Inhibitors von Blaszczyk, Roman, Brzezinska, Joanna, Dymek, Barbara, Stanczak, Paulina S, Mazurkiewicz, Marcin, Olczak, Jacek, Nowicka, Julita, Dzwonek, Karolina, Zagozdzon, Agnieszka, Golab, Jakub, Golebiowski, Adam

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Arginase 1/2 Inhibitor OATD-02: From Discovery to First-in-man Setup in Cancer Immunotherapy von Borek, Bartlomiej, Nowicka, Julita, Gzik, Anna, Dziegielewski, Marek, Jedrzejczak, Karol, Brzezinska, Joanna, Grzybowski, Marcin, Stanczak, Paulina, Pomper, Paulina, Zagozdzon, Agnieszka, Rejczak, Tomasz, Matyszewski, Krzysztof, Golebiowski, Adam, Olczak, Jacek, Lisiecki, Kamil, Tyszkiewicz, Magdalena, Kania, Magdalena, Piasecka, Sylwia, Cabaj, Anna, Dera, Paulina, Mulewski, Krzysztof, Chrzanowski, Jacek, Kusmirek, Damian, Sobolewska, Elzbieta, Magdycz, Marta, Mucha, Lukasz, Masnyk, Marek, Golab, Jakub, Nowotny, Marcin, Nowak, Elzbieta, Napiorkowska-Gromadzka, Agnieszka, Pikul, Stanislaw, Jazwiec, Radoslaw, Dzwonek, Karolina, Dobrzanski, Pawel, Meyring, Michael, Skowronek, Krzysztof, Iwanowski, Piotr, Zaslona, Zbigniew, Blaszczyk, Roman

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Comparative analysis of RNA 3D structure prediction methods: towards enhanced modeling of RNA-Ligand interactions von C, NITHIN

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Comparative analysis of RNA 3D structure prediction methods: towards enhanced modeling of RNA-Ligand interactions von C, NITHIN

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Comparative analysis of RNA 3D structure prediction methods: towards enhanced modeling of RNA-Ligand interactions von C, NITHIN

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