Importance of the Azole Moiety of Cimetidine Derivatives for the Inhibition of Human Multidrug and Toxin Extrusion Transporter 1 (hMATE1) von Shinya, Susumu, Kawai, Kentaro, Tarui, Atsushi, Karuo, Yukiko, Sato, Kazuyuki, Matsuda, Masaya, Kitatani, Kazuyuki, Kobayashi, Naoki, Nabe, Takeshi, Otsuka, Masato, Omote, Masaaki

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Identification and Synthesis of DDI-6, a Quinolinol Analog Capable of Activating Both Caenorhabditis elegans and Mouse Spermatozoa von Karuo, Yukiko, Shiraki, Riona, Yoshida, Ayaka, Tsunokawa, Ryo, Nakahara-Yamada, Mayuko, Tarui, Atsushi, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki, Nishimura, Hitoshi

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Development of Drug Discovery Platforms Using Artificial Intelligence and Cheminformatics von Kawai, Kentaro, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Kataoka, Makoto, Omote, Masaaki

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Pentafluorosulfanyl-substituted biaryl derivatives as MATE-type transporter inhibitors targeting drug-resistant bacteria von Shinya, Susumu, Kawai, Kentaro, Kobayashi, Naoki, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Otsuka, Masato, Omote, Masaaki

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Synthesis of fluoroalkenes and fluoroenynes via cross-coupling reactions using novel multihalogenated vinyl ethers von Karuo, Yukiko, Hirata, Keita, Tarui, Atsushi, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki

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Fluorophenylalkyl-substituted cyanoguanidine derivatives as bacteria-selective MATE transporter inhibitors for the treatment of antibiotic-resistant infections von Shinya, Susumu, Kawai, Kentaro, Kobayashi, Naoki, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Otsuka, Masato, Omote, Masaaki

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Rhodium-catalyzed homo-coupling reaction of aryl Grignard reagents and its application for the synthesis of an integrin inhibitor von Sato, Kazuyuki, Teranishi, Satoki, Sakaue, Atsushi, Karuo, Yukiko, Tarui, Atsushi, Kawai, Kentaro, Takeda, Hiroyuki, Kinashi, Tatsuo, Omote, Masaaki

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Synthesis of aryl 2-bromo-2-chloro-1,1-difluoroethyl ethers through the base-mediated reaction between phenols and halothane von Karuo, Yukiko, Kametani, Ayaka, Tarui, Atsushi, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki

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Synthesis of new fluorescent molecules having an aggregation-induced emission property derived from 4-fluoroisoxazoles von Sato, Kazuyuki, Kawasaki, Akira, Karuo, Yukiko, Tarui, Atsushi, Kawai, Kentaro, Omote, Masaaki

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LCP: Simple Representation of Docking Poses for Machine Learning: A Case Study on Xanthine Oxidase Inhibitors von Kawai, Kentaro, Asanuma, Yoshitaka, Kato, Toshiki, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Omote, Masaaki

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Effect of Structural Descriptors on the Design of Cyclin Dependent Kinase Inhibitors Using Similarity‐based Molecular Evolution von Kawai, Kentaro, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Omote, Masaaki

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Decarboxylative Aldol Reaction of α,α-Difluoro-β-keto Esters: Easy Access to Difluoroenolate von Tarui, Atsushi, Shimomura, Hiroshi, Yasuno, Yohei, Karuo, Yukiko, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki

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Ligand-Promoted Asymmetric Imino-Reformatsky Reaction of Ethyl Dibromofluoroacetate von Tarui, Atsushi, Nishimura, Haruka, Ikebata, Takeshi, Tahira, Asuka, Sato, Kazuyuki, Omote, Masaaki, Minami, Hideki, Miwa, Yoshihisa, Ando, Akira

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Synthesis of Small Fluorescent Molecules and Evaluation of Photophysical Properties von Ogawa, Futa, Karuo, Yukiko, Yamazawa, Ryuji, Miyanaga, Kanae, Hori, Kazushige, Tani, Keita, Yamada, Kengo, Saito, Yuki, Funabiki, Kazumasa, Tarui, Atsushi, Sato, Kazuyuki, Ito, Kiyoshi, Kawai, Kentaro, Omote, Masaaki

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Synthesis of 2,2-difluoro-2-arylethylamines as fluorinated analogs of octopamine and noradrenaline

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Synthesis of 2-aryl-3-trifluoromethylquinolines using (E)-trimethyl(3,3,3-trifluoroprop-1-enyl)silane von Omote, Masaaki, Tanaka, Miyuu, Tanaka, Miki, Ikeda, Akari, Tarui, Atsushi, Sato, Kazuyuki, Ando, Akira

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Development of a fluorogenic small substrate for dipeptidyl peptidase-4 von Ogawa, Futa, Takeda, Masanori, Miyanaga, Kanae, Tani, Keita, Yamazawa, Ryuji, Ito, Kiyoshi, Tarui, Atsushi, Sato, Kazuyuki, Omote, Masaaki

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Rh-Catalyzed reductive Mannich-type reaction and its application towards the synthesis of (±)-ezetimibe von Isoda, Motoyuki, Sato, Kazuyuki, Kunugi, Yurika, Tokonishi, Satsuki, Tarui, Atsushi, Omote, Masaaki, Minami, Hideki, Ando, Akira

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Diastereoselective synthesis of 2-fluoroaziridine-2-carboxylates by Reformatsky-type aza-Darzens reaction von Tarui, Atsushi, Kawashima, Naoto, Sato, Kazuyuki, Omote, Masaaki, Ando, Akira

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Asymmetric Reductive Aldol-Type Reaction with Carbonyl Compounds Using Dialkyl Tartrate as a Chiral Ligand von Isoda, Motoyuki, Sato, Kazuyuki, Tokura, Yoriko, Tarui, Atsushi, Omote, Masaaki, Ando, Akira

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