Using Triethynylphosphine Ligands Bearing Bulky End Caps To Create a Holey Catalytic Environment:  Application to Gold(I)-Catalyzed Alkyne Cyclizations von Ochida, Atsuko, Ito, Hideto, Sawamura, Masaya

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Discovery and Structure–Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious Antimalarials von Laleu, Benoît, Akao, Yuichiro, Ochida, Atsuko, Duffy, Sandra, Lucantoni, Leonardo, Shackleford, David M, Chen, Gong, Katneni, Kasiram, Chiu, Francis C. K, White, Karen L, Chen, Xue, Sturm, Angelika, Dechering, Koen J, Crespo, Benigno, Sanz, Laura M, Wang, Binglin, Wittlin, Sergio, Charman, Susan A, Avery, Vicky M, Cho, Nobuo, Kamaura, Masahiro

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Monocoordinating, Compact Phosphane Immobilized on Silica Surface: Application to Rhodium-Catalyzed Hydrosilylation of Hindered Ketones von Hamasaka, Go, Ochida, Atsuko, Hara, Kenji, Sawamura, Masaya

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Electronically Tunable Compact Trialkylphosphines: SMAPs-bridged Bicyclic Phosphines von Ochida, Atsuko, Ito, Shinichiro, Miyahara, Takahiro, Ito, Hajime, Sawamura, Masaya

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Synthesis, Properties, and Catalytic Applications of Caged, Compact Trialkylphosphine 4-Phenyl-1-phospha-4-silabicyclo[2.2.2]octane von Ochida, Atsuko, Hamasaka, Go, Yamauchi, Yoshihiro, Kawamorita, Soichiro, Oshima, Naoya, Hara, Kenji, Ohmiya, Hirohisa, Sawamura, Masaya

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顧みられない熱帯病に対するパートナーシップ活動 von 赤尾, 雄一郎, 落田, 温子, 村西, 廣哉, 野村, 泉, 一川, 隆史

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Nonvolatile Me3P-like P-Donor Ligand:  Synthesis and Properties of 4-Phenyl-1-phospha-4-silabicyclo[2.2.2]octane von Ochida, Atsuko, Hara, Kenji, Ito, Hajime, Sawamura, Masaya

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Partnership Activity for Neglected Tropical Diseases von Akao, Yuichiro, Ochida, Atsuko, Muranishi, Hiroya, Nomura, Izumi, Ichikawa, Takashi

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Phosphorus Ligands with a Large Cavity: Synthesis of Triethynylphosphines with Bulky End Caps and Application to the Rhodium-Catalyzed Hydrosilylation of Ketones von Ochida, Atsuko, Sawamura, Masaya

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Pharmacological inhibitory profile of TAK-828F, a potent and selective orally available RORγt inverse agonist von Shibata, Akira, Uga, Keiko, Sato, Takayuki, Sagara, Masaki, Igaki, Keiko, Nakamura, Yoshiki, Ochida, Atsuko, Kono, Mitsunori, Shirai, Junya, Yamamoto, Satoshi, Yamasaki, Masashi, Tsuchimori, Noboru

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Discovery of [cis-3-({(5R)‑5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro‑1H‑inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5H)‑yl}carbonyl)­cyclobutyl]­acetic Acid (TAK-828... von Kono, Mitsunori, Ochida, Atsuko, Oda, Tsuneo, Imada, Takashi, Banno, Yoshihiro, Taya, Naohiro, Masada, Shinichi, Kawamoto, Tetsuji, Yonemori, Kazuko, Nara, Yoshi, Fukase, Yoshiyuki, Yukawa, Tomoya, Tokuhara, Hidekazu, Skene, Robert, Sang, Bi-Ching, Hoffman, Isaac D, Snell, Gyorgy P, Uga, Keiko, Shibata, Akira, Igaki, Keiko, Nakamura, Yoshiki, Nakagawa, Hideyuki, Tsuchimori, Noboru, Yamasaki, Masashi, Shirai, Junya, Yamamoto, Satoshi

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Nonbisphosphonate inhibitors of Plasmodium falciparum FPPS/GGPPS von Kabeche, Stephanie, Aida, Jumpei, Akther, Thamina, Ichikawa, Takashi, Ochida, Atsuko, Pulkoski-Gross, Michael J., Smith, Mark, Humphries, Paul S., Yeh, Ellen

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Synthesis and properties of SMAPs 1-phospha-4-silabicyclo[2.2.2]octane derivatives von Ochida, Atsuko, Sawamura, Masaya

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Cyclization of Nonterminal Alkynic β-Keto Esters Catalyzed by Gold(I) Complex with a Semihollow, End-Capped Triethynylphosphine Ligand von Ito, Hideto, Makida, Yusuke, Ochida, Atsuko, Ohmiya, Hirohisa, Sawamura, Masaya

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Collaborative Virtual Screening Identifies a 2‑Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi Infection von Tawaraishi, Taisuke, Ochida, Atsuko, Akao, Yuichiro, Itono, Sachiko, Kamaura, Masahiro, Akther, Thamina, Shimada, Mitsuyuki, Canan, Stacie, Chowdhury, Sanjoy, Cao, Yafeng, Condroski, Kevin, Engkvist, Ola, Francisco, Amanda, Ghosh, Sunil, Kaki, Rina, Kelly, John M., Kimura, Chiaki, Kogej, Thierry, Nagaoka, Kazuya, Naito, Akira, Pairaudeau, Garry, Radu, Constantin, Roberts, Ieuan, Shum, David, Watanabe, Nao-aki, Xie, Huanxu, Yonezawa, Shuji, Yoshida, Osamu, Yoshida, Ryu, Mowbray, Charles, Perry, Benjamin

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Collaborative Virtual Screening Identifies a 2-Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi Infection von Tawaraishi, Taisuke, Ochida, Atsuko, Akao, Yuichiro, Itono, Sachiko, Kamaura, Masahiro, Akther, Thamina, Shimada, Mitsuyuki, Canan, Stacie, Chowdhury, Sanjoy, Cao, Yafeng, Condroski, Kevin, Engkvist, Ola, Francisco, Amanda, Ghosh, Sunil, Kaki, Rina, Kelly, John M, Kimura, Chiaki, Kogej, Thierry, Nagaoka, Kazuya, Naito, Akira, Pairaudeau, Garry, Radu, Constantin, Roberts, Ieuan, Shum, David, Watanabe, Nao-Aki, Xie, Huanxu, Yonezawa, Shuji, Yoshida, Osamu, Yoshida, Ryu, Mowbray, Charles, Perry, Benjamin

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Identification of novel quinazolinedione derivatives as RORγt inverse agonist von Fukase, Yoshiyuki, Sato, Ayumu, Tomata, Yoshihide, Ochida, Atsuko, Kono, Mitsunori, Yonemori, Kazuko, Koga, Keiko, Okui, Toshitake, Yamasaki, Masashi, Fujitani, Yasushi, Nakagawa, Hideyuki, Koyama, Ryoukichi, Nakayama, Masaharu, Skene, Robert, Sang, Bi-Ching, Hoffman, Isaac, Shirai, Junya, Yamamoto, Satoshi

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Optimization of Methionyl tRNA-Synthetase Inhibitors for Treatment of Cryptosporidium Infection von Buckner, Frederick S, Ranade, Ranae M, Gillespie, J Robert, Shibata, Sayaka, Hulverson, Matthew A, Zhang, Zhongsheng, Huang, Wenlin, Choi, Ryan, Verlinde, Christophe L M J, Hol, Wim G J, Ochida, Atsuko, Akao, Yuichiro, Choy, Robert K M, Van Voorhis, Wesley C, Arnold, Sam L M, Jumani, Rajiv S, Huston, Christopher D, Fan, Erkang

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Discovery of orally efficacious RORγt inverse agonists. Part 2: Design, synthesis, and biological evaluation of novel tetrahydroisoquinoline derivatives von Kono, Mitsunori, Oda, Tsuneo, Tawada, Michiko, Imada, Takashi, Banno, Yoshihiro, Taya, Naohiro, Kawamoto, Tetsuji, Tokuhara, Hidekazu, Tomata, Yoshihide, Ishii, Naoki, Ochida, Atsuko, Fukase, Yoshiyuki, Yukawa, Tomoya, Fukumoto, Shoji, Watanabe, Hiroyuki, Uga, Keiko, Shibata, Akira, Nakagawa, Hideyuki, Shirasaki, Mikio, Fujitani, Yasushi, Yamasaki, Masashi, Shirai, Junya, Yamamoto, Satoshi

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Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffolds von Shirai, Junya, Tomata, Yoshihide, Kono, Mitsunori, Ochida, Atsuko, Fukase, Yoshiyuki, Sato, Ayumu, Masada, Shinichi, Kawamoto, Tetsuji, Yonemori, Kazuko, Koyama, Ryoukichi, Nakagawa, Hideyuki, Nakayama, Masaharu, Uga, Keiko, Shibata, Akira, Koga, Keiko, Okui, Toshitake, Shirasaki, Mikio, Skene, Robert, Sang, BiChing, Hoffman, Isaac, Lane, Wes, Fujitani, Yasushi, Yamasaki, Masashi, Yamamoto, Satoshi

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