Dose Number as a Tool to Guide Lead Optimization for Orally Bioavailable Compounds in Drug Discovery von Wuelfing, W. Peter, El Marrouni, Abdellatif, Lipert, Maya P, Daublain, Pierre, Kesisoglou, Filippos, Converso, Antonella, Templeton, Allen C

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Synthesis of HIV NNRTI Doravirine Analogues via Visible-Light Photoredox Decarboxylative Cross-Coupling von Suen, Linda M., Wang, Cheng, Hunter, David N., Mitchell, Helen J., Converso, Antonella, ElMarrouni, Abdellatif

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Development of a sp2–sp3 Stille Cross-Coupling for Rapid Synthesis of HIV NNRTI Doravirine Analogues von ElMarrouni, Abdellatif, Campbell, Mark, Perkins, James J, Converso, Antonella

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Comparison of amine additives most effective in the new methyltrioxorhenium-catalyzed epoxidation process von Adolfsson, Hans, Converso, Antonella, Sharpless, K.Barry

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Development of a sp 2 -sp 3 Stille Cross-Coupling for Rapid Synthesis of HIV NNRTI Doravirine Analogues von ElMarrouni, Abdellatif, Campbell, Mark, Perkins, James J, Converso, Antonella

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Studies toward the Synthesis of Azadirachtin, Part 2: Construction of Fully Functionalized ABCD Ring Frameworks and Unusual Intramolecular Reactions Induced by Close-Proximity Effe... von Nicolaou, K. C., Sasmal, Pradip K., Koftis, Theocharis V., Converso, Antonella, Loizidou, Eriketi, Kaiser, Florian, Roecker, A. J., Dellios, Constantinos C., Sun, Xiao-Wen, Petrovic, Goran

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Simple and efficient routes for the preparation of isoxazolidinyl nucleosides containing cytosine and 5-methyl-cytosine as new potential anti-HIV drugs von Colacino, Evelina, Converso, Antonella, Liguori, Angelo, Napoli, Anna, Siciliano, Carlo, Sindona, Giovanni

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2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: multigram display of azide and cyanide components on a versatile scaffold von Díaz, David Díaz, Converso, Antonella, Sharpless, K Barry, Finn, M G

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Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity von Wang, Cheng, Adam, Gregory C., Burlein, Christine, Carroll, Steven, Dankulich, William, Diamond, Tracy, Grobler, Jay, Heath, Jeffrey, Johnson, Adam, Klein, Daniel, Krosky, Daniel, Narayan, Kartik, Ou, Yangsi, Sanders, John, Sharma, Sujata, Xu, Min, Converso, Antonella

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Augmenting Hit Identification by Virtual Screening Techniques in Small Molecule Drug Discovery von Yan, Xin Cindy, Sanders, John M, Gao, Ying-Duo, Tudor, Matthew, Haidle, Andrew M, Klein, Daniel J, Converso, Antonella, Lesburg, Charles A, Zang, Yi, Wood, Harold B

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A Phenotypic Screen Identifies Potent DPP9 Inhibitors Capable of Killing HIV‑1 Infected Cells von Moore, Keith P., Schwaid, Adam G., Tudor, Matthew, Park, Sangho, Beshore, Douglas C., Converso, Antonella, Shipe, William D., Anand, Rajan, Lan, Ping, Moningka, Remond, Rothman, Deborah M., Sun, Wanying, Chi, An, Cornella-Taracido, Ivan, Adam, Gregory C., Bahnck-Teets, Carolyn, Carroll, Steven S., Fay, John F., Goh, Shih Lin, Lusen, Jeffrey, Quan, Shuo, Rodriguez, Silveria, Xu, Min, Andrews, Christine L., Song, Cheng, Filzen, Tracey, Li, Jing, Hollenstein, Kaspar, Klein, Daniel J., Lammens, Alfred, Lim, U-Ming, Fang, Zhiyu, McHale, Carolyn, Li, Yuan, Lu, Meiqing, Diamond, Tracy L., Howell, Bonnie J., Zuck, Paul, Balibar, Carl J.

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Discovery of 4-arylquinoline-2-carboxamides, highly potent and selective class of mGluR2 negative allosteric modulators: From HTS to activity in animal models von Shu, Youheng, Diamond, Tracy L., Hershey, James C., Huang, Shaei, Magliaro, Brian C., O'Brien, Julie A., Schlegel, Kelly-Ann S., Puri, Vanita, Uebele, Victor N., Uslaner, Jason M., Wang, Cheng, Converso, Antonella

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Nucleophilic Substitution by Grignard Reagents on Sulfur Mustards von Converso, Antonella, Saaidi, Pierre-Loïc, Sharpless, K. Barry, Finn, M. G

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Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator von Rudd, Michael T., Manley, Peter J., Hanney, Barbara, Meng, Zhaoyang, Shu, Youheng, de Leon, Pablo, Frie, Jessica L., Han, Yongxin, Wai, Jenny Miu-Chun, Yang, Zhi-Qiang, Perkins, James J., Hurzy, Danielle M., Manikowski, Jesse J., Zhu, Hong, Bungard, Christopher J., Converso, Antonella, Meissner, Robert S., Cosden, Mali L., Hayashi, Ikuo, Ma, Lei, O’Brien, Julie, Uebele, Victor N., Schachter, Joel B., Bhandari, Neetesh, Ward, Gwendolyn J., Fillgrove, Kerry L., Lu, Bing, Liang, Yuexia, Dubost, David C., Puri, Vanita, Eddins, Donnie M., Vardigan, Joshua D., Drolet, Robert E., Kern, Jonathan T., Uslaner, Jason M.

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Discovery of a Distinct Chemical and Mechanistic Class of Allosteric HIV‑1 Integrase Inhibitors with Antiretroviral Activity von Burlein, Christine, Wang, Cheng, Xu, Min, Bhatt, Triveni, Stahlhut, Mark, Ou, Yangsi, Adam, Gregory C, Heath, Jeffrey, Klein, Daniel J, Sanders, John, Narayan, Kartik, Abeywickrema, Pravien, Heo, Mee Ra, Carroll, Steven S, Grobler, Jay A, Sharma, Sujata, Diamond, Tracy L, Converso, Antonella, Krosky, Daniel J

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2,6-Dichloro-9-thiabicyclo[3.3.1]nonane:  A Privileged, Bivalent Scaffold for the Display of Nucleophilic Components von Converso, Antonella, Burow, Kristina, Marzinzik, Andreas, Sharpless, K. Barry, Finn, M. G

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Analysis of T-cell clones in systemic lupus erythematosus von Converso, M, Bertero, MT, Vallario, A, Caligaris-Cappio, F

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Kinetic Analysis of Membrane Potential Dye Response to NaV1.7 Channel Activation Identifies Antagonists with Pharmacological Selectivity against NaV1.5 von Finley, Michael, Cassaday, Jason, Kreamer, Tony, Li, Xinnian, Solly, Kelli, O’Donnell, Greg, Clements, Michelle, Converso, Antonella, Cook, Sean, Daley, Chris, Kraus, Richard, Lai, Ming-Tain, Layton, Mark, Lemaire, Wei, Staas, Donnette, Wang, Jixin

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Development of thioquinazolinones, allosteric Chk1 kinase inhibitors von Converso, Antonella, Hartingh, Timothy, Garbaccio, Robert M., Tasber, Edward, Rickert, Keith, Fraley, Mark E., Yan, Youwei, Kreatsoulas, Constantine, Stirdivant, Steve, Drakas, Bob, Walsh, Eileen S., Hamilton, Kelly, Buser, Carolyn A., Mao, Xianzhi, Abrams, Marc T., Beck, Stephen C., Tao, Weikang, Lobell, Rob, Sepp-Lorenzino, Laura, Zugay-Murphy, Joan, Sardana, Vinod, Munshi, Sanjeev K., Jezequel-Sur, Sylvie Marie, Zuck, Paul D., Hartman, George D.

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Adenosine analogue inhibitors of S-adenosylhomocysteine hydrolase von Converso, Antonella, Hartingh, Timothy, Fraley, Mark E., Garbaccio, Robert M., Hartman, George D., Huang, Shaei Y., Majercak, John M., McCampbell, Alexander, Na, Sang Jin, Ray, William J., Savage, Mary J., Wolffe, Carrie, Yeh, Suzie, Yu, Yuanjiang, White, Rebecca, Zhang, Rena

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