Discovery of N‑(3-Carbamoyl-5,5,7,7-tetramethyl-5,7-dihydro‑4H‑thieno[2,3‑c]pyran-2-yl)‑lH‑pyrazole-5-carboxamide (GLPG1837), a Novel Potentiator Which Can Open Class III Mutant Cy... von Van der Plas, Steven E, Kelgtermans, Hans, De Munck, Tom, Martina, Sébastien L. X, Dropsit, Sébastien, Quinton, Evelyne, De Blieck, Ann, Joannesse, Caroline, Tomaskovic, Linda, Jans, Mia, Christophe, Thierry, van der Aar, Ellen, Borgonovi, Monica, Nelles, Luc, Gees, Maarten, Stouten, Pieter, Van Der Schueren, Jan, Mammoliti, Oscar, Conrath, Katja, Andrews, Martin

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One-pot tandem 1,4–1,2-addition of phosphites to quinolines von De Blieck, Ann, Masschelein, Kurt G. R., Dhaene, Fréderic, Rozycka-Sokolowska, Ewa, Marciniak, Bernard, Drabowicz, Jozef, Stevens, Christian V.

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Accelerating GPCR Drug Discovery With Conformation-Stabilizing VHHs von Laeremans, Toon, Sands, Zara A, Claes, Pieter, De Blieck, Ann, De Cesco, Stephane, Triest, Sarah, Busch, Andreas, Felix, David, Kumar, Abhinav, Jaakola, Veli-Pekka, Menet, Christel

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Diphosphonylation of Aromatic Diazaheterocycles and Theoretical Rationalization of Product Yields von De Blieck, Ann, Catak, Saron, Debrouwer, Wouter, Drabowicz, Józef, Hemelsoet, Karen, Verstraelen, Toon, Waroquier, Michel, Van Speybroeck, Veronique, Stevens, Christian V.

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Design of a potent and selective dual JAK1/TYK2 inhibitor von Mammoliti, Oscar, Menet, Christel, Cottereaux, Céline, Blanc, Javier, De Blieck, Ann, Coti, Ghjuvanni, Geney, Raphaël, Oste, Line, Ostyn, Koen, Palisse, Adeline, Quinton, Evelyne, Schmitt, Benoit, Borgonovi, Monica, Parent, Isabelle, Jagerschmidt, Catherine, De Vos, Steve, Vayssiere, Béatrice, López-Ramos, Miriam, Shoji, Kenji, Brys, Reginald, Amantini, David, Galien, René, Joannesse, Caroline

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Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis von Van der Plas, Steven E, Kelgtermans, Hans, Mammoliti, Oscar, Menet, Christel, Tricarico, Giovanni, De Blieck, Ann, Joannesse, Caroline, De Munck, Tom, Lambin, Dominique, Cowart, Marlon, Dropsit, Sebastien, Martina, Sebastien L X, Gees, Maarten, Wesse, Anne-Sophie, Conrath, Katja, Andrews, Martin

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Regio‐ and Diastereoselective Functionalization of 3‐Amino‐hexahydrooxazoninones von Schurgers, Ben, Wouters, Johan, De Blieck, Ann, Van Lommen, Guy, Menet, Christel, Verniest, Guido

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Correction to “Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis” von Van der Plas, Steven E, Kelgtermans, Hans, Mammoliti, Oscar, Menet, Christel, Tricarico, Giovanni, De Blieck, Ann, Joannesse, Caroline, De Munck, Tom, Lambin, Dominique, Cowart, Marlon, Dropsit, Sebastien, Martina, Sebastien L. X, Gees, Maarten, Wesse, Anne-Sophie, Conrath, Katja, Andrews, Martin

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A safe production method for acetone cyanohydrin von Heugebaert, Thomas S.A., Roman, Bart I., De Blieck, Ann, Stevens, Christian V.

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Discovery of N -(3-Carbamoyl-5,5,7,7-tetramethyl-5,7-dihydro-4 H -thieno[2,3- c ]pyran-2-yl)-l H -pyrazole-5-carboxamide (GLPG1837), a Novel Potentiator Which Can Open Class III Mu... von Van der Plas, Steven E., Kelgtermans, Hans, De Munck, Tom, Martina, Sébastien L. X., Dropsit, Sébastien, Quinton, Evelyne, De Blieck, Ann, Joannesse, Caroline, Tomaskovic, Linda, Jans, Mia, Christophe, Thierry, van der Aar, Ellen, Borgonovi, Monica, Nelles, Luc, Gees, Maarten, Stouten, Pieter, Van Der Schueren, Jan, Mammoliti, Oscar, Conrath, Katja, Andrews, Martin

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Synthesis of Epibatidine Analogues Having a 2-Substituted 2-Azabicyclo[2.2.2]octane Skeleton von Wauters, Iris, De Blieck, Ann, Muylaert, Koen, Heugebaert, Thomas S. A., Stevens, Christian V.

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One-pot tandem 1,4-1,2-addition of phosphites to quinolines von De Blieck, Ann, Masschelein, Kurt G R, Dhaene, Fréderic, Rozycka-Sokolowska, Ewa, Marciniak, Bernard, Drabowicz, Jozef, Stevens, Christian V

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Diphosphonylation of Aromatic Diazaheterocycles and Theoretical Rationalization of Product Yields von De Blieck, Ann, Catak, Saron, Debrouwer, Wouter, Drabowicz, Józef, Hemelsoet, Karen, Verstraelen, Toon, Waroquier, Michel, Van Speybroeck, Veronique, Stevens, Christian V.

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Synthesis of 1-substituted epibatidine analogues and their in vitro and in vivo evaluation as alfa-4-beta-2 nicotinic acetylcholine receptor ligands von Heugebaert, Thomas, Van Overtveldt, Melissa, De Blieck, Ann, Wuyts, Benjamin, Augustijns, Patrick, Ponce-Gamez, Eugenia, Rivera, Alicia, De Groote, Dominic, Lefebvre, Romain, Wouters, Patrick, Meert, Theo, Devulder, Jacques, Stevens, Christian

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Synthesis of 1-substituted epibatidine analogues and their in vitro and in vivo evaluation as α 4 β 2 nicotinic acetylcholine receptor ligands von Heugebaert, Thomas S. A., Van Overtveldt, Melissa, De Blieck, Ann, Wuyts, Benjamin, Augustijns, Patrick, Ponce-Gámez, Eugenia, Rivera, Alicia, De Groote, Dominic, Lefebvre, Romain A., Wouters, Patrick, Meert, Theo, Devulder, Jacques, Stevens, Christian V.

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One-Pot Tandem 1,4- and 1,2-Addition of Phosphites to α,β-Unsaturated Hydrazones von Stevens, Christian V., Van Meenen, Ellen, Masschelein, Kurt G., Moonen, Kristof, De Blieck, Ann, Drabowicz, Jozef

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Synthesis of 1-substituted epibatidine analogues and their and evaluation as αβ nicotinic acetylcholine receptor ligands von Heugebaert, Thomas S. A, Van Overtveldt, Melissa, De Blieck, Ann, Wuyts, Benjamin, Augustijns, Patrick, Ponce-Gámez, Eugenia, Rivera, Alicia, De Groote, Dominic, Lefebvre, Romain A, Wouters, Patrick, Meert, Theo, Devulder, Jacques, Stevens, Christian V

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Synthesis of 1-substituted epibatidine analogues and their in vitroand in vivoevaluation as alpha sub(4) beta sub(2) nicotinic acetylcholine receptor ligands von Heugebaert, Thomas SA, Van Overtveldt, Melissa, De Blieck, Ann, Wuyts, Benjamin, Augustijns, Patrick, Ponce-Gamez, Eugenia, Rivera, Alicia, De Groote, Dominic, Lefebvre, Romain A, Wouters, Patrick, Meert, Theo, Devulder, Jacques, Stevens, Christian V

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Compuestos para el tratamiento del dolor, en particular el dolor neuropático, y/u otras enfermedades o trastornos que se asocian con at2r y/o señalización mediada por at2r von Christel Jeanne Marie MENET, Ann DE BLIECK

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COMPOUNDS FOR THE TREATMENT OF PAIN, IN PARTICULAR NEUROPATHIC PAIN, AND/OR OTHER DISEASES OR DISORDERS THAT ARE ASSOCIATED WITH AT2R AND/OR AT2R MEDIATED SIGNALING von MENET Christel Jeanne Marie, DE BLIECK Ann

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