Halogen–Aromatic π Interactions Modulate Inhibitor Residence Times von Heroven, Christina, Georgi, Victoria, Ganotra, Gaurav K., Brennan, Paul, Wolfreys, Finn, Wade, Rebecca C., Fernández‐Montalván, Amaury E., Chaikuad, Apirat, Knapp, Stefan

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Considerations for improved performance of competition association assays analysed with the Motulsky–Mahan's “kinetics of competitive binding” model von Georgi, Victoria, Dubrovskiy, Alexey, Steigele, Stephan, Fernández‐Montalván, Amaury E.

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Inhibition of BUB1 Kinase by BAY 1816032 Sensitizes Tumor Cells toward Taxanes, ATR, and PARP Inhibitors In Vitro and In Vivo von Siemeister, Gerhard, Mengel, Anne, Fernández-Montalván, Amaury E, Bone, Wilhelm, Schröder, Jens, Zitzmann-Kolbe, Sabine, Briem, Hans, Prechtl, Stefan, Holton, Simon J, Mönning, Ursula, von Ahsen, Oliver, Johanssen, Sandra, Cleve, Arwed, Pütter, Vera, Hitchcock, Marion, von Nussbaum, Franz, Brands, Michael, Ziegelbauer, Karl, Mumberg, Dominik

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Treating Cancer by Spindle Assembly Checkpoint Abrogation: Discovery of Two Clinical Candidates, BAY 1161909 and BAY 1217389, Targeting MPS1 Kinase von Schulze, Volker K, Klar, Ulrich, Kosemund, Dirk, Wengner, Antje M, Siemeister, Gerhard, Stöckigt, Detlef, Neuhaus, Roland, Lienau, Philip, Bader, Benjamin, Prechtl, Stefan, Holton, Simon J, Briem, Hans, Marquardt, Tobias, Schirok, Hartmut, Jautelat, Rolf, Bohlmann, Rolf, Nguyen, Duy, Fernández-Montalván, Amaury E, Bömer, Ulf, Eberspaecher, Uwe, Brüning, Michael, Döhr, Olaf, Raschke, Marian, Kreft, Bertolt, Mumberg, Dominik, Ziegelbauer, Karl, Brands, Michael, von Nussbaum, Franz, Koppitz, Marcus

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Characterization of 12 GnRH peptide agonists – a kinetic perspective von Nederpelt, Indira, Georgi, Victoria, Schiele, Felix, Nowak‐Reppel, Katrin, Fernández‐Montalván, Amaury E., IJzerman, Adriaan P., Heitman, Laura H.

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Discovery and Characterization of BAY 1214784, an Orally Available Spiroindoline Derivative Acting as a Potent and Selective Antagonist of the Human Gonadotropin-Releasing Hormone... von Panknin, Olaf, Wagenfeld, Andrea, Bone, Wilhelm, Bender, Eckhard, Nowak-Reppel, Katrin, Fernández-Montalván, Amaury E, Nubbemeyer, Reinhard, Bäurle, Stefan, Ring, Sven, Schmees, Norbert, Prien, Olaf, Schäfer, Martina, Friedrich, Christian, Zollner, Thomas M, Steinmeyer, Andreas, Mueller, Thomas, Langer, Gernot

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Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains von Bouché, Léa, Christ, Clara D, Siegel, Stephan, Fernández-Montalván, Amaury E, Holton, Simon J, Fedorov, Oleg, ter Laak, Antonius, Sugawara, Tatsuo, Stöckigt, Detlef, Tallant, Cynthia, Bennett, James, Monteiro, Octovia, Díaz-Sáez, Laura, Siejka, Paulina, Meier, Julia, Pütter, Vera, Weiske, Jörg, Müller, Susanne, Huber, Kilian V. M, Hartung, Ingo V, Haendler, Bernard

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Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action von Fernández-Montalván, Amaury E, Berger, Markus, Kuropka, Benno, Koo, Seong Joo, Badock, Volker, Weiske, Joerg, Puetter, Vera, Holton, Simon J, Stöckigt, Detlef, ter Laak, Antonius, Centrella, Paolo A, Clark, Matthew A, Dumelin, Christoph E, Sigel, Eric A, Soutter, Holly H, Troast, Dawn M, Zhang, Ying, Cuozzo, John W, Keefe, Anthony D, Roche, Didier, Rodeschini, Vincent, Chaikuad, Apirat, Díaz-Sáez, Laura, Bennett, James M, Fedorov, Oleg, Huber, Kilian V. M, Hübner, Jan, Weinmann, Hilmar, Hartung, Ingo V, Gorjánácz, Mátyás

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ATAD2 is an epigenetic reader of newly synthesized histone marks during DNA replication von Koo, Seong Joo, Fernández-Montalván, Amaury E, Badock, Volker, Ott, Christopher J, Holton, Simon J, von Ahsen, Oliver, Toedling, Joern, Vittori, Sarah, Bradner, James E, Gorjánácz, Mátyás

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Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2 von Eggert, Erik, Hillig, Roman C, Koehr, Silke, Stöckigt, Detlef, Weiske, Jörg, Barak, Naomi, Mowat, Jeffrey, Brumby, Thomas, Christ, Clara D, ter Laak, Antonius, Lang, Tina, Fernandez-Montalvan, Amaury E, Badock, Volker, Weinmann, Hilmar, Hartung, Ingo V, Barsyte-Lovejoy, Dalia, Szewczyk, Magdalena, Kennedy, Steven, Li, Fengling, Vedadi, Masoud, Brown, Peter J, Santhakumar, Vijayaratnam, Arrowsmith, Cheryl H, Stellfeld, Timo, Stresemann, Carlo

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Characterization of the Menin-MLL Interaction as Therapeutic Cancer Target von Brzezinka, Krzysztof, Nevedomskaya, Ekaterina, Lesche, Ralf, Haegebarth, Andrea, Ter Laak, Antonius, Fernández-Montalván, Amaury E, Eberspaecher, Uwe, Werbeck, Nicolas D, Moenning, Ursula, Siegel, Stephan, Haendler, Bernard, Eheim, Ashley L, Stresemann, Carlo

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Binding kinetics in drug discovery - A current perspective von Georgi, Victoria, Andres, Dorothee, Fernandez-Montalvan, Amaury E, Stegmann, Christian M, Becker, Andreas, Mueller-Fahrnow, Anke

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Buriti oil as an alternative to the use of antimicrobials in broiler diets von Carvalho, Francisca Luana A, Lopes, Patrícia M, Moura, Francinete A S, Dourado, Leilane B R, Souza, Reneton G DE, Feitoza, Alison C, Oliveira, Amaury N DE, Biagiotti, Daniel

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Acidentes de trabalho e o uso de equipamentos de proteção individuais pelos profissionais de saúde em um Hospital Terciário von Andrade, Filipe Castro de, Silva Filho, Amaury de Castro e, Castro, Maria Euridéa de, Costa, Pedro Henrique Sá, Silva, Dilson Feitoza da

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5.2 Cuff and Tonometer Based Device for Assessment of Carotid to Femoral Pulse Wave Velocity: Validation According to Artery Society Guidelines von Butlin, M., Bozec, E., Millet-Amaury, E., Pucci, G., Battista, F., Qasem, A., Schillaci, G., Boutouyrie, P., Avolio, A.

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Cuff and tonometer based device for assessment of carotid to femoral pulse wave velocity: Validation according to Artery Society Guidelines von Butlin, M, Bozec, E, Millet-Amaury, E, Pucci, G, Battista, F, Qasem, A, Schillaci, G, Boutouyrie, P, Avolio, A

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INFECÇÃO POR COVID-19 EM PACIENTES TRANSPLANTADOS DE FÍGADO von Hyppolito, Elodie Bomfim, Justa, Beatriz Hyppolito da, Mendes, Karen Soares, Fontenele, Thaís Azevedo Souza, Barroso, Júlia do Carmo, Studart, Isabela Carvalho, Caronne, Lívia, Araújo Filho, Antônio Haroldo, Pereira, Karla Brandão, Rocha, Tarciso Daniel dos Santos da, Gomes, Cynthia Viana Ferreira, Azevedo, Clébia, Pereira, Heloisa Vidal Alves, Feitosa Neto, Bartolomeu Alves, Miranda, Leda Fátima Rocha, Coelho, Gustavo Rêgo, Mesquita, Denissa Ferreira Gomes de, Garcia, Paulo Ewerton, Silva Filho, Amaury de Castro e, Pires Neto, Roberto da Justa, Girão, Evelyne Santana, Garcia, José Huygens Parente

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Halogenaromatische π‐Wechselwirkungen modulieren die Verweilzeit von Inhibitoren von Heroven, Christina, Georgi, Victoria, Ganotra, Gaurav K., Brennan, Paul, Wolfreys, Finn, Wade, Rebecca C., Fernández‐Montalván, Amaury E., Chaikuad, Apirat, Knapp, Stefan

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Abstract 4691: Identification and characterization of BRPF1 bromodomain inhibitors von Haendler, Bernard, Bouché, Léa, Siegel, Stephan, Fernandez-Montalvan, Amaury E., Sugawara, Tatsuo, Meier, Julia, Knapp, Stefan, Gamble, Vicki

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Abstract 160: High target binding affinity with long lasting cellular target engagement and high dose intermittent schedule of PI3K inhibitor copanlisib contribute to the potent an... von Fernández-Montalván, Amaury E., Georgi, Victoria, Vasta, James, Glaeske, Sarah, Puetter, Vera, Robers, Matthew B., Moenning, Ursula, Sturz, Andrea, Lefranc, Julien, Ziegelbauer, Karl, Brands, Michael, Stegmann, Christian, Scott, William J., Liu, Ningshu

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