Molecular Basis for the Inhibition of Human α-Thrombin by the Macrocyclic Peptide Cyclotheonamide A von Maryanoff, Bruce E., Qiu, Xiayang, Padmanabhan, K. P., Tulinsky, Alexander, Almond, Harold R., Andrade-Gordon, Patricia, Greco, Michael N., Kauffman, Jack A., Nicolaou, K. C., Liu, Aijn, Brungs, Peter H., Fusetani, Nobuhiro

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Aroyl(aminoacyl)pyrroles, a New Class of Anticonvulsant Agents von Carson, John R, Carmosin, Richard J, Pitis, Philip M, Vaught, Jeffry L, Almond, Harold R, Stables, James P, Wolf, Harold H, Swinyard, Ewart A, White, H. Steve

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Alpha(2) adrenoceptor agonists as potential analgesic agents. 3. Imidazolylmethylthiophenes von Boyd, R E, Press, J B, Rasmussen, C R, Raffa, R B, Codd, E E, Connelly, C D, Li, Q S, Martinez, R P, Lewis, M A, Almond, H R, Reitz, A B

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Gaussian docking functions von McGann, Mark R., Almond, Harold R., Nicholls, Anthony, Grant, J. Andrew, Brown, Frank K.

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2-Substituted 1-azabicycloalkanes, a new class of non-opiate antinociceptive agents von Carson, John R, Carmosin, Richard J, Vaught, Jeffry L, Gardocki, Joseph F, Costanzo, Michael J, Raffa, Robert B, Almond, Harold R

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2-Ethynylbenzenealkanamines. A new class of calcium entry blockers von Carson, J. R, Almond, H. R, Brannan, M. D, Carmosin, R. J, Flaim, S. F, Gill, A, Gleason, M. M, Keely, S. L, Ludovici, D. W

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Stereochemistry and mechanism of the Wittig reaction: diastereomeric reaction intermediates and analysis of the reaction course von MARYANOFF, B. E, REITZ, A. B, MUTTER, M. S, INNERS, R. R, ALMOND, H. R. JR, WHITTLE, R. R, OLOFSON, R. A

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Structure-Function Analysis of Urotensin II and Its Use in the Construction of a Ligand-Receptor Working Model von Kinney, William A., Almond, Jr, Harold R., Qi, Jenson, Smith, Charles E., Santulli, Rosemary J., de Garavilla, Lawrence, Andrade-Gordon, Patricia, Cho, Daniel S., Everson, Anita M., Feinstein, Mark A., Leung, Perry A., Maryanoff, Bruce E.

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Potent, Small-Molecule Inhibitors of Human Mast Cell Tryptase. Antiasthmatic Action of a Dipeptide-Based Transition-State Analogue Containing a Benzothiazole Ketone von Costanzo, Michael J, Yabut, Stephen C, Almond, Harold R, Andrade-Gordon, Patricia, Corcoran, Thomas W, de Garavilla, Lawrence, Kauffman, Jack A, Abraham, William M, Recacha, Rosario, Chattopadhyay, Debashish, Maryanoff, Bruce E

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Pharmaceuticals and related drugs von Janicki, Casimir A, Gilpin, Roger K, Moyer, Ernest, Almond, Harold R, Erlich, Ronald H

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α2 Adrenoceptor Agonists as Potential Analgesic Agents. 3. Imidazolylmethylthiophenes von Boyd, Robert E, Rasmussen, C. Royce, Press, Jeffery B, Raffa, Robert B, Codd, Ellen E, Connelly, Charlene D, Li, Quan S, Martinez, Rebecca P, Lewis, Martin A, Almond, Harold R, Reitz, Allen B

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In-Depth Study of Tripeptide-Based α-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S 1 ‘ Subsite and Its Implications to Structure-Based Drug Design von Costanzo, Michael J., Almond, Harold R., Hecker, Leonard R., Schott, Mary R., Yabut, Stephen C., Zhang, Han-Cheng, Andrade-Gordon, Patricia, Corcoran, Thomas W., Giardino, Edward C., Kauffman, Jack A., Lewis, Joan M., de Garavilla, Lawrence, Haertlein, Barbara J., Maryanoff, Bruce E.

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Reaction of Haloperidol with 5-(Hydroxymethyl)-2-furfuraldehyde, an Impurity in Anhydrous Lactose von Janicki, Casimir A., Almond, Harold R.

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Nonpeptide Inhibitors of Cathepsin G:  Optimization of a Novel β-Ketophosphonic Acid Lead by Structure-Based Drug Design von Greco, Michael N, Hawkins, Michael J, Powell, Eugene T, Almond, Harold R, Corcoran, Thomas W, de Garavilla, Lawrence, Kauffman, Jack A, Recacha, Rosario, Chattopadhyay, Debashish, Andrade-Gordon, Patricia, Maryanoff, Bruce E

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Stereospecific enammonium-iminium rearrangements in a benzo[a]quinolizidine system von Maryanoff, Bruce E, McComsey, David F, Leo, Gregory C, Almond, Harold R

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Dramatic reversal of diastereoselectivity in an N-acyliminium ion cyclization leading to hexahydropyrrolo[2,1-a]isoquinolines. A case of competing steric interactions von Maryanoff, Bruce E, McComsey, David F, Almond, Harold R, Mutter, Martin S, Bemis, Guy W, Whittle, Robert R, Olofson, R. A

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Stereochemistry and conformation of a nitrogen-containing, medium-sized ring: hexahydro-1-phenyl-3-benzazonine derivatives. High 1,4-diastereoselectivity in hydrogenation of an exo... von Maryanoff, Bruce E, Almond, Harold R

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Pharmaceuticals and related drugs von Huettemann, Richard E, Cotter, Mary L, Shaw, Charles J, Janicki, Casimir A, Almond, Harold R, Moyer, Ernest S, Shroff, Arvin P, Vestano, Frank

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NMR rate study on the Wittig reaction of 2,2-dimethylpropanal and tributylbutylidenephosphorane von Maryanoff, Bruce E., Reitz, Allen B., Graden, David W., Almond, Harold R.

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Stereoselective synthesis of β-aryl-β-amino esters von Cohen, Judith H, Abdel-Magid, Ahmed F, Almond, Harold R, Maryanoff, Cynthia A

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