SATURATED NITROGEN AND N-ACYLATED HETEROCYCLES POTENTIATING THE ACTIVITY OF AN ACTIVE ANTIBIOTIC AGAINST MYCOBACTERIA N von Nicolas WILLAND N, Benoit DEPREZ B, Lucie MAINGOT L, Priscille BRODIN P, Alain BAULARD A, Marion FLIPO M

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SPIROISOXAZOLINE COMPOUNDS HAVING AN ACTIVITY POTENTIATING THE ACTIVITY OF AN ANTIBIOTIC von Laurence AGOURIDAS-DUTOT L, Nicolas WILLAND N, Benoit DEPREZ B, Priscille BRODIN P, Alain BAULARD A, Matthieu Frederik DESROSES MF

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Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420 von Blondiaux, Nicolas, Moune, Martin, Desroses, Matthieu, Frita, Rosangela, Flipo, Marion, Mathys, Vanessa, Soetaert, Karine, Kiass, Mehdi, Delorme, Vincent, Djaout, Kamel, Trebosc, Vincent, Kemmer, Christian, Wintjens, René, Wohlkönig, Alexandre, Antoine, Rudy, Huot, Ludovic, Hot, David, Coscolla, Mireia, Feldmann, Julia, Gagneux, Sebastien, Locht, Camille, Brodin, Priscille, Gitzinger, Marc, Déprez, Benoit, Willand, Nicolas, Baulard, Alain R.

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Cyclodextrin-based nanocarriers containing a synergic drug combination: A potential formulation for pulmonary administration of antitubercular drugs von Salzano, Giuseppina, Wankar, Jitendra, Ottani, Stefano, Villemagne, Baptiste, Baulard, Alain R., Willand, Nicolas, Brodin, Priscille, Manet, Ilse, Gref, Ruxandra

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Intrinsic Antibacterial Activity of Nanoparticles Made of β‑Cyclodextrins Potentiates Their Effect as Drug Nanocarriers against Tuberculosis von Machelart, Arnaud, Salzano, Giuseppina, Li, Xue, Demars, Aurore, Debrie, Anne-Sophie, Menendez-Miranda, Mario, Pancani, Elisabetta, Jouny, Samuel, Hoffmann, Eik, Deboosere, Nathalie, Belhaouane, Imène, Rouanet, Carine, Simar, Sophie, Talahari, Smaïl, Giannini, Valerie, Villemagne, Baptiste, Flipo, Marion, Brosch, Roland, Nesslany, Fabrice, Deprez, Benoit, Muraille, Eric, Locht, Camille, Baulard, Alain R, Willand, Nicolas, Majlessi, Laleh, Gref, Ruxandra, Brodin, Priscille

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Direct Measurement of Hydrophobic Forces on Cell Surfaces Using AFM von Alsteens, David, Dague, Etienne, Rouxhet, Paul G, Baulard, Alain R, Dufrêne, Yves F

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Loss-of-function mutations in ndh do not confer delamanid, ethionamide, isoniazid, or pretomanid resistance in Mycobacterium tuberculosis von Pandey, Sushil, Vilchèze, Catherine, Werngren, Jim, Bainomugisa, Arnold, Mansjö, Mikael, Groenheit, Ramona, Miotto, Paolo, Cirillo, Daniela M, Coulter, Christopher, Baulard, Alain R, Schön, Thomas, Jacobs, Jr, William R, Djaout, Kamel, Köser, Claudio U

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A fragment merging approach towards the development of small molecule inhibitors of Mycobacterium tuberculosis EthR for use as ethionamide boosters von Nikiforov, Petar O, Surade, Sachin, Blaszczyk, Michal, Delorme, Vincent, Brodin, Priscille, Baulard, Alain R, Blundell, Tom L, Abell, Chris

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Both Nitro Groups Are Essential for High Antitubercular Activity of 3,5-Dinitrobenzylsulfanyl Tetrazoles and 1,3,4-Oxadiazoles through the Deazaflavin-Dependent Nitroreductase Acti... von Karabanovich, Galina, Fabiánová, Viktória, Vocat, Anthony, Dušek, Jan, Valášková, Lenka, Stolaříková, Jiřina, Kitson, Russell R. A., Pávek, Petr, Vávrová, Kateřina, Djaout, Kamel, Mikušová, Katarína, Baulard, Alain R., Cole, Stewart T., Korduláková, Jana, Roh, Jaroslav

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Crystal structure of the Mycobacterium tuberculosis VirS regulator reveals its interaction with the lead compound SMARt751 von Grosse, Camille, Sigoillot, Maud, Megalizzi, Véronique, Tanina, Abdalkarim, Willand, Nicolas, Baulard, Alain R., Wintjens, René

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EthR, a repressor of the TetR/CamR family implicated in ethionamide resistance in mycobacteria, octamerizes cooperatively on its operator von Engohang‐Ndong, Jean, Baillat, David, Aumercier, Marc, Bellefontaine, Flore, Besra, Gurdyal S., Locht, Camille, Baulard, Alain R.

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Structure of EthR in a Ligand Bound Conformation Reveals Therapeutic Perspectives against Tuberculosis von Frénois, Frédéric, Engohang-Ndong, Jean, Locht, Camille, Baulard, Alain R., Villeret, Vincent

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Tuberculosis: The drug development pipeline at a glance von Villemagne, Baptiste, Crauste, Céline, Flipo, Marion, Baulard, Alain R., Déprez, Benoit, Willand, Nicolas

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Exploring the Antitubercular Activity of Anthranilic Acid Derivatives: From MabA (FabG1) Inhibition to Intrabacterial Acidification von Faïon, Léo, Djaout, Kamel, Pintiala, Catalin, Piveteau, Catherine, Leroux, Florence, Biela, Alexandre, Slupek, Stéphanie, Antoine, Rudy, Záhorszká, Monika, Cantrelle, Francois-Xavier, Hanoulle, Xavier, Korduláková, Jana, Deprez, Benoit, Willand, Nicolas, Baulard, Alain R, Flipo, Marion

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Organization of the mycobacterial cell wall: a nanoscale view von Alsteens, David, Verbelen, Claire, Dague, Etienne, Raze, Dominique, Baulard, Alain R., Dufrêne, Yves F.

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Synthetic EthR inhibitors boost antituberculous activity of ethionamide von Baulard, Alain R, Willand, Nicolas, Dirié, Bertrand, Carette, Xavier, Bifani, Pablo, Singhal, Amit, Desroses, Matthieu, Leroux, Florence, Willery, Eve, Mathys, Vanessa, Déprez-Poulain, Rebecca, Delcroix, Guy, Frénois, Frédéric, Aumercier, Marc, Locht, Camille, Villeret, Vincent, Déprez, Benoit

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New active leads for tuberculosis booster drugs by structure-based drug discovery von Tatum, Natalie J, Liebeschuetz, John W, Cole, Jason C, Frita, Rosangela, Herledan, Adrien, Baulard, Alain R, Willand, Nicolas, Pohl, Ehmke

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Chemical Force Microscopy of Single Live Cells von Dague, Etienne, Alsteens, David, Latgé, Jean-Paul, Verbelen, Claire, Raze, Dominique, Baulard, Alain R, Dufrêne, Yves F

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Unique Mechanism of Action of the Thiourea Drug Isoxyl on Mycobacterium tuberculosis von Phetsuksiri, Benjawan, Jackson, Mary, Scherman, Hataichanok, McNeil, Michael, Besra, Gurdyal S., Baulard, Alain R., Slayden, Richard A., DeBarber, Andrea E., Barry, Clifton E., Baird, Mark S., Crick, Dean C., Brennan, Patrick J.

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Ethionamide Boosters: Synthesis, Biological Activity, and Structure−Activity Relationships of a Series of 1,2,4-Oxadiazole EthR Inhibitors von Flipo, Marion, Desroses, Matthieu, Lecat-Guillet, Nathalie, Dirié, Bertrand, Carette, Xavier, Leroux, Florence, Piveteau, Catherine, Demirkaya, Fatma, Lens, Zoé, Rucktooa, Prakash, Villeret, Vincent, Christophe, Thierry, Jeon, Hee Kyoung, Locht, Camille, Brodin, Priscille, Déprez, Benoit, Baulard, Alain R, Willand, Nicolas

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