Natural product fragment combination to performance-diverse pseudo-natural products von Grigalunas, Michael, Burhop, Annina, Zinken, Sarah, Pahl, Axel, Gally, José-Manuel, Wild, Niklas, Mantel, Yannik, Sievers, Sonja, Foley, Daniel J., Scheel, Rebecca, Strohmann, Carsten, Antonchick, Andrey P., Waldmann, Herbert

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Design, Synthesis, and Phenotypic Profiling of Pyrano‐Furo‐Pyridone Pseudo Natural Products von Christoforow, Andreas, Wilke, Julian, Binici, Aylin, Pahl, Axel, Ostermann, Claude, Sievers, Sonja, Waldmann, Herbert

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Assessing biologic/toxicologic effects of extractables from plastic contact materials for advanced therapy manufacturing using cell painting assay and cytotoxicity screening von Pahl, Ina, Pahl, Axel, Hauk, Armin, Budde, Dana, Sievers, Sonja, Fruth, Lothar, Menzel, Roberto

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Phenotyping Reveals Targets of a Pseudo‐Natural‐Product Autophagy Inhibitor von Foley, Daniel J., Zinken, Sarah, Corkery, Dale, Laraia, Luca, Pahl, Axel, Wu, Yao‐Wen, Waldmann, Herbert

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A Scaffold‐Diversity Synthesis of Biologically Intriguing Cyclic Sulfonamides von Zimmermann, Stefan, Akbarzadeh, Mohammad, Otte, Felix, Strohmann, Carsten, Sankar, Muthukumar Gomathi, Ziegler, Slava, Pahl, Axel, Sievers, Sonja, Kumar, Kamal

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Image‐Based Morphological Profiling Identifies a Lysosomotropic, Iron‐Sequestering Autophagy Inhibitor von Laraia, Luca, Garivet, Guillaume, Foley, Daniel J., Kaiser, Nadine, Müller, Sebastian, Zinken, Sarah, Pinkert, Thomas, Wilke, Julian, Corkery, Dale, Pahl, Axel, Sievers, Sonja, Janning, Petra, Arenz, Christoph, Wu, Yaowen, Rodriguez, Raphaël, Waldmann, Herbert

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Phenyl Esters Are Potent Inhibitors of Caseinolytic Protease P and Reveal a Stereogenic Switch for Deoligomerization von Hackl, Mathias W, Lakemeyer, Markus, Dahmen, Maria, Glaser, Manuel, Pahl, Axel, Lorenz-Baath, Katrin, Menzel, Thomas, Sievers, Sonja, Böttcher, Thomas, Antes, Iris, Waldmann, Herbert, Sieber, Stephan A

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Exploring Natural Product Fragments for Drug and Probe Discovery von Pahl, Axel, Waldmann, Herbert, Kumar, Kamal

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Synthesis of Indofulvin Pseudo‐Natural Products Yields a New Autophagy Inhibitor Chemotype von Burhop, Annina, Bag, Sukdev, Grigalunas, Michael, Woitalla, Sophie, Bodenbinder, Pia, Brieger, Lukas, Strohmann, Carsten, Pahl, Axel, Sievers, Sonja, Waldmann, Herbert

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A compound-target pairs dataset: differences between drugs, clinical candidates and other bioactive compounds von Heinzke, A. Lina, Zdrazil, Barbara, Leeson, Paul D., Young, Robert J., Pahl, Axel, Waldmann, Herbert, Leach, Andrew R.

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Discovery of a Novel Pseudo‐Natural Product Aurora Kinase Inhibitor Chemotype through Morphological Profiling von Wang, Lin, Yilmaz, Furkan, Yildirim, Okan, Schölermann, Beate, Bag, Sukdev, Greiner, Luca, Pahl, Axel, Sievers, Sonja, Scheel, Rebecca, Strohmann, Carsten, Squire, Christopher, Foley, Daniel J., Ziegler, Slava, Grigalunas, Michael, Waldmann, Herbert

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Spacial ScoreA Comprehensive Topological Indicator for Small-Molecule Complexity von Krzyzanowski, Adrian, Pahl, Axel, Grigalunas, Michael, Waldmann, Herbert

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The Cell Painting Assay as a Screening Tool for the Discovery of Bioactivities in New Chemical Matter von Pahl, Axel, Sievers, Sonja

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Phenotyping Reveals Targets of a Pseudo‐Natural‐Product Autophagy Inhibitor von Foley, Daniel J., Zinken, Sarah, Corkery, Dale, Laraia, Luca, Pahl, Axel, Wu, Yao‐Wen, Waldmann, Herbert

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Phenotypic profiling enables the targeted design of a novel pseudo-natural product class von Zinken, Sarah, Pahl, Axel, Grigalunas, Michael, Waldmann, Herbert

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Morphological profiling by means of the Cell Painting assay enables identification of tubulin-targeting compounds von Akbarzadeh, Mohammad, Deipenwisch, Ilka, Schoelermann, Beate, Pahl, Axel, Sievers, Sonja, Ziegler, Slava, Waldmann, Herbert

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Combination of Pseudo‐Natural Product Design and Formal Natural Product Ring Distortion Yields Stereochemically and Biologically Diverse Pseudo‐Sesquiterpenoid Alkaloids von Liu, Jie, Flegel, Jana, Otte, Felix, Pahl, Axel, Sievers, Sonja, Strohmann, Carsten, Waldmann, Herbert

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Morphological Profiling Identifies a Common Mode of Action for Small Molecules with Different Targets von Schneidewind, Tabea, Brause, Alexandra, Pahl, Axel, Burhop, Annina, Mejuch, Tom, Sievers, Sonja, Waldmann, Herbert, Ziegler, Slava

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Design, Synthesis, and Biological Evaluation of Chemically and Biologically Diverse Pyrroquinoline Pseudo Natural Products von Liu, Jie, Cremosnik, Gregor S., Otte, Felix, Pahl, Axel, Sievers, Sonja, Strohmann, Carsten, Waldmann, Herbert

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Chromopynones are pseudo natural product glucose uptake inhibitors targeting glucose transporters GLUT-1 and -3 von Karageorgis, George, Reckzeh, Elena S., Ceballos, Javier, Schwalfenberg, Melanie, Sievers, Sonja, Ostermann, Claude, Pahl, Axel, Ziegler, Slava, Waldmann, Herbert

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