Absorption and Drug Development: Solubility, Permeability, and Charge State von Avdeef, Alex

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Solubility of sparingly-soluble ionizable drugs von Avdeef, Alex

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Leakiness and Size Exclusion of Paracellular Channels in Cultured Epithelial Cell Monolayers-Interlaboratory Comparison von Avdeef, Alex

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Predicting Solubility of Newly-Approved Drugs (2016–2020) with a Simple ABSOLV and GSE(Flexible-Acceptor) Consensus Model Outperforming Random Forest Regression von Avdeef, Alex, Kansy, Manfred

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Trends in PhysChem Properties of Newly Approved Drugs over the Last Six Years; Predicting Solubility of Drugs Approved in 2021 von Avdeef, Alex, Kansy, Manfred

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Correction: Trends in PhysChem Properties of Newly Approved Drugs over the Last Six Years; Predicting Solubility of Drugs Approved in 2021 von Avdeef, Alex, Kansy, Manfred

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Coexistence of passive and carrier-mediated processes in drug transport von Sugano, Kiyohiko, Kansy, Manfred, Artursson, Per, Avdeef, Alex, Bendels, Stefanie, Di, Li, Ecker, Gerhard F, Faller, Bernard, Fischer, Holger, Gerebtzoff, Grégori, Lennernaes, Hans, Senner, Frank

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How Well Can the Caco-2/Madin−Darby Canine Kidney Models Predict Effective Human Jejunal Permeability? von Avdeef, Alex, Tam, Kin Y

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Prediction of aqueous intrinsic solubility of druglike molecules using Random Forest regression trained with Wiki-pS0 database von Avdeef, Alex

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Cocrystal Solubility Product Prediction Using an in combo Model and Simulations to Improve Design of Experiments von Avdeef, Alex

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Cocrystal solubility product analysis – Dual concentration-pH mass action model not dependent on explicit solubility equations von Avdeef, Alex

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Disproportionation of Pharmaceutical Salts: pH max and Phase-Solubility/pH Variance von Avdeef, Alex

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Disproportionation of Pharmaceutical Salts: pHmax and Phase-Solubility/pH Variance von Avdeef, Alex

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Solubility-pH profile of desipramine hydrochloride in saline phosphate buffer: Enhanced solubility due to drug-buffer aggregates von Marković, Olivera S., Pešić, Miloš P., Shah, Ankita V., Serajuddin, Abu T.M., Verbić, Tatjana Ž., Avdeef, Alex

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Solubility Challenge Revisited after Ten Years, with Multilab Shake-Flask Data, Using Tight (SD ∼ 0.17 log) and Loose (SD ∼ 0.62 log) Test Sets von Llinas, Antonio, Avdeef, Alex

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PAMPA—critical factors for better predictions of absorption von Avdeef, Alex, Bendels, Stefanie, Di, L.i., Faller, Bernard, Kansy, Manfred, Sugano, Kiyohiko, Yamauchi, Yukinori

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Evidence-based approach to assess passive diffusion and carrier-mediated drug transport von Di, Li, Artursson, Per, Avdeef, Alex, Ecker, Gerhard F., Faller, Bernard, Fischer, Holger, Houston, J. Brian, Kansy, Manfred, Kerns, Edward H., Krämer, Stefanie D., Lennernäs, Hans, Sugano, Kiyohiko

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Passive Lipoidal Diffusion and Carrier-Mediated Cell Uptake Are Both Important Mechanisms of Membrane Permeation in Drug Disposition von Smith, Dennis, Artursson, Per, Avdeef, Alex, Di, Li, Ecker, Gerhard F, Faller, Bernard, Houston, J. Brian, Kansy, Manfred, Kerns, Edward H, Krämer, Stefanie D, Lennernäs, Hans, van de Waterbeemd, Han, Sugano, Kiyohiko, Testa, Bernard

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“Flexible-Acceptor” General Solubility Equation for beyond Rule of 5 Drugs von Avdeef, Alex, Kansy, Manfred

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P-glycoprotein deficient mouse in situ blood–brain barrier permeability and its prediction using an in combo PAMPA model von Dagenais, Claude, Avdeef, Alex, Tsinman, Oksana, Dudley, Adam, Beliveau, Richard

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