Inhibitors Targeting RIPK1/RIPK3: Old and New Drugs von Martens, Sofie, Hofmans, Sam, Declercq, Wim, Augustyns, Koen, Vandenabeele, Peter

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Targeting ferroptosis protects against experimental (multi)organ dysfunction and death von Van Coillie, Samya, Van San, Emily, Goetschalckx, Ines, Wiernicki, Bartosz, Mukhopadhyay, Banibrata, Tonnus, Wulf, Choi, Sze Men, Roelandt, Ria, Dumitrascu, Catalina, Lamberts, Ludwig, Dams, Geert, Weyts, Wannes, Huysentruyt, Jelle, Hassannia, Behrouz, Ingold, Irina, Lele, Suhas, Meyer, Evelyne, Berg, Maya, Seurinck, Ruth, Saeys, Yvan, Vermeulen, An, van Nuijs, Alexander L. N., Conrad, Marcus, Linkermann, Andreas, Rajapurkar, Mohan, Vandenabeele, Peter, Hoste, Eric, Augustyns, Koen, Vanden Berghe, Tom

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ClpP Protease, a Promising Antimicrobial Target von Moreno-Cinos, Carlos, Goossens, Kenneth, Salado, Irene G, Van Der Veken, Pieter, De Winter, Hans, Augustyns, Koen

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Regulation of intestinal permeability: The role of proteases von Van Spaendonk, Hanne, Ceuleers, Hannah, Witters, Leonie, Patteet, Eveline, Joossens, Jurgen, Augustyns, Koen, Lambeir, Anne-Marie, De Meester, Ingrid, De Man, Joris G, De Winter, Benedicte Y

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Selected strategies to fight pathogenic bacteria von Plotniece, Aiva, Sobolev, Arkadij, Supuran, Claudiu T., Carta, Fabrizio, Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, Jari, Augustyns, Koen, Cos, Paul, De Vooght, Linda, Govaerts, Matthias, Aizawa, Juliana, Tammela, Päivi, Žalubovskis, Raivis

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Intrinsic temperature increase drives lipid metabolism towards ferroptosis evasion and chemotherapy resistance in pancreatic cancer von de Laat, Vincent, Topal, Halit, Spotbeen, Xander, Talebi, Ali, Dehairs, Jonas, Idkowiak, Jakub, Vanderhoydonc, Frank, Ostyn, Tessa, Zhao, Peihua, Jacquemyn, Maarten, Wölk, Michele, Sablina, Anna, Augustyns, Koen, Vanden Berghe, Tom, Roskams, Tania, Daelemans, Dirk, Fedorova, Maria, Topal, Baki, Swinnen, Johannes V.

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Visceral hypersensitivity in inflammatory bowel diseases and irritable bowel syndrome: The role of proteases von Ceuleers, Hannah, Van Spaendonk, Hanne, Hanning, Nikita, Heirbaut, Jelena, Lambeir, Anne-Marie, Joossens, Jurgen, Augustyns, Koen, De Man, Joris G, De Meester, Ingrid, De Winter, Benedicte Y

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Extended Structure–Activity Relationship and Pharmacokinetic Investigation of (4-Quinolinoyl)glycyl-2-cyanopyrrolidine Inhibitors of Fibroblast Activation Protein (FAP) von Jansen, Koen, Heirbaut, Leen, Verkerk, Robert, Cheng, Jonathan D, Joossens, Jurgen, Cos, Paul, Maes, Louis, Lambeir, Anne-Marie, De Meester, Ingrid, Augustyns, Koen, Van der Veken, Pieter

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A high-throughput target-based screening approach for the identification and assessment of Mycobacterium tuberculosis mycothione reductase inhibitors von Smiejkowska, Natalia, Oorts, Lauren, Van Calster, Kevin, De Vooght, Linda, Geens, Rob, Mattelaer, Henri-Philippe, Augustyns, Koen, Strelkov, Sergei V, Lamprecht, Dirk, Temmerman, Koen, Sterckx, Yann G-J, Cappoen, Davie, Cos, Paul

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Trans-cyclooctene—a Swiss army knife for bioorthogonal chemistry: exploring the synthesis, reactivity, and applications in biomedical breakthroughs von Adhikari, Karuna, Vanermen, Maarten, Da Silva, Gustavo, Van den Wyngaert, Tim, Augustyns, Koen, Elvas, Filipe

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Characterization of Structurally Diverse 18F‑Labeled d‑TCO Derivatives as a PET Probe for Bioorthogonal Pretargeted Imaging von Adhikari, Karuna, Dewulf, Jonatan, Vangestel, Christel, Van der Veken, Pieter, Stroobants, Sigrid, Elvas, Filipe, Augustyns, Koen

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Dipeptidyl peptidases in atherosclerosis: expression and role in macrophage differentiation, activation and apoptosis von Matheeussen, Veerle, Waumans, Yannick, Martinet, Wim, Van Goethem, Sebastiaan, Van der Veken, Pieter, Scharpé, Simon, Augustyns, Koen, De Meyer, Guido R. Y., De Meester, Ingrid

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Crystal structure of Porphyromonas gingivalis dipeptidyl peptidase 4 and structure-activity relationships based on inhibitor profiling von Rea, Dean, Van Elzen, Roos, De Winter, Hans, Van Goethem, Sebastiaan, Landuyt, Bart, Luyten, Walter, Schoofs, Liliane, Van Der Veken, Pieter, Augustyns, Koen, De Meester, Ingrid, Fülöp, Vilmos, Lambeir, Anne-Marie

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A Novel Ferroptosis Inhibitor UAMC-3203, a Potential Treatment for Corneal Epithelial Wound von Balla, Anusha, Tran, Bao, Valtari, Annika, Steven, Philipp, Scarpellini, Camilla, Augustyns, Koen, Urtti, Arto, Vellonen, Kati-Sisko, Ruponen, Marika

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An essential signal peptide peptidase identified in an RNAi screen of serine peptidases of Trypanosoma brucei von Moss, Catherine X, Brown, Elaine, Hamilton, Alana, Van der Veken, Pieter, Augustyns, Koen, Mottram, Jeremy C

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Structure–Activity Relationship Studies on Isoindoline Inhibitors of Dipeptidyl Peptidases 8 and 9 (DPP8, DPP9): Is DPP8-Selectivity an Attainable Goal? von Van Goethem, Sebastiaan, Matheeussen, Veerle, Joossens, Jurgen, Lambeir, Anne-Marie, Chen, Xin, De Meester, Ingrid, Haemers, Achiel, Augustyns, Koen, Van der Veken, Pieter

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From PERK to RIPK1: Design, synthesis and evaluation of novel potent and selective necroptosis inhibitors von Scarpellini, Camilla, Valembois, Sophie, Goossens, Kenneth, Vadi, Mike, Lanthier, Caroline, Klejborowska, Greta, Van Der Veken, Pieter, De Winter, Hans, Bertrand, Mathieu J M, Augustyns, Koen

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The Effect of a Novel Serine Protease Inhibitor on Inflammation and Intestinal Permeability in a Murine Colitis Transfer Model von Van Spaendonk, Hanne, Ceuleers, Hannah, Smet, Annemieke, Berg, Maya, Joossens, Jurgen, Van der Veken, Pieter, Francque, Sven M., Lambeir, Anne-Marie, De Man, Joris G., De Meester, Ingrid, Augustyns, Koen, De Winter, Benedicte Y.

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Spectrophores as one-dimensional descriptors calculated from three-dimensional atomic properties: applications ranging from scaffold hopping to multi-target virtual screening von Gladysz, Rafaela, Dos Santos, Fabio Mendes, Langenaeker, Wilfried, Thijs, Gert, Augustyns, Koen, De Winter, Hans

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The Effect of Serine Protease Inhibitors on Visceral Pain in Different Rodent Models With an Intestinal Insult von Ceuleers, Hannah, Hanning, Nikita, De bruyn, Michelle, De Man, Joris G, De Schepper, Heiko U, Li, Qian, Liu, Liansheng, Abrams, Steven, Smet, Annemieke, Joossens, Jurgen, Augustyns, Koen, De Meester, Ingrid, Pasricha, Pankaj J, De Winter, Benedicte Y

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