Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors von Heim-Riether, Alexander, Taylor, Steven J., Liang, Shuang, Gao, Donghong Amy, Xiong, Zhaoming, Michael August, E., Collins, Brandon K., Farmer, Bennett T., Haverty, Kathleen, Hill-Drzewi, Melissa, Junker, Hans-Dieter, Mariana Margarit, S., Moss, Neil, Neumann, Thomas, Proudfoot, John R., Keenan, Lana Smith, Sekul, Renate, Zhang, Qiang, Li, Jun, Farrow, Neil A.

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Reversal of H3K9me2 by a Small-Molecule Inhibitor for the G9a Histone Methyltransferase von Kubicek, Stefan, O'Sullivan, Roderick J., August, E. Michael, Hickey, Eugene R., Zhang, Qiang, Teodoro, Miguel L., Rea, Stephen, Mechtler, Karl, Kowalski, Jennifer A., Homon, Carol Ann, Kelly, Terence A., Jenuwein, Thomas

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Benzimidazolone as potent chymase inhibitor: Modulation of reactive metabolite formation in the hydrophobic (P 1) region von Lo, Ho Yin, Nemoto, Peter A., Kim, Jin Mi, Hao, Ming-Hong, Qian, Kevin C., Farrow, Neil A., Albaugh, Daniel R., Fowler, Danielle M., Schneiderman, Richard D., Michael August, E., Martin, Leslie, Hill-Drzewi, Melissa, Pullen, Steven S., Takahashi, Hidenori, De Lombaert, Stéphane

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SAR studies of non-zinc-chelating MMP-13 inhibitors: Improving selectivity and metabolic stability von Gao, Donghong Amy, Xiong, Zhaoming, Heim-Riether, Alexander, Amodeo, Laura, August, E. Michael, Cao, Xianhua, Ciccarelli, Leonard, Collins, Brandon K., Harrington, Kyle, Haverty, Kathleen, Hill-Drzewi, Melissa, Li, Xiang, Liang, Shuang, Margarit, Steluta Mariana, Moss, Neil, Nagaraja, Nelamangala, Proudfoot, John, Roman, Rene, Schlyer, Sabine, Keenan, Lana Smith, Taylor, Steven, Wellenzohn, Bernd, Wiedenmayer, Dieter, Li, Jun, Farrow, Neil A.

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Bioluminescent Method for Assaying Multiple Semicarbazide-Sensitive Amine Oxidase (SSAO) Family Members in Both 96- and 384-Well Formats von Peet, Gregory W., Lukas, Susan, Hill-Drzewi, Melissa, Martin, Leslie, Rybina, Irina V., Roma, Teresa, Shoultz, Alycia, Zhu, Xiang, Cazacu, Daniela, Kronkaitis, Anthony, Baptiste, Alistair, Raudenbush, Brian C., August, E. Michael, Modis, Louise Kelly

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Development of a High-Throughput Assay to Measure Histidine Decarboxylase Activity von August, E. Michael, Patnaude, Lori, Hopkins, Jerry, Studts, Joey, Gautschi, Elda, Shrutkowski, Anthony, Kronkaitis, Anthony, Brown, Martha, Kabcenell, Alisa, Rajotte, Daniel

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Abstract 5590: Screening of pediatric and adult sarcoma cell lines reveals novel patterns of sensitivity toward approved oncology drugs and investigational agents von August, E. Michael, Delosh, Rene, Laudeman, Julie, Ogle, Chad, Reinhart, Russell, Selby, Michael, Silvers, Thomas, Morris, Joel, Teicher, Beverly A.

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Abstract 4361: Target and drug discovery for recalcitrant, rare and neglected cancers von Monks, Anne, Rapisarda, Annamaria, Wrzeszczynski, Kazimierz O., August, E. Michael, Polley, Eric C., Kondapaka, Sudhir B., Kaur, Gurmeet, Newton, Dianne, Teicher, Beverley A.

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1-(2,3-Dideoxy-.beta.-D-glycero-pent-2-enofuranosyl)thymine. A highly potent and selective anti-HIV agent von Mansuri, Muzammil M, Starrett, John E, Ghazzouli, Ismail, Hitchcock, Michael J. M, Sterzycki, Roman Z, Brankovan, Vera, Lin, Tai Shun, August, E. Michael, Prusoff, William H

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Vehicle operator drowsiness alert von O 'SULLIVAN GARY R, AUGUST MICHAEL E, ROHR, JOSEPH, V

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Driver status display von DANIEL S. GLASER, GILL PATRICE, LORE JOSEPH V, SZERBA JOSEPH F, AUGUST MICHAEL E, GLASER DANIEL G

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3'-Deoxythymidin-2'-ene permeation of human lymphocyte H9 cells by nonfacilitated diffusion von August, E M, Birks, E M, Prusoff, W H

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Fluorescence polarization assay for determining histidine decarboxylase activity von August, E. Michael, Rajotte, Daniel

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Fluorescence polarization assay for determining histidine decarboxylase activity von AUGUST E. MICHAEL, RAJOTTE DANIEL

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Mechanism of Uptake of 3′‐Deoxythymidin‐2′‐ene (d4T) in Human Lymphocyte H9 Cellsa von AUGUST, E. MICHAEL, PRUSOFF, WILLIAM H.

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Cyclopentenyl uracil: An effective inhibitor of uridine salvage in vivo von Cysyk, Richard L., Malinowski, Nancy, Marquez, Victor, Zaharevitz, Daniel, August, E.Michael, Moyer, James D.

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Non-steroidal anti-inflammatory drugs and tumor progression: inhibition of fibroblast hyaluronic acid production by indomethacin and mefenamic acid von Michael August, E., Nguyen, Thuyly, Malinowski, Nancy M., Cysyk, Richard L.

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FLUORESCENCE POLARIZATION ASSAY FOR DETERMINING HISTIDINE DECARBOXYLASE ACTIVITY von AUGUST E. MICHAEL, RAJOTTE DANIEL

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FLUORESCENCE POLARIZATION ASSAY FOR DETERMINING HISTIDINE DECARBOXYLASE ACTIVITY von AUGUST, MICHAEL E, RAJOTTE, DANIEL

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Initial studies on the cellular pharmacology of 3'-deoxythymidin-2'-ene (d4t): A potent and selective inhibitor of human immunodeficiency virus von August, E.Michael, Marongiu, Maria Elena, Tai-Shun, Lin, Prusoff, William H.

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