Development of new drugs for an old target: the penicillin binding proteins von Zervosen, Astrid, Sauvage, Eric, Frère, Jean-Marie, Charlier, Paulette, Luxen, André

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Synthesis and biological evaluation of potential threonine synthase inhibitors: Rhizocticin A and Plumbemycin A von Gahungu, Mathias, Arguelles-Arias, Anthony, Fickers, Patrick, Zervosen, Astrid, Joris, Bernard, Damblon, Christian, Luxen, André

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New noncovalent inhibitors of penicillin-binding proteins from penicillin-resistant bacteria von Turk, Samo, Verlaine, Olivier, Gerards, Thomas, Zivec, Matej, Humljan, Jan, Sosič, Izidor, Amoroso, Ana, Zervosen, Astrid, Luxen, André, Joris, Bernard, Gobec, Stanislav

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Inhibition of Streptococcus pneumoniae Penicillin-Binding Protein 2x and Actinomadura R39 DD-Peptidase Activities by Ceftaroline von ZERVOSEN, Astrid, ZAPUN, Andre, FRERE, Jean-Marie

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Synthesis of an enantiopure thioester as key substrate for screening the sensitivity of penicillin binding proteins to inhibitors von Simon, Justine F., Bouillez, André, Frère, Jean-Marie, Luxen, André, Zervosen, Astrid

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Synthesis and Evaluation of 3-(Dihydroxyboryl)benzoic Acids as d,d-Carboxypeptidase R39 Inhibitors von Inglis, Steven R, Zervosen, Astrid, Woon, Esther C. Y, Gerards, Thomas, Teller, Nathalie, Fischer, Delphine S, Luxen, André, Schofield, Christopher J

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Interactions between Penicillin-Binding Proteins (PBPs) and Two Novel Classes of PBP Inhibitors, Arylalkylidene Rhodanines and Arylalkylidene Iminothiazolidin-4-ones von ZERVOSEN, Astrid, LU, Wei-Ping, ZHOULIANG CHEN, WHITE, Ronald E, DEMUTH, Thomas P, FRERE, Jean-Marie

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Fully automated radiosynthesis of N(1)-[(18)F]fluoroethyl-tryptophan and study of its biological activity as a new potential substrate for indoleamine 2,3-dioxygenase PET imaging von Henrottin, Jean, Lemaire, Christian, Egrise, Dominique, Zervosen, Astrid, Van den Eynde, Benoit, Plenevaux, Alain, Franci, Xavier, Goldman, Serge, Luxen, André

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Fully automated radiosynthesis of N 1 -[18 F]fluoroethyl-tryptophan and study of its biological activity as a new potential substrate for indoleamine 2,3-dioxygenase PET imaging von Henrottin, Jean, Lemaire, Christian, Egrise, Dominique, Zervosen, Astrid, Van den Eynde, Benoit, Plenevaux, Alain, Franci, Xavier, Goldman, Serge, Luxen, André

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Synthesis of protected α-alkyl lanthionine derivatives von Denoël, Thibaut, Zervosen, Astrid, Lemaire, Christian, Plenevaux, Alain, Luxen, André

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Stereoselective synthesis of lanthionine derivatives in aqueous solution and their incorporation into the peptidoglycan of Escherichia coli von Denoël, Thibaut, Zervosen, Astrid, Gerards, Thomas, Lemaire, Christian, Joris, Bernard, Blanot, Didier, Luxen, André

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N (1)-Fluoroalkyltryptophan Analogues: Synthesis and in vitro Study as Potential Substrates for Indoleamine 2,3-Dioxygenase von Henrottin, Jean, Zervosen, Astrid, Lemaire, Christian, Sapunaric, Frédéric, Laurent, Sophie, Van den Eynde, Benoit, Goldman, Serge, Plenevaux, Alain, Luxen, André

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Enantioselective synthesis of α-benzylated lanthionines and related tripeptides for biological incorporation into E. coli peptidoglycanElectronic supplementary information (ESI) av... von Denoël, Thibaut, Zervosen, Astrid, Lemaire, Christian, Joris, Bernard, Hervé, Mireille, Blanot, Didier, Zaragoza, Guillermo, Luxen, André

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Development of solid-supported methodology for the preparation of peptidoglycan fragments containing (2S,6R)-diaminopimelic acid von Simon, Justine F., Lamborelle, Nicolas, Zervosen, Astrid, Lemaire, Christian, Joris, Bernard, Luxen, André

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Enantioselective synthesis of α-benzylated lanthionines and related tripeptides for biological incorporation into E. coli peptidoglycan von Denoël, Thibaut, Zervosen, Astrid, Lemaire, Christian, Joris, Bernard, Hervé, Mireille, Blanot, Didier, Zaragoza, Guillermo, Luxen, André

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Fully automated radiosynthesis of N1-[18F]fluoroethyl-tryptophan and study of its biological activity as a new potential substrate for indoleamine 2,3-dioxygenase PET imaging von Henrottin, Jean, Lemaire, Christian, Egrise, Dominique, Zervosen, Astrid, Van den Eynde, Benoit, Plenevaux, Alain, Franci, Xavier, Goldman, Serge, Luxen, André

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N 1‑Fluoroalkyltryptophan Analogues: Synthesis and in vitro Study as Potential Substrates for Indoleamine 2,3-Dioxygenase von Henrottin, Jean, Zervosen, Astrid, Lemaire, Christian, Sapunaric, Frédéric, Laurent, Sophie, Van den Eynde, Benoit, Goldman, Serge, Plenevaux, Alain, Luxen, André

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Specific Structural Features of the N-Acetylmuramoyl- l-Alanine Amidase AmiD from Escherichia coli and Mechanistic Implications for Enzymes of This Family von Kerff, Frédéric, Petrella, Stéphanie, Mercier, Frédéric, Sauvage, Eric, Herman, Raphaël, Pennartz, Anne, Zervosen, Astrid, Luxen, André, Frère, Jean-Marie, Joris, Bernard, Charlier, Paulette

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Synthesis and evaluation of boronic acids as inhibitors of Penicillin Binding Proteins of classes A, B and C von Zervosen, Astrid, Bouillez, André, Herman, Alexandre, Amoroso, Ana, Joris, Bernard, Sauvage, Eric, Charlier, Paulette, Luxen, André

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Unexpected Tricovalent Binding Mode of Boronic Acids within the Active Site of a Penicillin-Binding Protein von Zervosen, Astrid, Herman, Raphael, Kerff, Frédéric, Herman, Alexandre, Bouillez, André, Prati, Fabio, Pratt, R. F, Frère, Jean-Marie, Joris, Bernard, Luxen, André, Charlier, Paulette, Sauvage, Eric

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