Synthesis of Akt Inhibitor Ipatasertib. Part 2. Total Synthesis and First Kilogram Scale-up von Remarchuk, Travis, St-Jean, Frederic, Carrera, Diane, Savage, Scott, Yajima, Herbert, Wong, Brian, Babu, Srinivasan, Deese, Alan, Stults, Jeffrey, Dong, Michael W, Askin, David, Lane, Jonathan W, Spencer, Keith L

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First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin von Hansen, Karl B, Balsells, Jaume, Dreher, Spencer, Hsiao, Yi, Kubryk, Michele, Palucki, Michael, Rivera, Nelo, Steinhuebel, Dietrich, Armstrong, Joseph D, Askin, David, Grabowski, Edward J. J

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A highly catalytic robust palladium catalyzed cyanation of aryl bromides von Maligres, Peter E., Waters, Marjorie S., Fleitz, Fred, Askin, David

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Polar Radical Pair Pathway To Assemble the Pyrimidinone Core of the HIV Integrase Inhibitor Raltegravir Potassium von Pye, Philip J, Zhong, Yong-Li, Jones, Gavin O, Reamer, Robert A, Houk, Kendall N, Askin, David

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Efficient synthesis of functionalized pyrimidones via microwave-accelerated rearrangement reaction von Zhong, Yong-Li, Zhou, Hua, Gauthier, Donald R., Askin, David

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Practical and efficient synthesis of N-halo compounds von Zhong, Yong-Li, Zhou, Hua, Gauthier, Donald R., Lee, Jaemoon, Askin, David, Dolling, Ulf H., Volante, Ralph P.

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Development of a practical synthesis to PI3K α-selective inhibitor GDC-0326 von Koenig, Stefan G., Green, Keena L., Müller, Barbara, Sowell, C. Gregory, Askin, David, Gosselin, Francis

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The transition from fellowship: finding a job von Askin, David

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152. SMOKING PREDICTS VITAMIN D DEFICIENCY IN A FRAGILITY FRACTURE POPULATION von Fitzgerald, Gillian, Askin, David, McDonald, Niamh, Mullan, Ronan

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Molecular Basis and Functional Consequences of the Dominant Effects of the Mutant Band 3 on the Structure of Normal Band 3 in Southeast Asian Ovalocytosis von Kuma, Hiroyuki, Abe, Yoshito, Askin, David, Bruce, Lesley J, Hamasaki, Tomohiro, Tanner, Michael J. A, Hamasaki, Naotaka

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289Bone Health in OrthoRehab - Room to Improve or a Bone of Contention? von Finnegan, John, Brien, Helen O, Khan, Waqar, Harkins, Patricia, Askin, David, Kennelly, Sean, Coughlan, Tara

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289; Bone Health in OrthoRehab - Room to Improve or a Bone of Contention? von Finnegan, John, Brien, Helen O, Khan, Waqar, Harkins, Patricia, Askin, David, Kennelly, Sean, Coughlan, Tara

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Mobility one week after a hip fracture – can it be predicted? von Fitzgerald, Michelle, Blake, Catherine, Askin, David, Quinlan, John, Coughlan, Tara, Cunningham, Caitriona

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Manufacture of the PI3K β‑Sparing Inhibitor Taselisib. Part 1: Early-Stage Development Routes to the Bromobenzoxazepine Core von Remarchuk, Travis, Angelaud, Rémy, Askin, David, Kumar, Archana, Thompson, Andrew S, Cheng, Hua, Reichwein, John F, Chen, Yanping, St-Jean, Frédéric

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An efficient synthesis of 4-chromanones von Zhong, Yong-Li, Boruta, David T., Gauthier, Donald R., Askin, David

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Highly Efficient Synthesis of a Staphylococcus aureus Targeting Payload to Enable the First Antibody–Antibiotic Conjugate von Linghu, Xin, Segraves, Nathaniel L., Abramovich, Ifat, Wong, Nicholas, Müller, Barbara, Neubauer, Nadja, Fantasia, Serena, Rieth, Sebastian, Bachmann, Stephan, Jansen, Michael, Sowell, C. Gregory, Askin, David, Koenig, Stefan G., Gosselin, Francis

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Cover Feature: Highly Efficient Synthesis of a Staphylococcus aureus Targeting Payload to Enable the First Antibody–Antibiotic Conjugate (Chem. Eur. J. 12/2018) von Linghu, Xin, Segraves, Nathaniel L., Abramovich, Ifat, Wong, Nicholas, Müller, Barbara, Neubauer, Nadja, Fantasia, Serena, Rieth, Sebastian, Bachmann, Stephan, Jansen, Michael, Sowell, C. Gregory, Askin, David, Koenig, Stefan G., Gosselin, Francis

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A Practical, Protecting-Group-Free Synthesis of a PI3K/mTOR Inhibitor von Tian, Qingping, Hoffmann, Ursula, Humphries, Theresa, Cheng, Zhigang, Hidber, Pirmin, Yajima, Herbert, Guillemot-Plass, Maud, Li, Jane, Bromberger, Ulrike, Babu, Srinivasan, Askin, David, Gosselin, Francis

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Synthesis of the orally active spiroindoline-based growth hormone secretagogue, MK-677 von Maligres, Peter E., Houpis, Ioannis, Rossen, Kai, Molina, Audrey, Sager, Jess, Upadhyay, Veena, Wells, Kenneth M., Reamer, Robert A., Lynch, Joseph E., Askin, David, Volante, R.P., Reider, Paul J., Houghton, Peter

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Preparation of a clinically investigated ras farnesyl transferase inhibitor von Maligres, Peter E., Waters, Marjorie S., Weissman, Steven A., McWilliams, J. Christopher, Lewis, Stephanie, Cowen, Jennifer, Reamer, Robert A., Volante, R. P., Reider, Paul J., Askin, David

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