Small molecule inhibitors reveal PTK6 kinase is not an oncogenic driver in breast cancers von Qiu, Luping, Levine, Kymberly, Gajiwala, Ketan S, Cronin, Ciarán N, Nagata, Asako, Johnson, Eric, Kraus, Michelle, Tatlock, John, Kania, Robert, Foley, Timothy, Sun, Shaoxian

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Discovery of 3-aryloxy-lactam analogs as potent androgen receptor full antagonists for treating castration resistant prostate cancer von Guo, Chuangxing, Kephart, Susan, Ornelas, Martha, Gonzalez, Javier, Linton, Angelica, Pairish, Mason, Nagata, Asako, Greasley, Samantha, Elleraas, Jeff, Hosea, Natilie, Engebretsen, Jon, Fanjul, Andrea N.

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Critical Assessment of State‐of‐the‐Art Ligand‐Based Virtual Screening Methods von Sciabola, Simone, Torella, Rubben, Nagata, Asako, Boehm, Markus

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Discovery of PF-06873600, a CDK2/4/6 Inhibitor for the Treatment of Cancer von Freeman-Cook, Kevin D, Hoffman, Robert L, Behenna, Douglas C, Boras, Britton, Carelli, Jordan, Diehl, Wade, Ferre, Rose Ann, He, You-Ai, Hui, Andrea, Huang, Buwen, Huser, Nanni, Jones, Rhys, Kephart, Susan E, Lapek, John, McTigue, Michele, Miller, Nichol, Murray, Brion W, Nagata, Asako, Nguyen, Lisa, Niessen, Sherry, Ninkovic, Sacha, O’Doherty, Inish, Ornelas, Martha A, Solowiej, James, Sutton, Scott C, Tran, Khanh, Tseng, Elaine, Visswanathan, Ravi, Xu, Meirong, Zehnder, Luke, Zhang, Qin, Zhang, Cathy, Dann, Stephen

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An allosteric cyclin E-CDK2 site mapped by paralog hopping with covalent probes von Zhang, Yuanjin, Liu, Zhonglin, Hirschi, Marscha, Brodsky, Oleg, Johnson, Eric, Won, Sang Joon, Nagata, Asako, Bezwada, Divya, Petroski, Matthew D, Majmudar, Jaimeen D, Niessen, Sherry, VanArsdale, Todd, Gilbert, Adam M, Hayward, Matthew M, Stewart, Al E, Nager, Andrew R, Melillo, Bruno, Cravatt, Benjamin F

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Protein redox chemistry: post-translational cysteine modifications that regulate signal transduction and drug pharmacology von Wani, Revati, Nagata, Asako, Murray, Brion W

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Discovery of Allosteric, Potent, Subtype Selective, and Peripherally Restricted TrkA Kinase Inhibitors von Bagal, Sharan K, Omoto, Kiyoyuki, Blakemore, David C, Bungay, Peter J, Bilsland, James G, Clarke, Philip J, Corbett, Matthew S, Cronin, Ciaran N, Cui, J. Jean, Dias, Rebecca, Flanagan, Neil J, Greasley, Samantha E, Grimley, Rachel, Johnson, Eric, Fengas, David, Kitching, Linda, Kraus, Michelle L, McAlpine, Indrawan, Nagata, Asako, Waldron, Gareth J, Warmus, Joseph S

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Discovery of N‑((3R,4R)‑4-Fluoro-1-(6-((3-methoxy-1-methyl‑1H‑pyrazol-4-yl)amino)-9-methyl‑9H‑purin-2-yl)pyrrolidine-3-yl)acrylamide (PF-06747775) through Structure-Based Drug Desi... von Planken, Simon, Behenna, Douglas C, Nair, Sajiv K, Johnson, Theodore O, Nagata, Asako, Almaden, Chau, Bailey, Simon, Ballard, T. Eric, Bernier, Louise, Cheng, Hengmiao, Cho-Schultz, Sujin, Dalvie, Deepak, Deal, Judith G, Dinh, Dac M, Edwards, Martin P, Ferre, Rose Ann, Gajiwala, Ketan S, Hemkens, Michelle, Kania, Robert S, Kath, John C, Matthews, Jean, Murray, Brion W, Niessen, Sherry, Orr, Suvi T. M, Pairish, Mason, Sach, Neal W, Shen, Hong, Shi, Manli, Solowiej, James, Tran, Khanh, Tseng, Elaine, Vicini, Paolo, Wang, Yuli, Weinrich, Scott L, Zhou, Ru, Zientek, Michael, Liu, Longqing, Luo, Yiqin, Xin, Shuibo, Zhang, Chengyi, Lafontaine, Jennifer

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Design of oxobenzimidazoles and oxindoles as novel androgen receptor antagonists von Guo, Chuangxing, Pairish, Mason, Linton, Angelica, Kephart, Susan, Ornelas, Martha, Nagata, Asako, Burke, Benjamin, Dong, Liming, Engebretsen, Jon, Fanjul, Andrea N.

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Discovery of N -((3 R ,4 R )-4-Fluoro-1-(6-((3-methoxy-1-methyl-1 H -pyrazol-4-yl)amino)-9-methyl-9 H -purin-2-yl)pyrrolidine-3-yl)acrylamide (PF-06747775) through Structure-Based... von Planken, Simon, Behenna, Douglas C., Nair, Sajiv K., Johnson, Theodore O., Nagata, Asako, Almaden, Chau, Bailey, Simon, Ballard, T. Eric, Bernier, Louise, Cheng, Hengmiao, Cho-Schultz, Sujin, Dalvie, Deepak, Deal, Judith G., Dinh, Dac M., Edwards, Martin P., Ferre, Rose Ann, Gajiwala, Ketan S., Hemkens, Michelle, Kania, Robert S., Kath, John C., Matthews, Jean, Murray, Brion W., Niessen, Sherry, Orr, Suvi T. M., Pairish, Mason, Sach, Neal W., Shen, Hong, Shi, Manli, Solowiej, James, Tran, Khanh, Tseng, Elaine, Vicini, Paolo, Wang, Yuli, Weinrich, Scott L., Zhou, Ru, Zientek, Michael, Liu, Longqing, Luo, Yiqin, Xin, Shuibo, Zhang, Chengyi, Lafontaine, Jennifer

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Second task execution assistance device and non-transitory computer readable storage medium von Yokoyama, Shizuka, Yamamoto, Takeshi, Nagata, Asako, Ota, Yuji

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Driving control device and vehicle behavior suggestion device von Yokoyama, Shizuka, Yamamoto, Takeshi, Nagata, Asako, Ota, Yuji

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Drive mode switch control device and drive mode switch control method von Mori, Takuya, Yagyu, Akihiko, Nagata, Asako, Chiba, Kunihiko

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PYRIDO[4,3-D]PYRIMIDINE COMPOUNDS von SPANGLER, Jillian Elyse, PLANKEN, Simon Paul, SUTTON, Scott Channing, NAGATA, Asako, YANG, Shouliang, DEFOREST, Jacob Cole

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DRIVE MODE SWITCH CONTROL DEVICE AND DRIVE MODE SWITCH CONTROL METHOD von MORI, Takuya, NAGATA, Asako, YAGYU, Akihiko, CHIBA, Kunihiko

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PRESENTATION CONTROL DEVICE, PRESENTATION CONTROL PROGRAM, AND DRIVING CONTROL DEVICE von KUME, Takuya, KOJIMA, Kazuki, NAGATA, Asako, YAMAMOTO, Takeshi, YOKOYAMA, Shizuka

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DRIVING CONTROL DEVICE AND VEHICLE BEHAVIOR SUGGESTION DEVICE von OTA, Yuji, NAGATA, Asako, YAMAMOTO, Takeshi, YOKOYAMA, Shizuka

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HMI control device, HMI control program product, driving control device, and driving control program product von Kume, Takuya, Yokoyama, Shizuka, Yamamoto, Takeshi, Nagata, Asako, Kojima, Kazuki, Ota, Yuji

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INFORMATION PRESENTATION CONTROL DEVICE von OTA, Yuji, NAGATA, Asako, YOKOYAMA, Shizuka, YAMAMOTO, Takeshi

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CDK2 INHIBITORS von FREEMAN-COOK, Kevin Daniel, SUTTON, Scott Channing, NAGATA, Asako, BEHENNA, Douglas Carl, NINKOVIC, Sacha, HOFFMAN, Robert Louis

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