Discovery and Pharmacokinetic and Pharmacological Properties of the Potent and Selective MET Kinase Inhibitor 1‑{6-[6-(4-Fluorophenyl)-[1,2,4]triazolo[4,3‑b]pyridazin-3-ylsulfanyl]... von Ugolini, Antonio, Kenigsberg, Mireille, Rak, Alexey, Vallée, Francois, Houtmann, Jacques, Lowinski, Maryse, Capdevila, Cécile, Khider, Jean, Albert, Eva, Martinet, Nathalie, Nemecek, Conception, Grapinet, Sandrine, Bacqué, Eric, Roesner, Manfred, Delaisi, Christine, Calvet, Loreley, Bonche, Fabrice, Semiond, Dorothée, Egile, Coumaran, Goulaouic, Hélène, Schio, Laurent

Volltext

The use of virtual screening and differential scanning fluorimetry for the rapid identification of fragments active against MEK1 von Amaning, Kwame, Lowinski, Maryse, Vallee, Francois, Steier, Valerie, Marcireau, Christophe, Ugolini, Antonio, Delorme, Cecile, Foucalt, Frédéric, McCort, Gary, Derimay, Nathalie, Andouche, Cyrielle, Vougier, Stephanie, Llopart, Sylvie, Halland, Nis, Rak, Alexey

Volltext

Abstract 2911: SAR125844: a potent and selective ATP-competitive inhibitor of MET kinase von Schio, Laurent, Nemecek, Conception, Ugolini, Antonio, Wentzler, Sylvie, Grapinet, Sandrine, Khider, Jean, Albert, Eva, Dischamps, Nathalie, Gay, Frédéric, Sonnefraud, Véronique, Bacqué, Eric, Kenigsberg, Mireille, Goulaouic, Hélène, Dagallier, Anne, Vallée, François, Bonche, Fabrice, Lengauer, Christoph

Volltext

Facile access to (S)-1,2,4-butanetriol and its derivatives von Hanessian, Stephen, Ugolini, Antonio, Dubé, Daniel, Glamyan, Ani

Volltext

Design of bivalent ligands using hydrogen bond linkers: synthesis and evaluation of inhibitors for human β-tryptase von Vaz, Roy J., Gao, Zhongli, Pribish, James, Chen, Xin, Levell, Julian, Davis, Larry, Albert, Eva, Brollo, Maurice, Ugolini, Antonio, Cramer, Dona M., Cairns, Jennifer, Sides, Keith, Liu, Feng, Kwong, Jennifer, Kang, Jiesheng, Rebello, Sam, Elliot, Michael, Lim, HengKeang, Chellaraj, Vinolia, Singleton, Robert W., Li, Yi

Volltext

derivados de 6-(6-0-ciclo alquil ou 6-nh-ciclo alquil-triazolo piridazina sulfanil) benzotiazóis e benzimadazóis: preparo, aplicação como medicamentos e utilização como inibidores... von Conception Nemecek, Eric Bacque, Baptiste Ronan, Antonio Ugolini, Sylvie Wentzler, Dominique Damour (Falecido)

Volltext bestellen

DERIVES DE 6-(6-SUBSTITUE-TRIAZOLOPYRIDAZINE-SULFANYL) 5-FLUORO-BENZOTHIAZOLES ET 5-FLUORO-BENZIMIDAZOLES : PREPARATION, APPLICATION COMME MEDICAMENTS ET UTILISATION COMME INHIBITE... von UGOLINI ANTONIO, NEMECEK CONCEPTION

Volltext bestellen

Novel Indole Derivatives, Preparation Thereof as Medicinal Products and Pharmaceutical Compositions, and Especially as KDR Inhibitors von BOUCHARD HERVE, UGOLINI ANTONIO

Volltext bestellen

6-triazolopyridazine sulfanyl benzothiazole derivatives as MET inhibitors von WENTZLER SYLVIE, UGOLINI ANTONIO, ALBERT EVA, BACQUE ERIC, NEMECEK CONCEPTION

Volltext bestellen

derivados de 6-(6-substituido-triazolo piridazina-sufanil) 5-flúor-benzo-tiazóis e 5-flúor-benzimidazóis: preparo, aplicação como medicamentos e utilização como inibidores de met... von ANTONIO UGOLINI, CONCEPTION NEMECEK, DIMINIQUE DAMOUR, SYLVIE WENTZLER, ERIC BACQUE

Volltext bestellen

NOVEL 6-TRIAZOLOPYRIDAZINE SULPHANYL BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, PROCESS FOR PREPARING SAME, USE THEREOF AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND NOVEL USE... von WENTZLٌٌٌُُُER SYLVIE, UGOLINI ANTONIO, ALBERT EVA, BACQUE ERIC, NEMECEK CONCEPTION

Volltext bestellen

"derivados de 6-(6-nh-subistituído-triazolopiridazina-sulfanil) benzotiazóis e benzimidazóis: preparo, aplicação como medicamentos e utilização como inibidores de met" von ANTONIO UGOLINI, CONCEPTION NEMECEK, SYLVIE WENTZLER, ERIC BACQUE

Volltext bestellen

NOVEL 6-TRIAZOLOPYRIDAZINESULFANYL BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, METHOD FOR PRODUCTION THEREOF AND APPLICATION AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS AND NOV... von UGOLINI, ANTONIO, NEMECEK, CONCEPTION, WENTZLER, SYLVIE, BACQUE, ERIC, ALBERT, EVA

Volltext bestellen

NOVEL 6-TRIAZOLOPYRIDAZINE SULFANYL BENZOTHIAZOLE DERIVATIVES AS MET INHIBITORS von WENTZLER SYLVIE, UGOLINI ANTONIO, ALBERT EVA, BACQUE ERIC, NEMECEK CONCEPTION

Volltext bestellen

6-triazolopyridazine sulfanyl benzothiazole derivatives as MET inhibitors von WENTZLER SYLVIE, UGOLINI ANTONIO, ALBERT EVA, BACQUE ERIC, NEMECEK CONCEPTION

Volltext bestellen

Stereocontrolled synthesis of the spiro ketal unit of avermectin B1a aglycon von Hanessian, Stephen, Ugolini, Antonio, Therien, Michel

Volltext

DERIVADOS DE 6-TRIAZOL PIRIDAZINA - SULFANIL BENZOTIAZOL E BENZIMIDAZOL, O RESPECTIVO PROCESSO DE PREPARO, A RESPECTIVA APLICAÇÃO A TÍTULO DE MEDICAMENTOS, COMPOSIÇÕES FARMACÊUTICA... von EVA ALBERT, ANTONIO UGOLINI, SYLVIE WENTZLER, ERIC BACQUE, CONCEPTIONS NEMECEK

Volltext bestellen

NOUVEAUX DERIVES DE L'INDOLE, LEUR PREPARATION A TITRE DE MEDICAMENTS, COMPOSITIONS PHARMACEUTIQUES ET NOTAMMENT COMME INHIBITEURS DE KDR von BOUCHARD HERVE, UGOLINI ANTONIO

Volltext bestellen

Synthesis of (+)-avermectin B1a von Hanessian, Stephen, Ugolini, Antonio, Dube, Daniel, Hodges, Paul J, Andre, Christiane

Volltext

NOVEL 6-TRIAZOLOPYRIDAZINESULFANYL BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, METHOD FOR PRODUCTION THEREOF AND APPLICATION AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS AND NOV... von WENTZLER SYLVIE, UGOLINI ANTONIO, ALBERT EVA, BACQUE, ERIC, NEMECEK CONCEPTION

Volltext bestellen