Discovery of Sisunatovir (RV521), an Inhibitor of Respiratory Syncytial Virus Fusion von Cockerill, G. Stuart, Angell, Richard M, Bedernjak, Alexandre, Chuckowree, Irina, Fraser, Ian, Gascon-Simorte, Jose, Gilman, Morgan S. A, Good, James A. D, Harland, Rachel, Johnson, Sara M, Ludes-Meyers, John H, Littler, Edward, Lumley, James, Lunn, Graham, Mathews, Neil, McLellan, Jason S, Paradowski, Michael, Peeples, Mark E, Scott, Claire, Tait, Dereck, Taylor, Geraldine, Thom, Michelle, Thomas, Elaine, Villalonga Barber, Carol, Ward, Simon E, Watterson, Daniel, Williams, Gareth, Young, Paul, Powell, Kenneth

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N-(3-Cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)amides as potent, selective, inhibitors of JNK2 and JNK3 von Angell, Richard M., Atkinson, Francis L., Brown, Murray J., Chuang, Tsu Tshen, Christopher, John A., Cichy-Knight, Maria, Dunn, Allison K., Hightower, Kendra E., Malkakorpi, Susanna, Musgrave, James R., Neu, Margarete, Rowland, Paul, Shea, Robyn L., Smith, Jeffery L., Somers, Donald O., Thomas, Sonia A., Thompson, Gladstone, Wang, Ruolan

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Biphenyl amide p38 kinase inhibitors 4: DFG-in and DFG-out binding modes von Angell, Richard M., Angell, Tony D., Bamborough, Paul, Bamford, Mark J., Chung, Chun-wa, Cockerill, Stuart G., Flack, Stephen S., Jones, Katherine L., Laine, Dramane I., Longstaff, Timothy, Ludbrook, Steve, Pearson, Rosannah, Smith, Kathryn J., Smee, Penny A., Somers, Don O., Walker, Ann L.

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Development of a Fluorescence Intensity Assay for the Mitotic Serine/Threonine Protein Kinase Aurora-A von Slatter, Andrew F., Campbell, Spencer, Angell, Richard M.

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Selective Plasma Hydrolysis of Glucocorticoid γ-Lactones and Cyclic Carbonates by the Enzyme Paraoxonase: An Ideal Plasma Inactivation Mechanism von Biggadike, Keith, Angell, Richard M, Burgess, Colin M, Farrell, Rosanne M, Hancock, Ashley P, Harker, Andy J, Irving, Wendy R, Ioannou, Chris, Procopiou, Panayiotis A, Shaw, Rupert E, Solanke, Yemisi E, Singh, Onkar M. P, Snowden, Michael A, Stubbs, Rob J, Walton, Sarah, Weston, Helen E

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Biphenyl amide p38 kinase inhibitors 1: Discovery and binding mode von Angell, Richard M., Bamborough, Paul, Cleasby, Anne, Cockerill, Stuart G., Jones, Katherine L., Mooney, Christopher J., Somers, Donald O., Walker, Ann L.

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Biphenyl amide p38 kinase inhibitors 2: Optimisation and SAR von Angell, Richard M., Angell, Tony D., Bamborough, Paul, Brown, David, Brown, Murray, Buckton, Jacky B., Cockerill, Stuart G., Edwards, Chris D., Jones, Katherine L., Longstaff, Tim, Smee, Penny A., Smith, Kathryn J., Somers, Don O., Walker, Ann L., Willson, Malcolm

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N-4-Pyrimidinyl-1H-indazol-4-amine inhibitors of Lck: Indazoles as phenol isosteres with improved pharmacokinetics von Bamborough, Paul, Angell, Richard M., Bhamra, Inder, Brown, David, Bull, James, Christopher, John A., Cooper, Anthony W.J., Fazal, Lynsey H., Giordano, Ilaria, Hind, Lucy, Patel, Vipulkumar K., Ranshaw, Lisa E., Sims, Martin J., Skone, Philip A., Smith, Kathryn J., Vickerstaff, Emma, Washington, Melanie

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Novel glucocorticoid antedrugs possessing a 21-(γ-lactone) ring von Angell, Richard M., Biggadike, Keith, Farrell, Rosanne M., Flack, Stephen S., Hancock, Ashley P., Irving, Wendy R., Lynn, Sean M., Procopiou, Panayiotis A.

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Enantioselective synthesis of homoallylic alcohols using (E)-but-2-enyl-trichlorosilane and chiral diamines von M. Angell, Richard, G. M. Barrett, Anthony, Christopher Braddock, D., Swallow, Steven, D. Vickery, Benjamin

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2'-Methyl-5'-(1,3,4-Oxadiazol-2-yl)-1,1'-Biphenyl-4-Carboxamide Derivatives and Their Use As P38 Kinase Inhibitors von SMITH KATHRYN J, BAMBOROUGH PAUL, COCKERILL GEORGE S, WALKER ANN L, ANGELL RICHARD M

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Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis von DEBOECK NIGEL M, LONGSTAFF TIMOTHY, BAMBOROUGH PAUL, ANGELL RICHARD M, BALDWIN IAN R, SWANSON STEPHEN

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2'-Methyl-5'-(1,3,4-oxadiazol-2-yl)-1,1'-biphenyl-4-carboxamide derivatives and their use as p38 kinase inhibitors von SMITH KATHRYN J, BAMBOROUGH PAUL, COCKERILL GEORGE S, WALKER ANN L, ANGELL RICHARD M

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HETEROARYLSUBSTITUIERTE BIPHENYLDERIVATE ALS INHIBITOREN VON P38-KINASE von WALKER, ANN LOUISE, ANGELL, RICHARD M, LI-KWAIUNG, ANNE-MARIE, SWANSON, STEPHEN, SMITH, KATHRYN JANE, BAMBOROUGH, PAUL, BALDWIN, IAN R, MERRICK, SUZANNE, JOY, LONGSTAFF, TIMOTHY

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2' -METHYL-5-(1,3,4-OXADIAZOL-2-YL)-1,1'-BIPHENYL-4-CARBOXAMIDE DERIVATIVES AND THEIR USE AS P38 KINASE INHIBITORS von ANGELL, RICHARD M, WALKER, ANN, LOUISE, BAMBOROUGH, PAUL, COCKERILL, GEORGE, STUART

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Biphenyl-Derivatives as p38 Kinase Inhibitors von ASTON NICOLA M, BAMBOROUGH PAUL, COCKERILL GEORGE S, FLACK STEPHEN S, WALKER ANN L, BAMFORD MARK J, ANGELL RICHARD M, LAINE DRAMANE I

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Biphenylcarboxylic Amide Derivatives as p38 Kinase Inhibitors von ASTON NICOLA M, BAMBOROUGH PAUL, COCKERILL GEORGE S, FLACK STEPHEN S, WALKER ANN L, BAMFORD MARK J, ANGELL RICHARD M, LAINE DRAMANE I

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HETEROARYLSUBSTITUIERTE BIPHENYLDERIVATE ALS INHIBITOREN VON P38-KINASE von WALKER, ANN LOUISE, ANGELL, RICHARD M, LI-KWAIUNG, ANNE-MARIE, SWANSON, STEPHEN, MERRICK, SUZANNE JOY, SMITH, KATHRYN JANE, BAMBOROUGH, PAUL, BALDWIN, IAN R, LONGSTAFF, TIMOTHY

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HETEROARYL SUBSTITUTED BIPHENYL DERIVATIVES AS P38 KINASE INHIBITORS von WALKER, ANN LOUISE, ANGELL, RICHARD M, LI-KWAIUNG, ANNE-MARIE, SWANSON, STEPHEN, MERRICK, SUZANNE JOY, SMITH, KATHRYN JANE, BAMBOROUGH, PAUL, BALDWIN, IAN R, LONGSTAFF, TIMOTHY

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ChemInform Abstract: Novel Glucocorticoid Antedrugs Possessing a 21-(γ-Lactone) Ring von Angell, Richard M., Biggadike, Keith, Farrell, Rosanne M., Flack, Stephen S., Hancock, Ashley P., Irving, Wendy R., Lynn, Sean M., Procopiou, Panayiotis A.

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