Synthesis of Nucleoside Phosphate and Phosphonate Prodrugs von Pradere, Ugo, Garnier-Amblard, Ethel C, Coats, Steven J, Amblard, Franck, Schinazi, Raymond F

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Metabolism, Biochemical Actions, and Chemical Synthesis of Anticancer Nucleosides, Nucleotides, and Base Analogs von Shelton, Jadd, Lu, Xiao, Hollenbaugh, Joseph A, Cho, Jong Hyun, Amblard, Franck, Schinazi, Raymond F

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Agonist of RORA Attenuates Nonalcoholic Fatty Liver Progression in Mice via Up-regulation of MicroRNA 122 von Chai, Chofit, Cox, Bryan, Yaish, Dayana, Gross, Devora, Rosenberg, Nofar, Amblard, Franck, Shemuelian, Zohar, Gefen, Maytal, Korach, Amit, Tirosh, Oren, Lanton, Tali, Link, Henrike, Tam, Joseph, Permyakova, Anna, Ozhan, Gunes, Citrin, Jonathan, Liao, Haixing, Tannous, Mirna, Hahn, Michal, Axelrod, Jonathan, Arretxe, Enara, Alonso, Cristina, Martinez-Arranz, Ibon, Betés, Pablo Ortiz, Safadi, Rifaat, Salhab, Ahmad, Amer, Johnny, Tber, Zahira, Mengshetti, Seema, Giladi, Hilla, Schinazi, Raymond F., Galun, Eithan

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Assessment of a Computational Approach to Predict Drug Resistance Mutations for HIV, HBV and SARS-CoV-2 von Patel, Dharmeshkumar, Ono, Suzane K, Bassit, Leda, Verma, Kiran, Amblard, Franck, Schinazi, Raymond F

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Baicalein and Baicalin Inhibit SARS-CoV-2 RNA-Dependent-RNA Polymerase von Zandi, Keivan, Musall, Katie, Oo, Adrian, Cao, Dongdong, Liang, Bo, Hassandarvish, Pouya, Lan, Shuiyun, Slack, Ryan L, Kirby, Karen A, Bassit, Leda, Amblard, Franck, Kim, Baek, AbuBakar, Sazaly, Sarafianos, Stefan G, Schinazi, Raymond F

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Synthesis of 4'-Substituted Carbocyclic Uracil Derivatives and Their Monophosphate Prodrugs as Potential Antiviral Agents von Biteau, Nicolas G, Amichai, Sarah A, Azadi, Niloufar, De, Ramyani, Downs-Bowen, Jessica, Lecher, Julia C, MacBrayer, Tamara, Schinazi, Raymond F, Amblard, Franck

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The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir von Dinh, Tung, Tber, Zahira, Rey, Juan S, Mengshetti, Seema, Annamalai, Arun S, Haney, Reed, Briganti, Lorenzo, Amblard, Franck, Fuchs, James R, Cherepanov, Peter, Kim, Kyungjin, Schinazi, Raymond F, Perilla, Juan R, Kim, Baek, Kvaratskhelia, Mamuka

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Studies on the Efficacy, Potential Cardiotoxicity and Monkey Pharmacokinetics of GLP-26 as a Potent Hepatitis B Virus Capsid Assembly Modulator von Hurwitz, Selwyn J, McBrearty, Noreen, Arzumanyan, Alla, Bichenkov, Eugene, Tao, Sijia, Bassit, Leda, Chen, Zhe, Kohler, James J, Amblard, Franck, Feitelson, Mark A, Schinazi, Raymond F

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Structural and Antiviral Studies of the Human Norovirus GII.4 Protease von Muzzarelli, Kendall M, Kuiper, Benjamin, Spellmon, Nicholas, Brunzelle, Joseph, Hackett, Justin, Amblard, Franck, Zhou, Shaoman, Liu, Peng, Kovari, Iulia A, Yang, Zhe, Schinazi, Raymond F, Kovari, Ladislau C

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Synthesis of 4'-Substituted-2'-Deoxy-2'-α-Fluoro Nucleoside Analogs as Potential Antiviral Agents von Kasthuri, Mahesh, Li, Chengwei, Verma, Kiran, Russell, Olivia Ollinger, Dickson, Lyndsey, McCormick, Louise, Bassit, Leda, Amblard, Franck, Schinazi, Raymond F

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Why Certain Repurposed Drugs Are Unlikely to Be Effective Antivirals to Treat SARS-CoV-2 Infections von Hurwitz, Selwyn J, De, Ramyani, LeCher, Julia C, Downs-Bowen, Jessica A, Goh, Shu Ling, Zandi, Keivan, McBrayer, Tamara, Amblard, Franck, Patel, Dharmeshkumar, Kohler, James J, Bhasin, Manoj, Dobosh, Brian S, Sukhatme, Vikas, Tirouvanziam, Rabindra M, Schinazi, Raymond F

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Synthesis of Novel N4-Hydrocytidine Analogs as Potential Anti-SARS-CoV-2 Agents von Amblard, Franck, LeCher, Julia C., De, Ramyani, Goh, Shu Ling, Li, Chengwei, Kasthuri, Mahesh, Biteau, Nicolas, Zhou, Longhu, Tber, Zahira, Downs-Bowen, Jessica, Zandi, Keivan, Schinazi, Raymond F.

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Cu(I)-catalyzed Huisgen azide-alkyne 1,3-dipolar cycloaddition reaction in nucleoside, nucleotide, and oligonucleotide chemistry von Amblard, Franck, Cho, Jong Hyun, Schinazi, Raymond F

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Synthesis and antiviral evaluation of 2′,2′,3′,3′-tetrafluoro nucleoside analogs von Sari, Ozkan, Bassit, Leda, Gavegnano, Christina, McBrayer, Tamara R., McCormick, Louise, Cox, Bryan, Coats, Steven J., Amblard, Franck, Schinazi, Raymond F.

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Ordered stacking of F-actin layers and mixed lipid bilayers: a columnar liquid crystal von Caillé, A, Artzner, F, Amblard, F

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Abstract 1458 Biochemical and structural characterization of second-generation inhibitors targeting the SARS-CoV-2 3CL protease von Muczynski, Michael, Engel, Joseph, Amblard, Franck, Patel, Dharmeshkumar, Schinazi, Raymond, Kovari, Ladislau

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Approaches to hepatitis C treatment and cure using NS5A inhibitors von Kohler, James J, Nettles, James H, Amblard, Franck, Hurwitz, Selwyn J, Bassit, Leda, Stanton, Richard A, Ehteshami, Maryam, Schinazi, Raymond F

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Efficient synthesis of nucleoside aryloxy phosphoramidate prodrugs utilizing benzyloxycarbonyl protection von Cho, Jong Hyun, Amblard, Franck, Coats, Steven J., Schinazi, Raymond F.

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Comparison of anti-SARS-CoV-2 activity and intracellular metabolism of remdesivir and its parent nucleoside von Tao, Sijia, Zandi, Keivan, Bassit, Leda, Ong, Yee Tsuey, Verma, Kiran, Liu, Peng, Downs-Bowen, Jessica A., McBrayer, Tamara, LeCher, Julia C., Kohler, James J., Tedbury, Philip R., Kim, Baek, Amblard, Franck, Sarafianos, Stefan G., Schinazi, Raymond F.

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Diastereoselective Synthesis of 2′-Dihalopyrimidine Ribonucleoside Inhibitors of Hepatitis C Virus Replication von Zhou, Longhu, Zhang, Hongwang, Li, Chengwei, De Schutter, Coralie, Sari, Ozkan, Mengshetti, Seema, Zhou, Shaoman, Kasthuri, Mahesh, Coats, Steven J, Schinazi, Raymond F, Amblard, Franck

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