Lipase-catalyzed asymmetric hydrolysis of esters having remote chiral/prochiral centers von Hughes, David L, Bergan, J. J, Amato, J. S, Bhupathy, M, Leazer, J. L, McNamara, J. M, Sidler, D. R, Reider, P. J, Grabowski, E. J. J

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Synthesis of unsymmetrical dithioacetals: an efficient synthesis of a novel LTD4 antagonist, L-660,711 von McNamara, J. M, Leazer, J. L, Bhupathy, M, Amato, J. S, Reamer, R. A, Reider, P. J, Grabowski, E. J. J

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Enantioretentive alkylation of acyclic amino acids von Karady, Sandor, Amto, Joseph S., Weinstock, Leonard M.

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Tumor Microenvironment and Cellular Stress: Signaling, Metabolism, Imaging, and Therapeutic Targets von Koumenis, Constantinos, Hammond, Ester, Giaccia, Amato

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Enzymes and practical asymmetric synthesis von Bhupathy, M., Hughes, D. L., Amato, J. S., Bergan, J. J., Leazer, J. L., Lovelace, T. C., McNamara, J. M., Reamer, R. A., Sidler, D. R., Grabowski, E. J. J., Reider, P. J., Shinkai, I.

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Synthesis of chiral dithioacetals: a chemoenzymic synthesis of a novel LTD4 antagonist von Hughes, D. L, Bergan, J. J, Amato, J. S, Reider, P. J, Grabowski, E. J. J

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Process development for the production of the ( S)-acid precursor of a novel elastase inhibitor (L-694,458) through the lipase-catalyzed kinetic resolution of a β-lactam benzyl est... von Roberge, Christopher, Cvetovich, Raymond J., Amato, Joseph S., Pecore, Victor, Hartner, Frederick W., Greasham, Randolph, Chartrain, Michel

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Utilization of .alpha.,.beta.-unsaturated acids as Michael acceptors for the synthesis of thieno[2,3-b]thiopyrans von Ponticello, Gerald S, Freedman, Mark B, Habecker, Charles N, Holloway, M. Katharine, Amato, Joseph S, Conn, Robin S, Baldwin, John J

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Cyclization of electrochemically generated nitrogen radicals. : A novel synthesis of 11-substituted dibenzo[a,d]cycloheptenimine derivatives von Karady, Sandor, Corley, Edward G., Abramson, Newton L., Amato, Joseph S., Weinstock, Leonard M.

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An Efficient Synthesis of a Dual PPAR α/γ Agonist and the Formation of a Sterically Congested α-Aryloxyisobutyric Acid via a Bargellini Reaction von Cvetovich, Raymond J, Chung, John Y. L, Kress, Michael H, Amato, Joseph S, Matty, Louis, Weingarten, M. David, Tsay, Fuh-Rong, Li, Zhen, Zhou, George

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Acylimidazolides as Versatile Synthetic Intermediates for the Preparation of Sterically Congested Amides and Ketones: A Practical Synthesis of Proscar von Bhattacharya, A., Williams, J. M., Amato, J. S., Dolling, U.-H., Grabowski, E. J. J.

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Synthesis of 1-tert-Butyl-4-chloropiperidine:  Generation of an N-tert-Butyl Group by the Reaction of a Dimethyliminium Salt with Methylmagnesium Chloride von Amato, Joseph S, Chung, John Y. L, Cvetovich, Raymond J, Gong, Xiaoyi, McLaughlin, Mark, Reamer, Robert A

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A New Preparation of Chloromethyl Methyl Ether Free of Bis[chloromethyl] Ether von Amato, J. S., Karady, S., Sletzinger, M., Weinstock, L. M.

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An Asymmetric Synthesis of L-694,458, a Human Leukocyte Elastase Inhibitor, via Novel Enzyme Resolution of β-Lactam Esters von Cvetovich, Raymond J, Chartrain, Michel, Hartner, Frederick W, Roberge, Christopher, Amato, Joseph S, Grabowski, Edward J. J

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Acrylate as an Efficient Dimethylamine Trap for the Practical Synthesis of 1-tert-Butyl-4-piperidone via Transamination von Amato, Joseph S, Chung, John Y. L, Cvetovich, Raymond J, Reamer, Robert A, Zhao, Dalian, Zhou, George, Gong, Xiaoyi

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Conversion of imidoyl chlorides to imines. A new method for the acyl exchange and cleavage of amides von Karady, S., Amato, J.S., Weinstock, L.M., Sletzinger, M.

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High temperature reactions of benzene von Firestone, R.A., Amato, J.S.

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A Highly Convergent Synthesis of a Fibrinogen Receptor Antagonist von Hartner, Frederick W, Cvetovich, Raymond J, Tsay, Fuh-Rong, Amato, Joseph S, Pipik, Brenda, Grabowski, Edward J. J, Reider, Paul J

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Oxime Formation of 4''-epi-(Acetylamino)-5-oxo-4''-deoxy-avermectin B1 von Cvetovich, Raymond J, Leonard, William R, Amato, Joseph S, DiMichele, Lisa M, Reamer, Robert A, Shuman, Richard F, Grabowski, Edward J. J

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Annelation of aromatic oxo compounds von Karady, Sandor, Amato, Joseph S, Reamer, Robert A, Weinstock, Leonard M

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