Pd- and Ni-Based Systems for the Catalytic Borylation of Aryl (Pseudo)halides with B2(OH)4 von Munteanu, Charissa, Spiller, Taylor E, Qiu, Jun, DelMonte, Albert J, Wisniewski, Steven R, Simmons, Eric M, Frantz, Doug E

Volltext

A Metal-Free Reductive N‑Alkylation of Indoles with Aldehydes von Clanton, Nicholas A, Spiller, Taylor E, Ortiz, Eliezer, Gao, Zhinong, Rodriguez-Poirier, Juan Manuel, DelMonte, Albert J, Frantz, Doug E

Volltext

Mechanistic Studies of a Pd-Catalyzed Direct Arylation En Route to Beclabuvir: Dual Role of a Tetramethylammonium Cation and an Unusual Turnover-Limiting Step von Hang, Chao, Ramirez, Antonio, Chan, Collin, Hsiao, Yi, DelMonte, Albert J, Simmons, Eric M

Volltext

Direct Lewis Acid Catalyzed Conversion of Enantioenriched N‑Acyloxazolidinones to Chiral Esters, Amides, and Acids von Stevens, Jason M, Parra-Rivera, Ana Cristina, Dixon, Darryl D, Beutner, Gregory L, DelMonte, Albert J, Frantz, Doug E, Janey, Jacob M, Paulson, James, Talley, Michael R

Volltext

Reinvestigation of the Isotope Effects for the Claisen and Aromatic Claisen Rearrangements:  The Nature of the Claisen Transition States von Meyer, Matthew P, DelMonte, Albert J, Singleton, Daniel A

Volltext

Cerium(III) Chloride-Mediated Stereoselective Reduction of a 4‑Substituted Cyclohexanone Using NaBH4 von Maity, Prantik, Gujjar, Manjunath, Vellingiri, Raghukumar, Lakshminarasimhan, Thirumalai, DelMonte, Albert J, Young, Ian S, Eastgate, Martin D, Vaidyanathan, Rajappa

Volltext

The First Kilogram Synthesis of Beclabuvir, an HCV NS5B Polymerase Inhibitor von Bien, Jeffrey, Davulcu, Akin, DelMonte, Albert J, Fraunhoffer, Kenneth J, Gao, Zhinong, Hang, Chao, Hsiao, Yi, Hu, Wenhao, Katipally, Kishta, Littke, Adam, Pedro, Aghogho, Qiu, Yuping, Sandoval, Maria, Schild, Richard, Soltani, Michelle, Tedesco, Anthony, Vanyo, Dale, Vemishetti, Purushotham, Waltermire, Robert E

Volltext

Coupling-Condensation Strategy for the Convergent Synthesis of an Imidazole-Fused 2‑Aminoquinoline NLRP3 Agonist von Bi, Cong, Chadwick, James, Davies, Merrill L., DelMonte, Albert J., Geng, Peng, Glace, Andrew W., Green, Rebecca A., Gurak, John A., Haley, Matthew W., He, Brian L., Inankur, Bahar, Jamison, Christopher R., Joe, Candice L., Kolotuchin, Sergei, Lin, Dong, Lou, Sha, Nye, Jeffrey, Ortiz, Adrian, Purdum, Geoffrey E., Rosso, Victor W., Shah, Mansi, Simmons, Eric M., Stevens, Jason M., Strotman, Neil A., Tan, Yichen, Zhang, Ling

Volltext

The Process Development of Ravuconazole: An Efficient Multikilogram Scale Preparation of an Antifungal Agent von Pesti, Jaan, Chen, Chien-Kuang, Spangler, Lori, DelMonte, Albert J, Benoit, Serge, Berglund, Derek, Bien, Jeffrey, Brodfuehrer, Paul, Chan, Yeung, Corbett, Elisabeth, Costello, Carrie, DeMena, Paul, Discordia, Robert P, Doubleday, Wendel, Gao, Zhinong, Gingras, Stephane, Grosso, John, Haas, Oscar, Kacsur, David, Lai, Chiajen, Leung, Simon, Miller, Melanie, Muslehiddinoglu, Jale, Nguyen, Nina, Qiu, Jun, Olzog, Martina, Reiff, Emily, Thoraval, Dominique, Totleben, Michael, Vanyo, Dale, Vemishetti, Purushotham, Wasylak, John, Wei, Chenkou

Volltext

Pd- and Ni-Based Systems for the Catalytic Borylation of Aryl (Pseudo)halides with B 2 (OH) 4 von Munteanu, Charissa, Spiller, Taylor E, Qiu, Jun, DelMonte, Albert J, Wisniewski, Steven R, Simmons, Eric M, Frantz, Doug E

Volltext

Experimental and Theoretical Kinetic Isotope Effects for Asymmetric Dihydroxylation. Evidence Supporting a Rate-Limiting “(3 + 2)” Cycloaddition von DelMonte, Albert J, Haller, Jan, Houk, K. N, Sharpless, K. Barry, Singleton, Daniel A, Strassner, Thomas, Thomas, Allen A

Volltext

Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H2O2 von Beutner, Gregory L, Cohen, Benjamin M, DelMonte, Albert J, Dixon, Darryl D, Fraunhoffer, Kenneth J, Glace, Andrew W, Lo, Ehrlic, Stevens, Jason M, Vanyo, Dale, Wilbert, Christopher

Volltext

Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor von Fraunhoffer, Kenneth J, DelMonte, Albert J, Beutner, Gregory L, Bultman, Michael S, Camacho, Kathryn, Cohen, Benjamin, Dixon, Darryl D, Fan, Yu, Fanfair, Dayne, Freitag, Adam J, Glace, Andrew W, Gonzalez-Bobes, Francisco, Gujjar, Manjunath, Haley, Matthew W, Hickey, Matthew R, Ho, Jeanne, Iyer, Vidya, Maity, Prantik, Patel, Sunil, Rosso, Victor W, Schmidt, Michael A, Stevens, Jason M, Tan, Yichen, Wilbert, Christopher, Young, Ian S, Yu, Miao

Volltext

Kilogram Synthesis of a Selective Serotonin Reuptake Inhibitor von Anthes, Robert, Bello, Osagie, Benoit, Serge, Chen, Chien-Kuang, Corbett, Elisabeth, Corbett, Richard M, DelMonte, Albert J, Gingras, Stephane, Livingston, Robert, Sausker, Justin, Soumeillant, Maxime

Volltext

Safe Scale-up of an Oxygen-Releasing Cleavage of Evans Oxazolidinone with Hydrogen Peroxide von Glace, Andrew W, Cohen, Benjamin M, Dixon, Darryl D, Beutner, Gregory L, Vanyo, Dale, Akpinar, Fulya, Rosso, Victor, Fraunhoffer, Kenneth J, DelMonte, Albert J, Santana, Edgar, Wilbert, Christopher, Gallo, Frank, Bartels, William

Volltext

Kilogram Synthesis of a Second-Generation LFA-1/ICAM Inhibitor von DelMonte, Albert J, Fan, Yu, Girard, Kevin P, Jones, Gregory S, Waltermire, Robert E, Rosso, Victor, Wang, Xuebao

Volltext

Small Molecule Antagonist of Leukocyte Function Associated Antigen-1 (LFA-1): Structure−Activity Relationships Leading to the Identification of 6-((5S,9R)-9-(4-Cyanophenyl)-3-(3,5-... von Watterson, Scott H, Xiao, Zili, Dodd, Dharmpal S, Tortolani, David R, Vaccaro, Wayne, Potin, Dominique, Launay, Michele, Stetsko, Dawn K, Skala, Stacey, Davis, Patric M, Lee, Deborah, Yang, Xiaoxia, McIntyre, Kim W, Balimane, Praveen, Patel, Karishma, Yang, Zheng, Marathe, Punit, Kadiyala, Pathanjali, Tebben, Andrew J, Sheriff, Steven, Chang, ChiehYing Y, Ziemba, Theresa, Zhang, Huiping, Chen, Bang-Chi, DelMonte, Albert J, Aranibar, Nelly, McKinnon, Murray, Barrish, Joel C, Suchard, Suzanne J, Murali Dhar, T. G

Volltext

An Improved Synthesis of a Selective Serotonin Reuptake Inhibitor von Anthes, Robert, Benoit, Serge, Chen, Chien-Kuang, Corbett, Elisabeth A, Corbett, Richard M, DelMonte, Albert J, Gingras, Stephane, Livingston, Robert C, Pendri, Yadagiri, Sausker, Justin, Soumeillant, Maxime

Volltext

Kilogram Synthesis of a LFA-1/ICAM Inhibitor von DelMonte, Albert J, Waltermire, Robert E, Fan, Yu, McLeod, Douglas D, Gao, Zhinong, Gesenberg, Kirsten D, Girard, Kevin P, Rosingana, Miguel, Wang, Xuebao, Kuehne-Willmore, Jennifer, Braem, Alan D, Castoro, John A

Volltext

Development of a Scalable Negishi Cross-Coupling Process for the Preparation of 2-Chloro-5-(1-(tetrahydro-2 H -pyran-2-yl)-1 H -pyrazol-5-yl)aniline von Joe, Candice L., Inankur, Bahar, Chadwick, James, Lou, Sha, Nye, Jeffrey, Strotman, Neil A., DelMonte, Albert J.

Volltext