Isocyanide-based multicomponent reactions in drug discovery von Akritopoulou-Zanze, Irini

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The Use of Three-Dimensional Shape and Electrostatic Similarity Searching in the Identification of a Melanin-Concentrating Hormone Receptor 1 Antagonist von Muchmore, Steven W., Souers, Andrew J., Akritopoulou-Zanze, Irini

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Kinase-targeted libraries: The design and synthesis of novel, potent, and selective kinase inhibitors von Akritopoulou-Zanze, Irini, Hajduk, Philip J.

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Small molecule library synthesis using segmented flow von Thompson, Christina M, Poole, Jennifer L, Cross, Jeffrey L, Akritopoulou-Zanze, Irini, Djuric, Stevan W

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Synthesis of substituted 3,4-dihydroquinolin-2(1 H)-one derivatives by sequential Ugi/acrylanilide [6π]-photocyclizations von Akritopoulou-Zanze, Irini, Whitehead, Alan, Waters, Jan E., Henry, Rodger F., Djuric, Stevan W.

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Configuration of heptopyranoside and heptofuranoside side chains: 2-anthroate, a powerful chromophore for exciton coupled CD von Akritopoulou-Zanze, Irini, Nakanishi, Koji, Stepowska, Halszka, Grzeszczyk, Barbara, Zamojski, Aleksander, Berova, Nina

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Theoretical and experimental CD of conformationally flexible complex molecules-application to ouabain pentanaphthoate and analogs von Dong, Jian-Guo, Guo, Jinsong, Akritopoulou-Zanze, Irini, Kawamura, Akira, Nakanishi, Koji, Berova, Nina

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A versatile synthesis of fused triazolo derivatives by sequential Ugi/alkyne-azide cycloaddition reactions von Akritopoulou-Zanze, Irini, Gracias, Vijaya, Djuric, Stevan W.

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De Novo Design, Synthesis, and Biological Evaluation of 3,4-Disubstituted Pyrrolidine Sulfonamides as Potent and Selective Glycine Transporter 1 Competitive Inhibitors von Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Li, Huanqiu, Lao, Yanbin, Amberg, Willi, Behl, Berthold, Akritopoulou-Zanze, Irini, Dietrich, Justin, Lange, Udo E. W, Pohlki, Frauke, Hoft, Carolin, Hornberger, Wilfried, Djuric, Stevan W, Sydor, Jens, Mezler, Mario, Relo, Ana Lucia, Vasudevan, Anil

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Discovery of Novel Aminotetralines and Aminochromanes as Selective and Competitive Glycine Transporter 1 (GlyT1) Inhibitors von Amberg, Willi, Lange, Udo E. W, Ochse, Michael, Pohlki, Frauke, Behl, Berthold, Relo, Ana Lucia, Hornberger, Wilfried, Hoft, Carolin, Mezler, Mario, Sydor, Jens, Wang, Ying, Zhao, Hongyu, Brewer, Jason T, Dietrich, Justin, Li, Huanqiu, Akritopoulou-Zanze, Irini, Lao, Yanbin, Hannick, Steven M, Ku, Yi-Yin, Vasudevan, Anil

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Synthesis of substituted fused pyridines, pyrazines and pyrimidines by sequential Ugi/inverse electron demand Diels–Alder transformations von Akritopoulou-Zanze, Irini, Wang, Ying, Zhao, Hongyu, Djuric, Stevan W.

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Concise Construction of Novel Bridged Bicyclic Lactams by Sequenced Ugi/RCM/Heck Reactions von Ribelin, Timothy P, Judd, Andrew S, Akritopoulou-Zanze, Irini, Henry, Rodger F, Cross, Jeffrey L, Whittern, David N, Djuric, Stevan W

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ChemInform Abstract: Applications of Isocyanides in the Synthesis of Heterocycles von Akritopoulou-Zanze, Irini

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Scaffold oriented synthesis. Part 4: Design, synthesis and biological evaluation of novel 5-substituted indazoles as potent and selective kinase inhibitors employing heterocycle fo... von Akritopoulou-Zanze, Irini, Wakefield, Brian D., Gasiecki, Alan, Kalvin, Douglas, Johnson, Eric F., Kovar, Peter, Djuric, Stevan W.

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Scaffold oriented synthesis. Part 3: Design, synthesis and biological evaluation of novel 5-substituted indazoles as potent and selective kinase inhibitors employing [2+3] cycloadd... von Akritopoulou-Zanze, Irini, Wakefield, Brian D., Gasiecki, Alan, Kalvin, Douglas, Johnson, Eric F., Kovar, Peter, Djuric, Stevan W.

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ChemInform Abstract: Applications of MCR-Derived Heterocycles in Drug Discovery von Akritopoulou-Zanze, Irini, Djuric, Stevan W.

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Synthesis of Novel and Uniquely Shaped 3-Azabicyclo[4.2.0]octan-4-one Derivatives by Sequential Ugi/[2+2] Ene−Enone Photocycloadditions von Akritopoulou-Zanze, Irini, Whitehead, Alan, Waters, Jan E, Henry, Rodger F, Djuric, Stevan W

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Synthesis of novel fused isoxazoles and isoxazolines by sequential Ugi/INOC reactions von Akritopoulou-Zanze, Irini, Gracias, Vijaya, Moore, Joel D, Djuric, Stevan W

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Topography-biased compound library design: the shape of things to come? von Akritopoulou-Zanze, Irini, Metz, James T., Djuric, Stevan W.

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An expedient route to diaza-spirocycles utilizing a sequential multicomponent α-aminoallylation/ring-closing metathesis strategy von Gracias, Vijaya, Gasiecki, Alan F., Moore, Joel D., Akritopoulou-Zanze, Irini, Djuric, Stevan W.

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