Protease Inhibitors:  Current Status and Future Prospects von Leung, Donmienne, Abbenante, Giovanni, Fairlie, David P

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Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency von Harrison, Rosemary S., Shepherd, Nicholas E., Hoang, Huy N., Ruiz-Gómez, Gloria, Hill, Timothy A., Driver, Russell W., Desai, Vishal S., Young, Paul R., Abbenante, Giovanni, Fairlie, David P., Klibanov, Alexander M.

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Isolation and Characterization of a Cone Snail Protease with Homology to CRISP Proteins of the Pathogenesis-related Protein Superfamily von Milne, Trudy J., Abbenante, Giovanni, Tyndall, Joel D.A., Halliday, Judy, Lewis, Richard J.

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Activity of Recombinant Dengue 2 Virus NS3 Protease in the Presence of a Truncated NS2B Co-factor, Small Peptide Substrates, and Inhibitors von Leung, Donmienne, Schroder, Kate, White, Helen, Fang, Ning-Xia, Stoermer, Martin J., Abbenante, Giovanni, Martin, Jennifer L., Young, Paul R., Fairlie, David P.

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Novel Helix-Constrained Nociceptin Derivatives Are Potent Agonists and Antagonists of ERK Phosphorylation and Thermal Analgesia in Mice von Harrison, Rosemary S, Ruiz-Gómez, Gloria, Hill, Timothy A, Chow, Shiao Y, Shepherd, Nicholas E, Lohman, Rink-Jan, Abbenante, Giovanni, Hoang, Huy N, Fairlie, David P

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Selective Hexapeptide Agonists and Antagonists for Human Complement C3a Receptor von Scully, Conor C. G, Blakeney, Jade S, Singh, Ranee, Hoang, Huy N, Abbenante, Giovanni, Reid, Robert C, Fairlie, David P

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Profiling the Enzymatic Properties and Inhibition of Human Complement Factor B von Le, Giang Thanh, Abbenante, Giovanni, Fairlie, David P.

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Potent Cyclic Antagonists of the Complement C5a Receptor on Human Polymorphonuclear Leukocytes. Relationships between Structures and Activity von March, Darren R, Proctor, Lavinia M, Stoermer, Martin J, Sbaglia, Robert, Abbenante, Giovanni, Reid, Robert C, Woodruff, Trent M, Wadi, Khemar, Paczkowski, Natalii, Tyndall, Joel D A, Taylor, Stephen M, Fairlie, David P

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Cleavage of hemoglobin by hookworm cathepsin D aspartic proteases and its potential contribution to host specificity von Williamson, Angela L., Brindley, Paul J., Abbenante, Giovanni, Prociv, Paul, Berry, Colin, Girdwood, Karen, Pritchard, David I., Fairlie, David P., Hotez, Peter J., Dalton, John P., Loukas, Alex

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Single Turn Peptide Alpha Helices with Exceptional Stability in Water von Shepherd, Nicholas E, Hoang, Huy N, Abbenante, Giovanni, Fairlie, David P

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Over One Hundred Peptide-Activated G Protein-Coupled Receptors Recognize Ligands with Turn Structure von Tyndall, Joel D. A, Pfeiffer, Bernhard, Abbenante, Giovanni, Fairlie, David P

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Twists or turns: stabilising alpha beta turns in tetrapeptides von Hoang, Huy N, Hill, Timothy A, Ruiz-Gómez, Gloria, Diness, Frederik, Mason, Jody M, Wu, Chongyang, Abbenante, Giovanni, Shepherd, Nicholas E, Fairlie, David P

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Correction: Twists or turns: stabilising alpha vs. beta turns in tetrapeptides von Hoang, Huy N., Hill, Timothy A., Ruiz-Gómez, Gloria, Diness, Frederik, Mason, Jody M., Wu, Chongyang, Abbenante, Giovanni, Shepherd, Nicholas E., Fairlie, David P.

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Twists or turns: stabilising alpha vs. beta turns in tetrapeptides von Hoang, Huy N, Hill, Timothy A, Ruiz-Gómez, Gloria, Diness, Frederik, Mason, Jody M, Wu, Chongyang, Abbenante, Giovanni, Shepherd, Nicholas E, Fairlie, David P

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Downsizing the BAD BH3 peptide to small constrained α-helices with improved ligand efficiency von Shepperd, Nicholas E., Harrison, Rosemary S., Ruiz-Gomez, Gloria, Abbenante, Giovanni, Mason, Jody M., Fairlie, David P.

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Downsizing the BAD BH3 peptide to small constrained α-helices with improved ligand efficiencyElectronic supplementary information (ESI) available: Peptide. See DOI: 10.1039/C6OB021... von Shepherd, Nicholas E, Harrison, Rosemary S, Ruiz-Gomez, Gloria, Abbenante, Giovanni, Mason, Jody M, Fairlie, David P

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Update 1 of: Over One Hundred Peptide-Activated G Protein-Coupled Receptors Recognize Ligands with Turn Structure von Ruiz-Gómez, Gloria, Tyndall, Joel D. A, Pfeiffer, Bernhard, Abbenante, Giovanni, Fairlie, David P

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Downsizing the BAD BH3 peptide to small constrained α-helices with improved ligand efficiency von Shepherd, Nicholas E, Harrison, Rosemary S, Ruiz-Gomez, Gloria, Abbenante, Giovanni, Mason, Jody M, Fairlie, David P

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Left- and Right-Handed Alpha-Helical Turns in Homo- and Hetero-Chiral Helical Scaffolds von Shepherd, Nicholas E, Hoang, Huy N, Abbenante, Giovanni, Fairlie, David P

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Correction: Downsizing the BAD BH3 peptide to small constrained α-helices with improved ligand efficiency von Shepherd, Nicholas E, Harrison, Rosemary S, Ruiz-Gomez, Gloria, Abbenante, Giovanni, Mason, Jody M, Fairlie, David P

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