Potency variation of small-molecule chymase inhibitors across species von Kervinen, Jukka, Crysler, Carl, Bayoumy, Shariff, Abad, Marta C., Spurlino, John, Deckman, Ingrid, Greco, Michael N., Maryanoff, Bruce E., de Garavilla, Lawrence

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Identification of Diaryl Ether-Based Ligands for Estrogen-Related Receptor α as Potential Antidiabetic Agents von Patch, Raymond J, Searle, Lily L, Kim, Alexander J, De, Debyendu, Zhu, Xizhen, Askari, Hossein B, O’Neill, John C, Abad, Marta C, Rentzeperis, Dionisios, Liu, Jianying, Kemmerer, Michael, Lin, Ling, Kasturi, Jyotsna, Geisler, John G, Lenhard, James M, Player, Mark R, Gaul, Micheal D

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4-Amino-6-arylamino-pyrimidine-5-carbaldehyde hydrazones as potent ErbB-2/EGFR dual kinase inhibitors von Xu, Guozhang, Abad, Marta C., Connolly, Peter J., Neeper, Michael P., Struble, Geoffrey T., Springer, Barry A., Emanuel, Stuart L., Pandey, Niranjan, Gruninger, Robert H., Adams, Mary, Moreno-Mazza, Sandra, Fuentes-Pesquera, Angel R., Middleton, Steven A.

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Optimization of a pyrazole hit from FBDD into a novel series of indazoles as ketohexokinase inhibitors von Zhang, Xuqing, Song, Fengbing, Kuo, Gee-Hong, Xiang, Amy, Gibbs, Alan C., Abad, Marta C., Sun, Weimei, Kuo, Lawrence C., Sui, Zhihua

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Structural determination of estrogen-related receptor γ in the presence of phenol derivative compounds von Abad, Marta C., Askari, Hossein, O’Neill, John, Klinger, Alexandra L., Milligan, Cynthia, Lewandowski, Frank, Springer, Barry, Spurlino, John, Rentzeperis, Dionisios

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Electron Density Guided Fragment-Based Lead Discovery of Ketohexokinase Inhibitors von Gibbs, Alan C, Abad, Marta C, Zhang, Xuqing, Tounge, Brett A, Lewandowski, Francis A, Struble, Geoffrey T, Sun, Weimei, Sui, Zhihua, Kuo, Lawrence C

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The X-ray crystallographic structure of Escherichia coli branching enzyme von Abad, Marta C, Binderup, Kim, Rios-Steiner, Jorge, Arni, Raghuvir K, Preiss, Jack, Geiger, James H

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7-Fluoroindazoles as Potent and Selective Inhibitors of Factor Xa von Lee, Yu-Kai, Parks, Daniel J, Lu, Tianbao, Thieu, Tho V, Markotan, Thomas, Pan, Wenxi, McComsey, David F, Milkiewicz, Karen L, Crysler, Carl S, Ninan, Nisha, Abad, Marta C, Giardino, Edward C, Maryanoff, Bruce E, Damiano, Bruce P, Player, Mark R

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Discovery of novel 4-amino-6-arylaminopyrimidine-5-carbaldehyde oximes as dual inhibitors of EGFR and ErbB-2 protein tyrosine kinases von Xu, Guozhang, Searle, Lily Lee, Hughes, Terry V., Beck, Amanda K., Connolly, Peter J., Abad, Marta C., Neeper, Michael P., Struble, Geoffrey T., Springer, Barry A., Emanuel, Stuart L., Gruninger, Robert H., Pandey, Niranjan, Adams, Mary, Moreno-Mazza, Sandra, Fuentes-Pesquera, Angel R., Middleton, Steven A., Greenberger, Lee M.

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Inhibitors of Ketohexokinase: Discovery of Pyrimidinopyrimidines with Specific Substitution that Complements the ATP-Binding Site von Maryanoff, Bruce E, O'Neill, John C, McComsey, David F, Yabut, Stephen C, Luci, Diane K, Jordan, Alfonzo D, Masucci, John A, Jones, William J, Abad, Marta C, Gibbs, Alan C, Petrounia, Ioanna

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Novel tetrahydroisoquinolines are histamine H3 antagonists and serotonin reuptake inhibitors von LETAVIC, Michael A, KEITH, John M, WILSON, Sandy J, MILLER, Kirsten L, LORD, Brian, MCALLISTER, Heather M, TOGNARELLI, D. J, JIEJUN WU, ABAD, Marta C, SCHUBERT, Carsten, LOVENBERG, Timothy W, CARRUTHERS, Nicholas I, JABLONOWSKI, Jill A, STOCKING, Emily M, GOMEZ, Leslie A, LY, Kiev S, MILLER, Jennifer M, BARBIER, Ann J, BONAVENTURE, Pascal, BOGGS, Jamin D

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Discovery, SAR, and X-ray structure of novel biaryl-based dipeptidyl peptidase IV inhibitors von Qiao, Lei, Baumann, Christian A., Crysler, Carl S., Ninan, Nisha S., Abad, Marta C., Spurlino, John C., DesJarlais, Renee L., Kervinen, Jukka, Neeper, Mike P., Bayoumy, Shariff S., Williams, Robyn, Deckman, Ingrid C., Dasgupta, Malini, Reed, Rolanda L., Huebert, Norman D., Tomczuk, Bruce E., Moriarty, Kevin J.

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Correction to Inhibitors of Ketohexokinase: Discovery of Pyrimidinopyrimidines with Specific Substitution that Complements the ATP-Binding Site von Maryanoff, Bruce E, O'Neill, John C, McComsey, David F, Yabut, Stephen C, Luci, Diane K, Jordan, Alfonzo D, Masucci, John A, Jones, William J, Abad, Marta C, Gibbs, Alan C, Petrounia, Ioanna

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The X-ray Crystallographic Structure of the Angiogenesis Inhibitor Angiostatin von Abad, Marta C., Arni, R.K., Grella, Davida K., Castellino, Francis J., Tulinsky, Alexander, Geiger, James H.

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Electron Density Guided Fragment-Based Drug Design—A Lead Generation Example von Abad, Marta C., Gibbs, Alan C., Zhang, Xuqing

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The X-ray Crystallographic Structure ofEscherichia coli Branching Enzyme von Marta C. Abad, Kim Binderup, Jorge Rios-Steiner, Raghuvir K. Arni, Jack Preiss, James H. Geiger

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Crystallization and preliminary X-ray diffraction studies of human angiostatin von Abad, Marta C., Geiger, James

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Crystallization and preliminary X-ray diffraction studies of Escherichia coli branching enzyme von Abad, Marta C., Binderup, Kim, Preiss, Jack, Geiger, James H.

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Novel tetrahydroisoquinolines are histamine H 3 antagonists and serotonin reuptake inhibitors von Letavic, Michael A., Keith, John M., Jablonowski, Jill A., Stocking, Emily M., Gomez, Leslie A., Ly, Kiev S., Miller, Jennifer M., Barbier, Ann J., Bonaventure, Pascal, Boggs, Jamin D., Wilson, Sandy J., Miller, Kirsten L., Lord, Brian, McAllister, Heather M., Tognarelli, D.J., Wu, Jiejun, Abad, Marta C., Schubert, Carsten, Lovenberg, Timothy W., Carruthers, Nicholas I.

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Structural determination of estrogen-related receptor '>/ in the presence of phenol derivative compounds von ABAD, Marta C, ASKARI, Hossein, O'NEILL, John, KLINGER, Alexandra L, MILLIGAN, Cynthia, LEWANDOWSKI, Frank, SPRINGER, Barry, SPURLINO, John, RENTZEPERIS, Dionisios

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