Synthesis and structural characterization of charybdotoxin, a potent peptidyl inhibitor of the high conductance Ca2(+)-activated K+ channel von Sugg, E.E., Garcia, M.L., Reuben, J.P., Patchett, A.A., Kaczorowski, G.J.

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Synthesis of N2-[(S)-1-Carboxy-3-phenylpropyl]-L-lysyl-L-proline (Lisinopril) von Wu, M.T., Douglas, A.W., Ondeyka, D.L., Payne, L.G., Ikeler, T.J., Joshua, H., Patchett, A.A.

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Design of a selective insulin receptor tyrosine kinase inhibitor and its effect on glucose uptake and metabolism in intact cells von Saperstein, Richard, Vicario, Pasquale P, Strout, H. Vincent, Brady, Edward, Slater, Eve E, Greenlee, William J, Ondeyka, Debra L, Patchett, Arthur A, Hangauer, David G

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Mechanism-based inactivation of alanine racemase by 3-halovinylglycines von THORNBERRY, N. A, BULL, H. G, TAUB, D, WILSON, K. E, GIMENEZ-GALLEGO, G, ROSEGAY, A, SODERMAN, D. D, PATCHETT, A. A

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Sulfones as peptide bond isosteres von Rivero, R.A., Greenlee, W.J., Patchett, A.A.

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AT1 selective angiotensin II antagonists with phenoxyphenylacetic acid as a biphenyl replacement part I von Fitch, K.J., Walsh, T.F., Patchett, A.A., Chang, R.S.L., Siegl, P.K.S., Faust, K.A., Chen, T.-B., Lotti, V.J., Kivlighn, S.D., Zingaro, G.J., Greenlee, W.J.

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Triazolinones as nonpeptide angiotensin II antagonists. 2. discovery of a potent and orally active triazolinone acylsulfonamide von Chang, L.L., Ashton, W.T., Flanagan, K.L., Naylor, E.M., Chakravarty, P.K., Patchett, A.A., Greenlee, W.J., Bendesky, R.J., Chen, T.-B., Faust, K.A., Kling, P.J., Schaffer, L.W., Schorn, T.W., Zingaro, G.J., Chang, R.S.L., Lotti, V.J., Kivlighn, S.D., Siegl, P.K.S.

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AT 1 selective angiotensin II antagonists with phenoxyphenylacetic acid as a biphenyl replacement part I von Fitch, K.J., Walsh, T.F., Patchett, A.A., Chang, R.S.L., Siegl, P.K.S., Faust, K.A., Chen, T.-B., Lotti, V.J., Kivlighn, S.D., Zingaro, G.J., Greenlee, W.J.

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Syntheses of α-ethynyl-3, 4-dihydroxyphenylalanine and α-vinyl-3, 4-dihydroxyphenylalanine von Taub, D., Patchett, A.A.

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Azapeptides: A new class of angiotensin-converting enzyme inhibitors von Greenlee, W.J., Thorsett, E.D., Springer, J.P., Patchett, A.A., Ulm, E.H., Vassil, T.C.

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Dipeptide mimics. Conformationally restricted inhibitors of angiotensin-converting enzyme von Thorsett, E.D., Harris, E.E., Aster, S., Peterson, E.R., Taub, D., Patchett, A.A., Ulm, E.H., Vassil, T.C.

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Benzolactams. A new class of converting enzyme inhibitors von Parsons, W.H., Davidson, J.L., Taub, D., Aster, S.D., Thorsett, E.D., Patchett, A.A., Ulm, E.H., Lamont, B.I.

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A general synthesis of α-vinyl-α-amino acids von Greenlee, W.J., Taub, D., Patchett, A.A.

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A potent nonpeptide cholecystokinin antagonist selective for peripheral tissues isolated from Aspergillus alliaceus von Chang, R.S.L, Lotti, V.J, Monaghan, R.L, Birnbaum, J, Stapley, E.O, Goetz, M.A, Albers-Schonberg, G, Patchett, A.A, Liesch, J.M, Hensens, O.D

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Halogenation of C16-macrolide antibiotics 17-haloleucomycins (A3) von Girotra, N.N., Patchett, A.A., Wendler, N.L.

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Preparation and hydrolysis of phenylbisdialkylaminocyclopropenium cations von Wu, M.T., Taub, D., Patchett, A.A.

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Halogenation of C 16-macrolide antibiotics 17-haloleucomycins (A 3) von Girotra, N.N., Patchett, A.A., Wendler, N.L.

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GR74785 von E.E HARRIS, A.A PATCHETT, E.D THORSETT, W. J. GREENLEE

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Addition of dimethyloxosulfonium methylide to steroidal 4,6-dien-3-ones: Steric effects on the formation of the 6,7-methylene group von Arth, G.E., Reynolds, G.F., Rasmusson, G.H., Chen, A., Patchett, A.A.

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Anthelmintic 2-Arylhydrazino- and 2-Arylazo-2-thiazolines von Wu, M.T., Waksmunski, F.S., Hoff, D.R., Fisher, M.H., Egerton, J.R., Patchett, A.A.

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