Kinase Screening and Profiling: Methods and Protocols von Zegzouti, Hicham, Goueli, Said A

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HotSpot: A Novel Methyltransferase Assay Platform for Drug Screening and Discovery von Horiuchi, Kurumi Y, Eason, Mia M, Ma, Haiching

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Rapid Identification of Protein Kinase Phosphorylation Site Motifs Using Combinatorial Peptide Libraries von Miller, Chad J., Turk, Benjamin E.

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A High-Throughput Radiometric Kinase Assay von Duong-Ly, Krisna C., Peterson, Jeffrey R.

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Bioluminescence Methods for Assaying Kinases in Quantitative High-Throughput Screening (qHTS) Format Applied to Yes1 Tyrosine Kinase, Glucokinase, and PI5P4Kα Lipid Kinase von Davis, Mindy I., Auld, Douglas S., Inglese, James

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From Enzyme to Whole Blood: Sequential Screening Procedure for Identification and Evaluation of p38 MAPK Inhibitors von Bauer, Silke M., Kubiak, Jakub M., Rothbauer, Ulrich, Laufer, Stefan

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Monitoring Protein Kinase Expression and Phosphorylation in Cell Lysates with Antibody Microarrays von Zhang, Hong, Shi, Xiaoqing, Pelech, Steven

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Determination of the Substrate Specificity of Protein Kinases with Peptide Micro- and Macroarrays von Lai, Shenshen, Winkler, Dirk F. H., Zhang, Hong, Pelech, Steven

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A High-Content Assay to Screen for Modulators of EGFR Function von Antczak, Christophe, Djaballah, Hakim

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HTRF Kinase Assay Development and Methods in Inhibitor Characterization von Jia, Yong, Manuia, Mari, Juarez, Jose

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Genetically Encoded Fluorescent Indicators to Visualize Protein Phosphorylation in Living Cells von Sato, Moritoshi, Umezawa, Yoshio

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Application of Eukaryotic Elongation Factor-2 Kinase (eEF-2K) for Cancer Therapy: Expression, Purification, and High-Throughput Inhibitor Screening von Tavares, Clint D. J., Devkota, Ashwini K., Dalby, Kevin N., Cho, Eun Jeong

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Characterization of an Engineered Src Kinase to Study Src Signaling and Biology von Gentry, Leanna R., Karginov, Andrei V., Hahn, Klaus M., Der, Channing J.

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Measuring Activity of Phosphoinositide Lipid Kinases Using a Bioluminescent ADP-Detecting Assay von Tai, Andrew W., Vidugiriene, Jolanta

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Screening One-Bead-One-Compound Peptide Libraries for Optimal Kinase Substrates von Trinh, Thi B., Pei, Dehua

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Using Bioluminescent Kinase Profiling Strips to Identify Kinase Inhibitor Selectivity and Promiscuity von Zegzouti, Hicham, Hennek, Jacquelyn, Goueli, Said A.

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Recombinant Kinase Production and Fragment Screening by NMR Spectroscopy von Han, Byeonggu, Ahn, Hee-Chul

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Dihydroartemisinin inhibits prostate cancer via JARID2/miR-7/miR-34a-dependent downregulation of Axl von Paccez, Juliano D., Duncan, Kristal, Sekar, Durairaj, Correa, Ricardo G., Wang, Yihong, Gu, Xuesong, Bashin, Manoj, Chibale, Kelly, Libermann, Towia A., Zerbini, Luiz F.

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Identification of Novel GSK-3β Hits Using Competitive Biophysical Assays von Balboni, Beatrice, Tripathi, Shailesh Kumar, Veronesi, Marina, Russo, Debora, Penna, Ilaria, Giabbai, Barbara, Bandiera, Tiziano, Storici, Paola, Girotto, Stefania, Cavalli, Andrea

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New 3-Aryl-2-(2-thienyl)acrylonitriles with High Activity Against Hepatoma Cells von Schaller, Eva, Ma, Andi, Gosch, Lisa Chiara, Klefenz, Adrian, Schaller, David, Goehringer, Nils, Kaps, Leonard, Schuppan, Detlef, Volkamer, Andrea, Schobert, Rainer, Biersack, Bernhard, Nitzsche, Bianca, Höpfner, Michael

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